“glucagon receptor”的搜索结果

产品 501 到 550 共 1712个

每页
页面:
  1. 9
  2. 10
  3. 11
  4. 12
  5. 13

设置降序顺序
  1. RAD140

    Catalog No. A21205
    Quick View
    androgen receptor modulator
    RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM). 了解更多
  2. LAS101057

    Catalog No. A21203
    Quick View
    A2B receptor antagonist
    LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. 了解更多
  3. MDL 105519

    Catalog No. A21192
    Quick View
    NMDA receptor antagonist
    MDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多
  4. TCN238

    Catalog No. A21191
    Quick View
    mGlu4 receptor modulator
    TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM. 了解更多
  5. Velneperit

    Catalog No. A21190
    Quick View
    NPY Y5 receptor antagonist
    Velneperit (S-2367) is a novel neuropeptide Y (NPY) Y5 receptor antagonist. 了解更多
  6. Befiradol

    Catalog No. A21189
    Quick View
    5-HT1A receptor agonist
    Befiradol (NLX-112) is a selective 5-HT1A receptor agonist. 了解更多
  7. CE-224535

    Catalog No. A21183
    Quick View
    P2X7 receptor antagonist
    CE-224535 is a selective P2X7 receptor antagonist. 了解更多
  8. L-655708

    Catalog No. A21181
    Quick View
    GABAA receptor inverse agonist
    L-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM). 了解更多
  9. SB-423562

    Catalog No. A21170
    Quick View
    calcium-sensing receptor (CaR) antagonist
    SB-423562 is a short-acting calcium-sensing receptor (CaR) antagonist. 了解更多
  10. SB-423557

    Catalog No. A21169
    Quick View
    alcium-sensing receptor (CaR) antagonist
    SB-423557 is an orally active calcium-sensing receptor (CaR) antagonist (IC50=520 nM), precursor of SB-423562 (IC50=73 nM). 了解更多
  11. PF-4778574

    Catalog No. A21157
    Quick View
    AMPA receptor positive allosteric modulator
    PF-4778574 is a potent AMPA receptor positive allosteric modulator (PAM) that has been shown to enhance cognition in animal models. 了解更多
  12. Tezosentan

    Catalog No. A21118
    Quick View
    endothelin (ET) receptor antagonist
    Tezosentan (RO 610612) is an endothelin (ET) receptor antagonist, with pA2s of 9.5, 7.7 for ETA and ETB receptors, respectively. 了解更多
  13. GLPG0492

    Catalog No. A21105
    Quick View
    androgen receptor modulator
    GLPG0492 is a novel selective androgen receptor modulator; exhibited anabolic activity on muscle, strongly dissociated from the androgenic activity on prostate after oral dosing. 了解更多
  14. LY2812223

    Catalog No. A21100
    Quick View
    mGlu2 receptor agonist
    LY2812223 is a highly potent, functionally selective mGlu2 receptor agonist with mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, respectively). 了解更多
  15. Nelonicline

    Catalog No. A21079
    Quick View
    neuronal nicotinic receptor agonist
    Nelonicline (ABT-126) is a selective neuronal nicotinic receptor agonist. 了解更多
  16. Transcrocetinate disodium

    Catalog No. A21051
    Quick View
    NMDA receptor antagonist
    Transcrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多
  17. Terutroban

    Catalog No. A20884
    Quick View
    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多
  18. Sparsentan

    Catalog No. A20879
    Quick View
    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  19. Clopidogrel thiolactone

    Catalog No. A20862
    Quick View
    P2Y12 receptor inhibitor
    Clopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent. 了解更多
  20. Azilsartan medoxomil monopotassium

    Catalog No. A20860
    Quick View
    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  21. APNEA

    Catalog No. A20845
    Quick View
    A3 adenosine receptor agonist
    APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. 了解更多
  22. SYM2206

    Catalog No. A20843
    Quick View
    AMPA receptor antagonist
    SYM 2206 is a novel, potent, non-competitive AMPA receptor antagonist. 了解更多
  23. Haloperidol hydrochloride

    Catalog No. A18304
    Quick View
    dopamine D2 receptor antagonist
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多
  24. Setiptiline

    Catalog No. A18090
    Quick View
    serotonin receptor antagonist
    Setiptiline(Org-8282) is a serotonin receptor antagonist. 了解更多
  25. Quinagolide hydrochloride

    Catalog No. A18038
    Quick View
    dopamine D2 receptor agonist
    Quinagolide hydrochloride is a selective dopamine D2 receptor agonist, also is a prolactin inhibitor. 了解更多
  26. Pyrantel tartrate

    Catalog No. A18032
    Quick View
    antinematodal thiophene nicotinic receptor agonist
    Pyrantel tartrate is an antinematodal thiophene nicotinic receptor agonist and can elicit spastic muscle paralysis in parasitic worms due to prolonged activation of the excitatory nicotinic acetylcholine (nACh) receptors on body wall muscle. 了解更多
  27. Oxytocin

