“sn 2”的搜索结果

产品 501 到 550 共 17249个

每页
页面:
  1. 9
  2. 10
  3. 11
  4. 12
  5. 13

设置降序顺序
  1. CRT0066101 free base

    Catalog No. A22539
    Quick View
    PRKDs inhibitor
    CRT0066101 is a PRKDs inhibitor. CRT0066101 suppressed the proliferation and migration of four bladder cancer cell lines in vitro. CRT0066101 blocked tumor growth in a mouse flank xenograft model of bladder cancer. 了解更多
  2. Osajin

    Catalog No. A22540
    Quick View
    Osajin is a bioactive isoflavone present in the fruit of Maclura pomifera, commonly referred to as the Osage orange. 了解更多
  3. ML095 HCl

    Catalog No. A22545
    Quick View
    PLAP inhibitor
    ML-095 is an inhibitor of PLAP (IC50 = 3.7 μM) that demonstrates high selectivity against the related alkaline phosphatases, TNAP and IAP (IC50s > 100 μM). 了解更多
  4. MC-Gly-Gly-Phe

    Catalog No. A22546
    Quick View
    MC-Gly-Gly-Phe is a cleavable linker used for antibody-drug conjugates (ADC). 了解更多
  5. Boc-Gly-Gly-Phe-Gly-OH

    Catalog No. A22547
    Quick View
    Boc-Gly-Gly-Phe-Gly-OH is a protease cleavable linker used for the antibody-drug conjugate (ADC). 了解更多
  6. Boc-Dap-NE

    Catalog No. A22548
    Quick View
    Boc-Dap-NE is a cleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs). 了解更多
  7. Navoximod free base

    Catalog No. A22549
    Quick View
    IDO1 inhibitor
    Navoximod, also known as IDO-IN-7 and NLG-1488, is an indoleamine 2,3-dioxygenase (IDO) inhibitor. 了解更多
  8. CP-609754

    Catalog No. A22550
    Quick View
    CP-609754, also known as CP-609,754, LNK 754 and OSI 754, is a potent farnesyltransferase inhibitor with potential anticancer activity. 了解更多
  9. ATPO

    Catalog No. A22552
    Quick View
    Ampa Receptor Antagonist
    ATPO is a potent and Selective Ampa Receptor Antagonist. 了解更多
  10. ML-193

    Catalog No. A22553
    Quick View
    GPR55 antagonist
    ML 193 is a selective GPR55 antagonist (IC50 = 221 nM). Exhibits >27-, >145- and >145-fold selectivity for GPR55 over CB1, GPR35 and CB2, respectively. Inhibits ERK signaling in vitro. 了解更多
  11. JNJ-10198409

    Catalog No. A22554
    Quick View
    PDGFRα/PDGFRβ inhbitor
    JNJ 10198409 is a potent platelet-derived growth factor receptor (PDGFR) inhibitor (IC50 values are 4.2 and 45 nM for PDGFRβ and PDGFRα, respectively). Also inhibits c-Abl, Lck, c-Src and Fyn kinases (IC50 values are 22, 100, 185 and 378 nM respectively). 了解更多
  12. SEP-363856 HCl

    Catalog No. A22555
    Quick View
    SEP-363856, also known as SEP-856, is an orally active and CNS active psychotropic agent. 了解更多
  13. MYF-01-37

    Catalog No. A22556
    Quick View
    TEAD inhibitor
    MYF-01-37 is a novel covalent inhibitor of TEAD targeting Cys380. 了解更多
  14. L-Leucine-13C6

    Catalog No. A22557
    Quick View
    L-LEUCINE-13C6, also known as 13C6-D-Leucine or L-?Leucine-?1,?2,?3,?4,?5,?5'-?13C6, is a fully 13C labelled D-Leucine. 了解更多
  15. Bractoppin

    Catalog No. A22558
    Quick View
    Bractoppin is a potent and selective inhibitor of phosphopeptide recognition by the BRCA1 tBRCT domain. 了解更多
  16. YUM70

    Catalog No. A22559
    Quick View
    GRP78 inhibitor
    YUM70 is a potent inhibitor of GRP78 (Glucose-regulated protein, 78 kDa). 了解更多
  17. BRD0705

    Catalog No. A22561
    Quick View
    GSK3α inhibitor
    BRD0705 is a potent, paralog selective and orally active GSK3α inhibitor. 了解更多
  18. Luzindole

