“AG 013736”的搜索结果

产品 451 到 500 共 3340个

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  1. MF 5137

    Catalog No. A20325
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    MF 5137 is a potent antibacterial agent. 了解更多
  2. Sigma-2 receptor antagonist 1

    Catalog No. A20310
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    sigma-2 (??-2) receptor antagonist
    Sigma-2 receptor antagonist 1 is a sigma-2 (??-2) receptor antagonist. 了解更多
  3. Droxicainide

    Catalog No. A20309
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    Droxicainide is an antiarrhythmic agent. 了解更多
  4. CNS-5161 hydrochloride

    Catalog No. A20308
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    NMDA ion-channel antagonist
    CNS-5161 hydrochloride is a novel NMDA ion-channel antagonist that interacts with the NMDA receptor/ion channel site to produce a noncompetitive blockade of the actions of glutamate. 了解更多
  5. Antifungal agent 1

    Catalog No. A20307
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    Antifungal agent 1 is a potent antifungal agent. 了解更多
  6. Diphenylterazine

    Catalog No. A20299
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    Diphenylterazine is a bioluminescence agent. 了解更多
  7. L162389

    Catalog No. A20297
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    angiotensin AT1 receptor antagonist
    L162389 is a potent antagonist of angiotensin AT1 receptor with Ki of 28 nM. 了解更多
  8. Fosmidomycin sodium salt

    Catalog No. A20292
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    Fosmidomycin sodium salt is a phosphonic acid antibiotic and a antimalarial drug, which is active against both Gram-negative and Gram-positive bacteria. 了解更多
  9. Telratolimod

    Catalog No. A20289
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    TLR7/8 agonist
    Telratolimod is a toll like receptors 7/8 (TLR7/8) agonist, with antitumor activity. 了解更多
  10. Abaperidone

    Catalog No. A20286
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    5-HT2A/dopamine D2 antagonist
    Abaperidone is a potent antagonist of 5-HT2A?receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM. 了解更多
  11. MRZ 2-514

    Catalog No. A20277
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    NMDA receptor (glycineB) antagonist
    MRZ 2-514 is an antagonist of the strychnine-insensitive modulatory site of the NMDA receptor (glycineB), with Ki of 33 μM. 了解更多
  12. Lidanserin

    Catalog No. A20266
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    5-HT2A/α1-adrenergic receptor antagonist
    Lidanserin is a drug which acts as a combined 5-HT2A and α1-adrenergic receptor antagonist. 了解更多
  13. Tefinostat

    Catalog No. A20258
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    pan HDAC inhibitor
    Tefinostat (CHR-2845) is a monocyte/macrophage-targeted pan HDAC inhibitor, cleaved into active acid CHR-2847 by the intracellular esterase human carboxylesterase-1 (hCE-1). Anti-monocytoid lineage leukaemias activity. 了解更多
  14. Azelaprag

    Catalog No. A20257
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    Azelaprag (Example 263.0) is an apelin receptor agonist drug candidate. 了解更多
  15. TBAJ-587

    Catalog No. A20256
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    anti-tuberculosis agent
    TBAJ-587, a potent anti-tuberculosis agent, inhibits M.tb strain H37Rv growth with MIC90s of 0.006 and <0.02 ?g/mL in MABA and LORA assay, respectively. 了解更多
  16. Spirendolol

    Catalog No. A20254
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    β adrenergic receptor antagonist
    Spirendolol is a β adrenergic receptor antagonist. 了解更多
  17. AGI-25696

    Catalog No. A20250
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    MATA2 inhibitors
    AGI-25696 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-25696 blocks growth of MTAP-deleted tumors in vivo. 了解更多
  18. Masupirdine free base

    Catalog No. A20245
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    5-HT6 receptor antagonist
    Masupirdine free base (SUVN-502 free base) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). 了解更多
  19. RORγt Inverse agonist 2

    Catalog No. A20243
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    RORγt inverse agonist
    RORγt Inverse agonist 2 is a selective, orally active RORγt inverse agonist with an EC50 of 119 nM. 了解更多
  20. AGI-24512

    Catalog No. A20237
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    MATA2 inhibitors
    AGI-24512 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-24512 blocks growth of MTAP-deleted cancer cells in vitro. 了解更多
  21. JAK-IN-4

    Catalog No. A20230
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    JAK inhibitor
    JAK-IN-4 is a prodrug of a JAK inhibitor, effective in murine collagen induced arthritis model. 了解更多
  22. Rilmazafone

    Catalog No. A20222
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    Rilmazafone is a water-soluble benzodiazepine prodrug that acts as a sedative and hypnotic neuropsychiatric agent. 了解更多
  23. Foscarbidopa

    Catalog No. A20221
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    dopamine receptor agonist
    Foscarbidopa (Carbidopa 4??-monophosphate) is a prodrug of Carbidopa, acts as a dopamine receptor agonist. 了解更多
  24. SSTR5 antagonist 1

    Catalog No. A20218
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    SSTR5 antagonist
    SSTR5 antagonist 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a). 了解更多
  25. Foslevodopa

    Catalog No. A20212
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    dopamine receptor agonist
    Foslevodopa is a dopamine receptor agonist. 了解更多
  26. ALB-127158(a)

    Catalog No. A20211
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    MCH1 receptor antagonist
    ALB-127158(a) is a potent and selective melanin concentrating hormone 1 (MCH1) receptor antagonist. 了解更多
  27. Oxythiamine