    Catalog No. A17988
    Quick View
    oxytocin receptor ligand
    Oxytocin (α-Hypophamine) is a mammalian neurohypophysial hormone; its actions are mediated by specific, high-affinity oxytocin receptors; ligand of oxytocin receptor. 了解更多
  28. (Z)-Thiothixene

    Catalog No. A17891
    Quick View
    Serotonergic receptor antagonist
    (Z)-Thiothixene is an antagonist of serotonergic receptor extracted from patent US 20150141345 A1. 了解更多
  29. Sunitinib

    Catalog No. A17858
    Quick View
    multi-targeted receptor tyrosine kinase inhibitor
    Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase inhibitor with IC50s of 80 nM and 2 nM for VEGFR2 and PDGFRβ, respectively. 了解更多
  30. Trimethobenzamide hydrochloride

    Catalog No. A17648
    Quick View
    D2 receptor blocker
    Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. 了解更多
  31. Ziprasidone hydrochloride

    Catalog No. A16790
    Quick View
    5-HT (serotonin)/dopamine receptor antagonist
    Ziprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  32. WAY-100635 Maleate

    Catalog No. A16787
    Quick View
    5-HT1A receptor antagonist
    WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. 了解更多
  33. Tamoxifen

    Catalog No. A16738
    Quick View
    selective estrogen receptor modulator (SERM)
    Tamoxifen (ICI 47699) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells. 了解更多
  34. SB-334867 free base

    Catalog No. A16695
    Quick View
    orexin OX1 receptor antagonist
    SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. 了解更多
  35. (R)-Baclofen

    Catalog No. A16680
    Quick View
    GABAB receptor agonist
    (R)-Baclofen(STX209) is a selective GABAB receptor agonist. 了解更多
  36. Ifenprodil tartrate

    Catalog No. A16583
    Quick View
    NMDA receptor antagonist
    Ifenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多
  37. Dexamethasone acetate

    Catalog No. A16494
    Quick View
    glucocorticoid receptor agonist
    Dexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. 了解更多
  38. Varenicline Tartrate

    Catalog No. A11618
    Quick View
    nicotinic receptor partial agonist
    Varenicline Tartrate(CP 526555;Champix) is a nicotinic receptor partial agonist; it stimulates nicotine receptors more weakly than nicotine itself does. 了解更多
  39. Taranabant

    Catalog No. A11578
    Quick View
    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  40. SB 271046 Hydrochloride

    Catalog No. A11573
    Quick View
    5-HT6 receptor antagonist
    SB271046 Hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9. 了解更多
  41. SU14813 maleate

    Catalog No. A11556
    Quick View
    multi-targeted receptor tyrosine kinases inhibitor
    SU14813 maleate is a multi-targeted receptor tyrosine kinases inhibitor with IC50s of 50, 2, 4, 15 nM for VEGFR2, VEGFR1, PDGFRβ and KIT. 了解更多
  42. Rivanicline oxalate

    Catalog No. A11544
    Quick View
    neuronal nicotinic receptor agonist
    Rivanicline oxalate (RJR-2403 oxalate; (E)-Metanicotine oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 3.6 μM). 了解更多
  43. Olcegepant

    Catalog No. A11512
    Quick View
    CGRP1 receptor
    Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. 了解更多
  44. Montelukast sodium

    Catalog No. A11490
    Quick View
    CysLT1 receptor antagonist
    Montelukast (sodium) (MK0476) is a potent, selective CysLT1 receptor antagonist. 了解更多
  45. JDTic

    Catalog No. A11468
    Quick View
    κ-opioid receptor antagonist
    JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. 了解更多
  46. IRAK inhibitor 3

    Catalog No. A11457
    Quick View
    IL-1 receptor-associated kinase (IRAK) kinase modulator
    IRAK inhibitor 3 is an interleukin-1 (IL-I) receptor-associated kinase (IRAK) kinase modulator extracted from patent WO2008030579 A2. 了解更多
  47. IRAK inhibitor 2

    Catalog No. A11456
    Quick View
    interleukin-1 receptor associated kinase inhibitor
    IRAK inhibitor 2 is interleukin-1 receptor associated kinase inhibitor . 了解更多
  48. CGS 21680

    Catalog No. A11354
    Quick View
    adenosine A2A receptor agonist
    CGS 21680 is a selective adenosine A2A receptor agonist, with a Ki of 27 nM. 了解更多
  49. Cabozantinib S-malate

    Catalog No. A11349
    Quick View
    multiple receptor tyrosine kinases inhibitor
    Cabozantinib S-malate (XL184 S-malate) is a potent multiple receptor tyrosine kinases inhibitor that inhibits VEGFR2, c-Met, Kit, Axl and Flt3 with IC50s of 0.035, 1.3, 4.6, 7 and 11.3 nM, respectively. 了解更多
  50. β3-AR agonist 1

    Catalog No. A12777
    Quick View
    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多

产品 501 到 550 共 1712个

每页
页面:
  1. 9
  2. 10
  3. 11
  4. 12
  5. 13

设置降序顺序
Rewards