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产品 401 到 450 共 2783个

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  1. Thiazolidinone-Derivatives-1

    Catalog No. A20355
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    Thiazolidinone-Derivatives-1 is an antiulcer agent which inhibits the secretion of gastric acid. 了解更多
  2. Dolutegravir intermediate-1

    Catalog No. A20351
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    integrase inhibitor
    Dolutegravir is an integrase inhibitor developed for the treatment of human immunodeficiency virus (HIV)-l infection. 了解更多
  3. GZD856

    Catalog No. A20345
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    PDGFRα/β inhibitor
    GZD856 is a novel and orally bioavailable PDGFRα/β inhibitor with IC50s of 68.6 and 136.6 nM, respectively. 了解更多
  4. MDL 19301

    Catalog No. A20341
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    MDL 19301 is a nonsteroidal, anti-inflammatory agent. 了解更多
  5. L002

    Catalog No. A20336
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    KAT3B inhibitor
    L002 is a novel potent, specific acetyltransferase p300 (KAT3B) inhibitor with an IC50 of 1.98 uM. 了解更多
  6. 2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide

    Catalog No. A20334
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    2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide is a compound that inhibits stress-induced ulcer and low toxicity, and can maintain the content of phospholipase A2 and prostaglandin E2 in ulcerated rats induced by water immersed restrained stress. 了解更多
  7. Nucleocidin

    Catalog No. A20329
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    Nucleocidin is an antitrypanosomal antibiotic, inhibiting the transfer of labeled amino acid from S-RNA to protein. 了解更多
  8. GLX351322

    Catalog No. A20327
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    Nox4 inhibitor
    GLX351322 is an inhibitor of NADPH oxidase 4 (Nox4), and inhibits hydrogen peroxide production from NOX4-overexpressing cells with an IC50 of 5 μM. 了解更多
  9. VH-298

    Catalog No. A20326
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    VHL:HIF-α interaction inhibitor
    VH-298 is a highly potent inhibitor of the VHL:HIF-α interaction with a Kd value of 80 to 90 nM, used in PROTAC technology. 了解更多
  10. SUN11602

    Catalog No. A20323
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    SUN11602 is a novel aniline compound with basic fibroblast growth factor-like activity. 了解更多
  11. ATM-3507

    Catalog No. A20320
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    tropomyosin inhibitor
    ATM-3507 is a potent tropomyosin inhibitor with IC50s from 3.83-6.84 μM in human melanoma cell lines. 了解更多
  12. HMR 1556

    Catalog No. A20313
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    IKs blocker
    HMR 1556, a chromanol derivative, is a IKs blocker with IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively. 了解更多
  13. Pemigatinib

    Catalog No. A20312
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    FGFR inhibitor
    Pemigatinib is a selective FGFR inhibitor in development for the treatment of patients with cholangiocarcinoma. 了解更多
  14. CNS-5161 hydrochloride

    Catalog No. A20308
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    NMDA ion-channel antagonist
    CNS-5161 hydrochloride is a novel NMDA ion-channel antagonist that interacts with the NMDA receptor/ion channel site to produce a noncompetitive blockade of the actions of glutamate. 了解更多
  15. MethADP

    Catalog No. A20303
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    CD73 inhibitor
    MethADP is a specific CD73 inhibitor. 了解更多
  16. Tazanolast

    Catalog No. A20296
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    Tazanolast is a selective mast-cell-stabilizing drug, on ozone-induced airway hyperresponsiveness in guinea pigs. 了解更多
  17. Dexanabinol

    Catalog No. A20290
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    Dexanabinol exhibits not only the antioxidant and neuroprotective activities in brain but also anti-inflammatory activity by inhibiting NF-κB and decreasing cytokines such as TNFα and interleukin-6, which could ensure the integrity of BBB and reduce cell apoptosis and death. 了解更多
  18. LAS-31180

    Catalog No. A20285
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    PDE3 inhibitor
    LAS-31180 is an inhibitor of phosphodiesterase 3, with positive inotropic and vasodilator properties. 了解更多
  19. Terbufibrol