    Catalog No. A20210
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    vitamin B1 antagonist
    Oxythiamine, an antimetabolite and a vitamin B1 antagonist, is a well-known thiamine antagonist and inhibitor of transketolase. 了解更多
  28. UT-155

    Catalog No. A20203
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    AR antagonist
    UT-155 is a selective and potent androgen receptor (AR) antagonist, with a Ki of 267 nM for UT-155 binding to AR-LBD. 了解更多
  29. NK-1 Antagonist 1

    Catalog No. A20201
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    NK-1 receptor antagonist
    NK-1 Antagonist 1 (Rolapitant intermediate) is an antagonist of NK-1 receptor, used in the research of NK-1 related diseases and conditions such as cough, overactive bladder, alcohol dependency and depression. 了解更多
  30. Runcaciguat

    Catalog No. A20200
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    soluble guanylate cyclase stimulator
    Runcaciguat is an orally active stimulator of soluble guanylate cyclase, and is used in the research of cardiovascular and renal diseases combined with selective partial adenosine A1 receptor agonists. 了解更多
  31. GPR84 antagonist 8

    Catalog No. A20193
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    GPR84 antagonist
    GPR84 antagonist 8 is a selective GPR84 antagonist. 了解更多
  32. Taminadenant

    Catalog No. A20190
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    adenosine receptor antagonist
    Taminadenant is an antagonist of adenosine receptor. 了解更多
  33. Oral antiplatelet agent 1

    Catalog No. A20188
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    Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro as well as antithrombotic efficacy in a rat model. P2Y receptor antagonist. 了解更多
  34. Irindalone

    Catalog No. A20187
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    serotonin 5-HT2 antagonist
    Irindalone is a novel serotonin 5-HT2 antagonist. 了解更多
  35. Wy 49051

    Catalog No. A20176
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    H1 receptor antagonist
    Wy 49051 is a potent, orally active H1 receptor antagonist, with IC50 of 44 nM. 了解更多
  36. (S,R,S)-AHPC-PEG6-C4-Cl

    Catalog No. A20169
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    (S,R,S)-AHPC-PEG6-C4-Cl is a small molecule HaloPROTAC that incorporates the (S,R,S)-AHPC based VHL ligand and 6-unit PEG linker. (S,R,S)-AHPC-PEG6-C4-Cl is capable of inducing the degradation of GFP-HaloTag7 in cell-based assays. 了解更多
  37. FK1052 hydrochloride

    Catalog No. A20164
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    5-HT3 /5-HT4 receptor dual antagonist
    FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist. 了解更多
  38. MMG-11

    Catalog No. A20159
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    human TLR2 antagonist
    MMG-11 is a potent and selective human TLR2 antagonist with low cytotoxicity. 了解更多
  39. (S,R,S)-AHPC-(C3-PEG)2-C6-Cl

    Catalog No. A20157
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    (S,R,S)-AHPC-(C3-?PEG)?2-?C6-?Cl is a small molecule HaloPROTAC that incorporates the (S,R,S)-AHPC based VHL ligand and 2-unit PEG linker. (S,R,S)-AHPC-(C3-?PEG)?2-?C6-?Cl is capable of inducing the degradation of GFP-HaloTag7 in cell-based assays. 了解更多
  40. 5-HT7 agonist 1

    Catalog No. A20143
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    5-HT7 receptor agonist
    5-HT7 agonist 1 is a selective 5-HT7 receptor agonist, with an IC50 of 222.93 nM, can be used for the 5-HT7 receptor related disease, such as CNS disorders. 了解更多
  41. DIQ3

    Catalog No. A20141
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    DIQ3 is a potent anti-cancer agent, nontoxic to normal human cell lines. 了解更多
  42. Ceftobiprole

    Catalog No. A20135
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    Ceftobiprole is a broad-spectrum cephalosporin with activity against Methicillin-resistant staphylococcus aureus (MRSA) with the MIC90 value of 2 mcg/mL. 了解更多
  43. Letrazuril

    Catalog No. A20132
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    Letrazuril is an anti-HIV agent. 了解更多
  44. GRK2-IN-1

    Catalog No. A20131
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    GRKs-IN-1, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=30 nM) and GRK5 (IC50=7.1 μM). GRKs-IN-1 is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine. 了解更多
  45. GPR40/FFAR1 modulator 1

    Catalog No. A20129
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    GPR40/FFAR1 agonist
    GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1). 了解更多
  46. Losmiprofen

    Catalog No. A20115
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    antiinflammatory agent
    Losmiprofen is a nonsteroidal antiinflammatory agent. 了解更多
  47. Furprofen

    Catalog No. A20107
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    Furprofen is an non-steroidal anti-inflammatory drug (NSAID) with analgesic properties. Furprofen acts via the inhibition of prostaglandin (PGE) synthesis. Furprofen can be treated orally for the relief of pain. 了解更多
  48. Saredutant

    Catalog No. A20096
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    NK2 receptor antagonist
    Saredutant is a selective NK2 receptor antagonist. 了解更多
  49. Pparδ agonist

    Catalog No. A20088
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    PPARδ agonist
    PPARδ agonist is a PPARδ agonist extracted from patent US20180071304, compound example 10. 了解更多
  50. Gemcabene

    Catalog No. A20083
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    lipid-lowering agent
    Gemcabene (PD-72953), a first-in-class lipid-lowering agent. 了解更多

产品 451 到 500 共 3340个

每页
页面:
  1. 8
  2. 9
  3. 10
  4. 11
  5. 12

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