“receptor”的搜索结果

产品 301 到 350 共 1701个

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  1. Sarmazenil

    Catalog No. A20487
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    benzodiazepine receptor antagonist
    Sarmazenil is a benzodiazepine receptor antagonist. 了解更多
  2. Tiodazosin

    Catalog No. A20463
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    ostsynaptic alpha adrenergic receptor antagonist
    Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist. 了解更多
  3. Org41841

    Catalog No. A20396
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    LHCGR/TSHR agonist
    Org41841 is a partial agonist of both luteinizing hormone/chorionic gonadotropin receptor (LHCGR) and thyroid-stimulating hormone receptor (TSHR) with EC50s of 0.2 and 7.7 μM, respectively. 了解更多
  4. Pirolate

    Catalog No. A20363
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    histamine H1 receptor
    Pirolate is a histamine H1 receptor. 了解更多
  5. JYL 1421

    Catalog No. A20350
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    TRPV1 receptor antagonist
    JYL 1421 is a TRPV1 receptor antagonist, with an IC50 of 8 nM. 了解更多
  6. (+)-Dihydrexidine hydrochloride

    Catalog No. A20339
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    dopamine D1 receptor agonist
    (+)-Dihydrexidine hydrochloride ((+)-DAR-0100 hydrochloride) is a dopamine D1 receptor agonist with an EC50 of 72± 21 nM. 了解更多
  7. L162389

    Catalog No. A20297
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    angiotensin AT1 receptor antagonist
    L162389 is a potent antagonist of angiotensin AT1 receptor with Ki of 28 nM. 了解更多
  8. Abaperidone

    Catalog No. A20286
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    5-HT2A/dopamine D2 antagonist
    Abaperidone is a potent antagonist of 5-HT2A?receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM. 了解更多
  9. MRZ 2-514

    Catalog No. A20277
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    NMDA receptor (glycineB) antagonist
    MRZ 2-514 is an antagonist of the strychnine-insensitive modulatory site of the NMDA receptor (glycineB), with Ki of 33 μM. 了解更多
  10. Lidanserin

    Catalog No. A20266
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    5-HT2A/α1-adrenergic receptor antagonist
    Lidanserin is a drug which acts as a combined 5-HT2A and α1-adrenergic receptor antagonist. 了解更多
  11. Spirendolol

    Catalog No. A20254
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    β adrenergic receptor antagonist
    Spirendolol is a β adrenergic receptor antagonist. 了解更多
  12. Foscarbidopa

    Catalog No. A20221
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    dopamine receptor agonist
    Foscarbidopa (Carbidopa 4??-monophosphate) is a prodrug of Carbidopa, acts as a dopamine receptor agonist. 了解更多
  13. Foslevodopa

    Catalog No. A20212
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    dopamine receptor agonist
    Foslevodopa is a dopamine receptor agonist. 了解更多
  14. ALB-127158(a)

    Catalog No. A20211
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    MCH1 receptor antagonist
    ALB-127158(a) is a potent and selective melanin concentrating hormone 1 (MCH1) receptor antagonist. 了解更多
  15. NK-1 Antagonist 1

    Catalog No. A20201
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    NK-1 receptor antagonist
    NK-1 Antagonist 1 (Rolapitant intermediate) is an antagonist of NK-1 receptor, used in the research of NK-1 related diseases and conditions such as cough, overactive bladder, alcohol dependency and depression. 了解更多
  16. Taminadenant

    Catalog No. A20190
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    adenosine receptor antagonist
    Taminadenant is an antagonist of adenosine receptor. 了解更多
  17. Wy 49051

    Catalog No. A20176
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    H1 receptor antagonist
    Wy 49051 is a potent, orally active H1 receptor antagonist, with IC50 of 44 nM. 了解更多
  18. FK1052 hydrochloride

    Catalog No. A20164
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    5-HT3 /5-HT4 receptor dual antagonist
    FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist. 了解更多
  19. Saredutant

    Catalog No. A20096
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    NK2 receptor antagonist
    Saredutant is a selective NK2 receptor antagonist. 了解更多
  20. Apimostinel

    Catalog No. A20075
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    NMDA receptor partial agonist
    Apimostinel (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist. 了解更多
  21. AR-A 2

    Catalog No. A20051
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    5-HT1B receptor antagonist
    AR-A 2 is a selective 5-HT1B receptor antagonist. 了解更多
  22. FITM

    Catalog No. A20047
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    mGlu1 receptor modulator
    FITM is a negative allosteric modulator of mGlu1 receptor with a Ki of 2.5 nM. 了解更多
  23. AP5

    Catalog No. A20042
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    AP5 exhibits potent and selective agonism for the GPR40 receptor with positive allosteric modulation of endogenous ligands (AgoPAM). AP5 demonstrates a rat hIP1 EC50 of 0.49±0.28 nM against the GPR40 receptor. 了解更多
  24. Pargolol hydrochloride

    Catalog No. A20035
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    β adrenergic receptor antagonist
    Pargolol hydrochloride is a β adrenergic receptor antagonist. 了解更多
  25. YK11

    Catalog No. A20033
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    Androgen receptor partial agonist
    YK11 is a partial agonist of androgen receptor, with osteogenic activity. 了解更多
  26. MK-8318

    Catalog No. A20030
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    CRTh2 receptor antagonist
    MK-8318 is a potent and selective CRTh2 receptor antagonist with a Ki of 5.0 nM. 了解更多
  27. ODM-204

    Catalog No. A20025
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    androgen receptor/CYP17A1 dual inhibitor
    ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme, with IC50s of 80?nM and 22 nM, respectively. 了解更多
  28. N6-(2-Phenylethyl)adenosine