    Catalog No. A20276
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    Terbufibrol has been shown highly active in reducing serum total cholesterol (TC) levels in the normal and hypercholesterolemic male rat. 了解更多
  20. N33-TEG-COOH

    Catalog No. A20274
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    PROTAC linker
    N33-TEG-COOH is a PROTAC linker containing four polyethylene glycol (PEG) units. 了解更多
  21. 1,2-Distearoyl-sn-glycero-3-phosphorylethanolamine

    Catalog No. A20272
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    1,2-Distearoyl-sn-glycero-3-phosphorylethanolamine (DSPE) is a phosphoethanolamine (PE) lipid that can be used in the synthesis of liposomes. 了解更多
  22. 2-Aminoacridone

    Catalog No. A20270
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    2-Aminoacridone is a widely used fluorophore (λexc=428 nm, λem=525 nm). 了解更多
  23. Gln-AMS

    Catalog No. A20260
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    AARS inhibitor
    Gln-AMS is an aminoacyl-tRNA synthetases (AARS) inhibitor, which binds the A-domain within the NRPS enzymes. 了解更多
  24. Tefinostat

    Catalog No. A20258
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    pan HDAC inhibitor
    Tefinostat (CHR-2845) is a monocyte/macrophage-targeted pan HDAC inhibitor, cleaved into active acid CHR-2847 by the intracellular esterase human carboxylesterase-1 (hCE-1). Anti-monocytoid lineage leukaemias activity. 了解更多
  25. AGI-25696

    Catalog No. A20250
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    MATA2 inhibitors
    AGI-25696 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-25696 blocks growth of MTAP-deleted tumors in vivo. 了解更多
  26. α-2,3-sialyltransferase-IN-1

    Catalog No. A20249
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    α-2,3-sialyltransferase inhibitor
    α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is a noncompetitive α-2,3-sialyltransferase inhibitor with an IC50 of 6 μM. 了解更多
  27. Arg-AMS

    Catalog No. A20248
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    arginyl tRNA synthetase inhibitor
    Arg-AMS is a potent nanomolar inhibitor of arginyl tRNA synthetase, which displays tightly bound inhibitory characteristics for the A-domains in non-ribosomal peptide synthetases (NRPS) enzymes. 了解更多
  28. Zabofloxacin

    Catalog No. A20246
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    antibacterial candidate for clinical trials
    Zabofloxacin (DW-224a Free base) is a novel fluoronaphthyridone quinolone with a 7-pyrrolidone substituent that is considered a potent antibacterial candidate for clinical trials. 了解更多
  29. PNU288034

    Catalog No. A20241
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    oxazolidinone antibiotic
    PNU288034 is a potent oxazolidinone antibiotic. 了解更多
  30. Talazoparib tosylate

    Catalog No. A20238
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    PARP1/2 inhibitor
    Talazoparib tosylate (BMN 673ts) is a novel, potent and orally available PARP1/2 inhibitor with an IC50 of 0.57 nM for PARP1. 了解更多
  31. AGI-24512

    Catalog No. A20237
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    MATA2 inhibitors
    AGI-24512 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-24512 blocks growth of MTAP-deleted cancer cells in vitro. 了解更多
  32. (S,R,S)-AHPC-PEG2-N3

    Catalog No. A20234
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    E3 ligase ligand-linker conjugate
    (S,R,S)-AHPC-PEG2-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 2-unit PEG linker used in PROTAC technology. 了解更多
  33. Antibacterial compound 1

    Catalog No. A20228
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    Antibacterial compound 1 is a oxazolidinone extracted from patent WO1999037630A1 with antibacterial activities. 了解更多
  34. MAT2A inhibitor 1

    Catalog No. A20226
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    MATA2 inhibitors
    MAT2A inhibitor 1 is a methionine adenosyltransferase 2A (MATA2) inhibitor with an IC50 less than l00 nM. 了解更多
  35. (S,R,S)-AHPC-PEG1-N3

