“glucagon receptor”的搜索结果

产品 551 到 600 共 1712个

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  1. RF9

    Catalog No. A12944
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    Neuropeptide FF receptor antagonist
    RF9 is a potent and selective Neuropeptide FF receptor antagonist, with Kis of 58??5 and 75??9 nM for hNPFF1R and hNPFF2R, respectively. 了解更多
  2. Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  3. CP-96486

    Catalog No. A12471
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    LTD4/PAF receptor antagonist
    CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. 了解更多
  4. FR167344 free base

    Catalog No. A12964
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    nonpeptide bradykinin receptor B2 antagonist
    FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. 了解更多
  5. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  6. Amelubant

    Catalog No. A12968
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    LTB4 receptor antagonist
    Amelubant (BIIL 284) is a potent, oral and long acting LTB4 receptor antagonist. 了解更多
  7. RPR104632

    Catalog No. A13385
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    NMDA receptor antagonist
    RPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. 了解更多
  8. Foropafant

    Catalog No. A13388
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    PAF receptor antagonist
    Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor. 了解更多
  9. AB-MECA

    Catalog No. A12189
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    A3 adenosine receptor agonist
    AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. 了解更多
  10. Edicotinib

    Catalog No. A13008
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    CSF-1 receptor inhibitor
    Edicotinib is a selective and orally available colony-stimulating factor-1 (CSF-1) receptor inhibitor, and has entered phase IIA clinical trial to study rheumatoid arthritis (RA) despite disease. 了解更多
  11. GLPG0187

    Catalog No. A13423
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    Integrin receptor antagonist
    GLPG0187 is a broad spectrum integrin receptor antagonist with antitumor activity; inhibits αvβ1-integrin with an IC50 of 1.3 nM. 了解更多
  12. LED209

    Catalog No. A12219
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    bacterial receptor QseC inhibitor
    LED209 is a potent small molecule inhibitor of bacterial receptor QseC, is a potent prodrug that is highly selective for QseC. 了解更多
  13. GV-196771A

    Catalog No. A13438
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    NMDA receptor antagonist
    GV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多
  14. Tiotropium Bromide

    Catalog No. A10934
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    muscarinic acetylcholine receptor (mAChR) antagonist
    Tiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多
  15. Valsartan

    Catalog No. A10962
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    angiotensin II receptor antagonist
    Valsartan (CGP-48933) is an angiotensin II receptor antagonist for the treatment of high blood pressure and heart failure. 了解更多
  16. Zafirlukast

    Catalog No. A11004
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    LTD4 receptor antagonist
    Zafirlukast is a potent orally active leukotriene D4 (LTD4) receptor antagonist. 了解更多
  17. Ziprasidone hydrochloride monohydrate

    Catalog No. A11008
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    5-HT (serotonin) and dopamine receptor antagonist
    Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  18. Acamprosate calcium

    Catalog No. A11308
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    GABA receptor agonist
    Acamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. 了解更多
  19. Sitaxsentan

    Catalog No. A11565
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    ETA receptor antagonist
    Sitaxsentan (IPI 1040; TBC-11251) is a selective endothelin A (ETA) receptor antagonist. Antihypertensive. Sitaxsentan is used in treatment of chronic heart failure. 了解更多
  20. Elacestrant

    Catalog No. A12244
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    Estrogen receptor degrader
    Elacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively. 了解更多
  21. DW-1350

    Catalog No. A12250
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    LTB4 receptor antagonist
    DW-1350 is a LTB4 receptor antagonist. 了解更多
  22. PRX933 hydrochloride

    Catalog No. A12261
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    5-HT2c receptor agonist
    PRX933 hydrochloride is a 5-HT2c receptor agonist extracted from patent WO 2014140631 A1. 了解更多
  23. AC260584

    Catalog No. A12264
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    M1 muscarinic receptor allosteric agonist
    AC260584 is an M1 muscarinic receptor allosteric agonist with a pEC50 of 7.6. 了解更多
  24. TY-52156

    Catalog No. A12265
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    S1P3 receptor antagonist
    TY-52156 is a potent and selective S1P3 receptor antagonist with a Ki value of 110 nM. 了解更多
  25. 5-HT4 antagonist 1