    Catalog No. A20011
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    A1 adenosine receptor agonist
    N6-(2-Phenylethyl)adenosine is a selective A1 adenosine receptor agonist. 了解更多
  29. D4-abiraterone

    Catalog No. A19987
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    androgen receptor antagonist
    D4-abiraterone is a major metabolite of abiraterone. D4-abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid-5a-reductase (SRD5A) and also an antagonist of androgen receptor. 了解更多
  30. Sulamserod

    Catalog No. A19984
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    5-HT4 receptor antagonist
    Sulamserod is a 5-HT4 receptor antagonist, with antiarrhythmic activities. 了解更多
  31. H3B-5942

    Catalog No. A19960
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    estrogen receptor covalent antagonist
    H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively. 了解更多
  32. 1,4-Chrysenequinone

    Catalog No. A19937
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    aryl hydrocarbon receptor activator
    1,4-Chrysenequinone, a polycyclic aromatic quinone, acts as an activator of aryl hydrocarbon receptor (AhR). 了解更多
  33. GC 14

    Catalog No. A19928
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    thyroid hormone receptor antagonist
    GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 35 nM and 200 nM for hTRβ and hTRα, respectively. 了解更多
  34. N6-Ethyladenosine

    Catalog No. A19918
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    Adenosine receptor agonist
    N6-Ethyladenosine is an adenosine derivative, acts as a Adenosine receptor agonist, with Kis of 4.9 and 4.7 nM for hA1AR and hA3AR, respectively. 了解更多
  35. YM-58790

    Catalog No. A19917
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    M3 muscarinic receptor antagonist
    YM-58790 is a potent antagonist of M3 muscarinic receptor, with Ki of 15 nM. 了解更多
  36. Leelamine hydrochloride

    Catalog No. A19910
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    CB1 agonist
    Leelamine hydrochloride is a tricyclic diterpene molecule that is extracted from the bark of pine trees. Leelamine hydrochloride is a cannabinoid receptor type 1 (CB1) agonist and a inhibitor of SREBP1-regulated fatty acid/lipid synthesis in prostate cancer cells that is not affected by androgen receptor status. 了解更多
  37. (Z)-Guggulsterone

    Catalog No. A19901
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    farnesoid X receptor antagonist
    (Z)-Guggulsterone is a phytosteroid found in the resin of the guggul plant, Commiphora mukul. It acts as an antagonist of the farnesoid X receptor in humans. 了解更多
  38. LM-1484

    Catalog No. A19872
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    CysLT1 receptor antagonist
    LM-1484 is an antagonist of CysLT1 receptor and displays a higher affinity for 3H-LTC4 sites. 了解更多
  39. AZD7594

    Catalog No. A19866
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    glucocorticoid receptor modulator
    AZD7594 is a potent selective nonsteroidal glucocorticoid receptor modulator, with an IC50 of 0.9 nM. 了解更多
  40. Ecastolol

    Catalog No. A19846
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    beta adrenergic receptor antagonist
    Ecastolol is a beta adrenergic receptor antagonist, with antianginal activities. 了解更多
  41. VU0467154

    Catalog No. A19842
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    mAChR modulator
    VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor (mAChR), potentiating the response to ACh with pEC50s of 7.75, 6.2 and 6 for rat, human and cynomolgus monkey M4 receptor, respectively. 了解更多
  42. Zuranolone

    Catalog No. A19805
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    GABAA receptor agonist
    Zuranolone is a potent GABAA receptor agonist with EC50s of 296 and 163 nM for α1β2γ2 and α4β3δ GABAA receptors, respectively. 了解更多
  43. LCB-2853

    Catalog No. A19790
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    TXA2 receptor
    LCB-2853 is an antagonist of thromboxane A2 (TXA2) receptor, with antiplatelet and antithrombotic activities. 了解更多
  44. ACP-105

    Catalog No. A19778
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    androgen receptor modulator
    ACP-105 is an orally available, selective amd potent androgen receptor modulator (SARM), with pEC50s of 9.0 and 9.3 for AR wild type and T877A mutant, respectively. 了解更多
  45. Dianicline dihydrochloride

    Catalog No. A19775
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    α4β2 nicotinic acetylcholine receptor partial agonist
    Dianicline dihydrochloride is a α4β2 nicotinic acetylcholine receptor partial agonist, a class of drugs that includes varenicline and cytisine for smoking cessation. 了解更多
  46. CGRP antagonist 1

    Catalog No. A19760
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    CGRP receptor antagonist
    CGRP antagonist 1 is a highly potent CGRP receptor antagonist with a Ki and IC50 of 35 and 57 nM, respectively. 了解更多
  47. GDC-0927

    Catalog No. A19747
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    estrogen receptor antagonist
    GDC-0927 (SRN-927) is a novel, potent, non-steroidal, orally bioavailable, selective estrogen receptor antagonist. 了解更多
  48. CGP48369

    Catalog No. A19745
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    angiotensin II receptor antagonist
    CGP48369 is a nonpeptidic angiotensin II receptor antagonist, used for anti-hypertensive research. 了解更多
  49. LSZ-102

    Catalog No. A19728
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    estrogen receptor degrader
    LSZ-102 is a potent, orally bioavailable selective estrogen receptor degrader with an IC50 of 0.2 nM. 了解更多
  50. NPS ALX Compound 4a

    Catalog No. A19703
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    5-HT6 receptor antagonist
    NPS ALX Compound 4a is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist with an IC50 of 7.2 nM, which also has a great binding affinity with Ki of 0.2 nM. 了解更多

产品 301 到 350 共 1701个

每页
页面:
  1. 5
  2. 6
  3. 7
  4. 8
  5. 9

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