    Catalog No. A20223
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    E3 ligase ligand-linker conjugate
    (S,R,S)-AHPC-PEG1-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 1-unit PEG linker used in PROTAC technology. 了解更多
  36. Rilmazafone

    Catalog No. A20222
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    Rilmazafone is a water-soluble benzodiazepine prodrug that acts as a sedative and hypnotic neuropsychiatric agent. 了解更多
  37. Foscarbidopa

    Catalog No. A20221
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    dopamine receptor agonist
    Foscarbidopa (Carbidopa 4??-monophosphate) is a prodrug of Carbidopa, acts as a dopamine receptor agonist. 了解更多
  38. (S,R,S)-AHPC-PEG4-N3

    Catalog No. A20214
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    E3 ligase ligand-linker conjugate
    (S,R,S)-AHPC-PEG4-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 4-unit PEG linker used in PROTAC technology. 了解更多
  39. Oxythiamine

    Catalog No. A20210
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    vitamin B1 antagonist
    Oxythiamine, an antimetabolite and a vitamin B1 antagonist, is a well-known thiamine antagonist and inhibitor of transketolase. 了解更多
  40. JH-VIII-157-02

    Catalog No. A20205
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    ALK inhibitor
    JH-VIII-157-02 is a structural analogue of alectinib, acts as an ALK inhibitor, and shows an IC50 of 2 nM for echinoderm microtubule-associated protein-like 4-ALK (EML4-ALK) G1202R in cells. 了解更多
  41. (S,R,S)-AHPC-PEG3-NH2 hydrochloride

    Catalog No. A20202
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    E3 ligase ligand-linker conjugate
    (S,R,S)-AHPC-PEG3-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 3-unit PEG linker used in PROTAC technology. 了解更多
  42. Runcaciguat

    Catalog No. A20200
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    soluble guanylate cyclase stimulator
    Runcaciguat is an orally active stimulator of soluble guanylate cyclase, and is used in the research of cardiovascular and renal diseases combined with selective partial adenosine A1 receptor agonists. 了解更多
  43. Levophacetoperane hydrochloride

    Catalog No. A20198
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    Levophacetoperane inhibits in vitro in a competitive manner, norepinephrin uptake and dopamine uptake. 了解更多
  44. (S,R,S)-AHPC-PEG2-NH2 hydrochloride

    Catalog No. A20191
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    E3 ligase ligand-linker conjugate
    (S,R,S)-AHPC-PEG2-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 2-unit PEG linker used in PROTAC technology. 了解更多
  45. Taminadenant

    Catalog No. A20190
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    adenosine receptor antagonist
    Taminadenant is an antagonist of adenosine receptor. 了解更多
  46. Irindalone

    Catalog No. A20187
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    serotonin 5-HT2 antagonist
    Irindalone is a novel serotonin 5-HT2 antagonist. 了解更多
  47. Hispidol

    Catalog No. A20185
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    Hispidol ((Z)-Hispidol) is a potential therapeutic for inflammatory bowel disease; inhibits TNF-α induced adhesion of monocytes to colon epithelial cells with an IC50 of 0.50 ?M. 了解更多
  48. Thalidomide-O-amido-C4-NH2

    Catalog No. A20184
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    E3 ligase ligand-linker conjugate
    Thalidomide-O-amido-C4-NH2 is a synthesized E3 ligase ligand-linker conjugate that incorporates the Thalidomide based cereblon ligand and a linker used in PROTAC technology. 了解更多
  49. (S,R,S)-AHPC-PEG4-NH2 hydrochloride

    Catalog No. A20180
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    E3 ligase ligand-linker conjugate
    (S,R,S)-AHPC-PEG4-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 4-unit PEG linker used in PROTAC technology. 了解更多
  50. ABT-072

    Catalog No. A20177
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    NS5B polymerase inhibitor
    ABT-072 is a nonnucleoside NS5B polymerase inhibitor and a candidate drug evaluated for treatment of hepatitis C virus. 了解更多

产品 401 到 450 共 2783个

每页
页面:
  1. 7
  2. 8
  3. 9
  4. 10
  5. 11

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