    Catalog No. A22563
    Quick View
    MT1/MT2 antagonist
    Luzindole, also known as N-0774, and N-acetyl-2-benzyltryptamine, is a melatonin receptor antagonist that preferentially targets MT1B over MT1A (Ki values are = 10-27 and 158-513 nM, respectively). 了解更多
  19. LM11A-31 HCl

    Catalog No. A22564
    Quick View
    p75NTR ligand
    LM11A-31 is a small-molecule p75NTR modulator and proNGF antagonist. 了解更多
  20. EMAC10101d

    Catalog No. A22565
    Quick View
    hCA II inhibitor
    EMAC10101d is a potent and selective inhibitor of Carbonic Anhydrase Isoform toward hCA II with an inhibitory activity in the low nanomolar range. Ki of 8.1 nM 了解更多
  21. ARS-1323-Alkyne

    Catalog No. A22566
    Quick View
    S-IIP inhibitor/KRASG12C Probe
    ARS-1323-Alkyne is a novel KRASG12C occupancy probe. 了解更多
  22. CC90001 free base

    Catalog No. A22567
    Quick View
    JNK inhibitor
    CC-90001 is a potent and selective JNK inhibitor. CC-90001 shows 12.9-fold selectivity for JNK1 over JNK2 in a cell-based model. CC-90001 can be used for the research of idiopathic pulmonary fibrosis 了解更多
  23. Pizuglanstat

    Catalog No. A22568
    Quick View
    prostaglandin synthase inhibitor
    Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor. 了解更多
  24. ZINC30303842

    Catalog No. A22569
    Quick View
    NSD2-PWWP1 antagonist
    ZINC30303842 is a NSD2-PWWP1 antagonist. 了解更多
  25. FB23 inhibitor

    Catalog No. A22571
    Quick View
    FB23 is a potent and selective inhibitor of N6-methyladenosine (m6A) demethylase FTO (fat mass and obesity associated protein). 了解更多
  26. UNC-669

    Catalog No. A22573
    Quick View
    L3MBTL domain inhibitor
    UNC-669 is a L3MBTL domain inhibitor. 了解更多
  27. SNIPER(CRABP)-11

    Catalog No. A22574
    Quick View
    PROTAC degrader
    SNIPER(CRABP)-11, also known as PROTAC cIAP1 degrader-?4, is a potent protein degrader. 了解更多
  28. Xanthurenic acid

    Catalog No. A22575
    Quick View
    II metabotropic glutamate receptor agonist
    Xanthurenic acid is a putative endogenous Group II metabotropic glutamate receptor agonist, on sensory transmission in the thalamus. 了解更多
  29. Propyl gallate

    Catalog No. A22576
    Quick View
    food antioxidant
    Propyl gallate is a common food antioxidant. Propyl gallate can inhibit the production of acrolein, glyoxal and methylglyoxal. 了解更多
  30. Methyl dihydrojasmonate

    Catalog No. A22577
    Quick View
    fragrance ingredient
    Methyl dihydrojasmonate is a fragrance ingredient with a jasmine-like odor, used in many fragrance mixtures. 了解更多
  31. Tetrahydropalmatine

    Catalog No. A22578
    Quick View
    analgesic agent
    Tetrahydropalmatine, an active component isolated from corydalis, possesses analgesic effects. Tetrahydropalmatine acts through inhibition of amygdaloid release of dopamine to inhibit an epileptic attack in rats. 了解更多
  32. Chelidonic acid

    Catalog No. A22579
    Quick View
    glutamate decarboxylase inhibitor
    Chelidonic acid is a glutamate decarboxylase inhibitor, with a Ki of 1.2 μM. 了解更多
  33. Flavokawain A

    Catalog No. A22580
    Quick View
    Anticancer agent
    Flavokawain A is found in Piper methysticum (kava plant). It suppresses expression of iNOS and COX-2 in macrophages, decreases expression of Ki67, XIAP and survivin in urothelial cell carcinoma cells, and inhibits degradation of NF-??B. 了解更多
  34. Suberoyl bis-hydroxamic acid

    Catalog No. A22581
    Quick View
    HDAC1 and HDAC3 inhibitor
    Suberoyl bis-hydroxamic acid (Suberohydroxamic acid; SBHA) is a competitive and cell-permeable HDAC1 and HDAC3 inhibitor with ID50 values of 0.25 μM and 0.30 μM, respectively. 了解更多
  35. Ethyl pyruvate

    Catalog No. A22582
    Quick View
    anti-inflammatory agent
    Ethyl pyruvate is a simple derivative of the endogenous metabolite, pyruvic acid. Ethyl pyruvate is an anti-inflammatory agent. 了解更多
  36. JTE-013

    Catalog No. A22583
    Quick View
    S1P2 antagonist
    JTE-013 is a potent and specific S1P2 (Sphingosine-1-Phosphate 2; EDG-5) antagonist. JTE-013 inhibits the specific binding of radiolabeled S1P to human and rat S1P2 with IC50s of 17 nM and 22 nM, respectively. 了解更多
  37. EAD1

    Catalog No. A22586
    Quick View
    autophagy inhibitor
    EAD1 is a potent autophagy inhibitor with antiproliferative activity in lung and pancreatic cancer cells. EAD1 also induces apoptosis. 了解更多
  38. IDO-IN-13

    Catalog No. A22587
    Quick View
    IDO1 inhibitor
    IDO-IN-13 is a potent indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor with an EC50 of 17 nM, extracted from patent WO2019040102A1, example 43. 了解更多
  39. AT-007

    Catalog No. A22588
    Quick View
    CNS penetrant Aldose Reductase inhibitor
    AT-007 is an orally active central nervous system (CNS) penetrant Aldose Reductase inhibitor for treatment of Galactosemia with an IC50 value of 100 pM. AT-007 reduces toxic galactitol levels and prevents disease complications in GALT deficiency rats. 了解更多
  40. Benzetimide hydrochloride

    Catalog No. A22589
    Quick View
    muscarinic acetylcholine receptor antagonist
    Benzetimide hydrochloride is a muscarinic acetylcholine receptor antagonist. 了解更多
  41. AER-271

    Catalog No. A22590
    Quick View
    AQP4 inhibitor
    AER-271, a phosphonate prodrug derivative of AER-270, is an aquaporin-4 (AQP4) inhibitor for the research of acute ischemic stroke. 了解更多
  42. ZK824190

    Catalog No. A22591
    Quick View
    uPA inhibitor
    ZK824190 is an orally available and selective urokinase plasminogen activator (uPA) inhibitor as a potential treatment for multiple sclerosis. IC50s of 237, 1600 and 1850 nM for uPA, tPA, and Plasmin, respectively. 了解更多
  43. SCH-23390 maleate

    Catalog No. A22592
    Quick View
    dopamine D1-like receptor antagonist
    SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively. 了解更多
  44. Lotamilast

    Catalog No. A22594
    Quick View
    PDE4 inhibitor
    Lotamilast (RVT-501; E6005) is a selective phosphodiesterase 4 (PDE4) inhibitor with an IC50 of 2.8 nM. 了解更多
  45. PF-06454589

    Catalog No. A22595
    Quick View
    LRRK2 inhibitor
    PF-06454589 is a potent and selective LRRK2 inhibitor. 了解更多
  46. NDI-091143

    Catalog No. A22596
    Quick View
    ACLY inhibitor
    NDI-091143 is a potent and high-affinity human ATP-citrate lyase (ACLY) inhibitor with an IC50 of 2.1 nM (ADP-Glo assay), a Ki of 7.0 nM and a Kd of 2.2 nM. 了解更多
  47. Carbutamide

    Catalog No. A22597
    Quick View
    hypoglycemic agent
    Carbutamide (BZ-55) is an orally active and first-generation sulfonylurea with hypoglycemic activity. 了解更多
  48. Carazolol

    Catalog No. A22598
    Quick View
    β-adrenergic receptor blocking agent
    Carazolol is a non-specific β-adrenergic receptor blocking agent and binds to β receptors irreversibly. 了解更多
  49. CKI-7

    Catalog No. A22599
    Quick View
    CK1 inhibitor
    CKI-7 is a potent and ATP-competitive casein kinase 1 (CK1) inhibitor with an IC50 of 6 μM and a Ki of 8.5 μM.CKI-7 is a selective Cdc7 kinase inhibitor. 了解更多
  50. Quipazine maleate

    Catalog No. A22600
    Quick View
    5-HT receptor agonist
    Quipazine maleate is a selective 5-HT receptor agonist that promotes the proliferation and apoptosis of human hepatocyte strain of L-02 strain and could also exert an excitatory effect on raphe neurons via stimulation of 5-HT2A receptors. 了解更多

产品 501 到 550 共 17249个

每页
页面:
  1. 9
  2. 10
  3. 11
  4. 12
  5. 13

设置降序顺序
Rewards