    Catalog No. A12268
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    5-HT4 receptor antagonist
    5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6. 了解更多
  26. lumateperone Tosylate

    Catalog No. A12279
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    5-HT2A receptor antagonist
    Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM). 了解更多
  27. AP521

    Catalog No. A12280
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    human 5-HT1A receptor agonist
    AP521 is an agonist of human 5-HT1A receptor with an IC50 of 94 nM. 了解更多
  28. CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  29. Pipequaline

    Catalog No. A12551
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    partial benzodiazepine receptor agonist
    Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. 了解更多
  30. Endothelin Mordulator 1

    Catalog No. A13040
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    endothelin receptor modulator
    Endothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders. 了解更多
  31. Veralipride

    Catalog No. A13132
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    D2 receptor antagonist
    Veralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. 了解更多
  32. ZD-1611

    Catalog No. A13151
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    ETA receptor antagonist
    ZD-1611 is a potent, orally active, selective ETA receptor antagonist, used for the research of ischemic stroke. 了解更多
  33. Chlorantraniliprole

    Catalog No. A13214
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    Chlorantraniliprole is an insecticide that potently and selectively activates insect ryanodine receptor, with EC50s of 40 nM and 50 nM for Drosophila melanogaster and H. virescens ryanodine receptor, and ?300-fold more potent than that in the mouse myoblast cell line, C2C12 (EC50, 14 μM). 了解更多
  34. BW 245C

    Catalog No. A13494
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    prostanoid DP-receptor (DP1) agonist
    BW 245C is a prostanoid DP-receptor (DP1) agonist, used to treat stroke. 了解更多
  35. SL910102

    Catalog No. A13591
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    Angiotensin AT1 receptor antagonist
    SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. 了解更多
  36. SX-3228

    Catalog No. A13687
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    benzodiazepine1 (BZ1) receptor agonist
    SX-3228 is a selective benzodiazepine1 (BZ1) receptor agonist with an IC50 of 17 nM. 了解更多
  37. GSK598809

    Catalog No. A13695
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    dopamine D3 Receptor (DRD3) antagonist
    GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist, with a pKi of 8.9. 了解更多
  38. VU6001376

    Catalog No. A13763
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    metabotropic glutamate receptor 4 modulator
    VU6001376 is a potent and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu4 PAM) with an EC50 of 50.1 nM. 了解更多
  39. Mozavaptan

    Catalog No. A16622
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    nonpeptide vasopressin V2 receptor antagonist
    Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM. 了解更多
  40. Sarcosine

    Catalog No. A16692
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    GlyT inhibitor/NMDA receptor
    Sarcosine is a glycine transporter type 1 (GlyT) inhibitor and an N-methyl-D-aspartate (NMDA) receptor co-agonist at the glycine binding site. 了解更多
  41. Tripelennamine hydrochloride

    Catalog No. A16767
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    H1-receptor antagonist
    Tripelennamine hydrochloride, a H1-receptor antagonist, is a psychoactive drug and member of the pyridine andethylenediamine classes that is used as an antipruritic and first-generation antihistamine. 了解更多
  42. Pirenzepine dihydrochloride

    Catalog No. A17916
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    M1 muscarinic receptor antagonist
    Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist. 了解更多
  43. Norepinephrine

    Catalog No. A11306
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    β1-selective adrenergic receptor agonist
    Norepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  44. CAY10471 Racemate

    Catalog No. A11760
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    Prostaglandin D2 receptor CRTH2 antagonist
    CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多
  45. CP-809101

    Catalog No. A12481
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    5-HT2C receptor agonist
    CP-809101 is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively. 了解更多
  46. MK-6913

    Catalog No. A12311
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    Estrogen receptor β agonist
    Tetrahydrofluoroene 52 is a potent and selective estrogen receptor β agonist. 了解更多
  47. 4-IBP

    Catalog No. A12314
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    σ1 激动剂
    4-IBP is a selective ??1 agonist with a high level of affinity for the ??1 receptor (Ki = 1.7 nM) and a moderate affinity for the ??2 receptor (Ki = 25.2 nM) . 了解更多
  48. Darenzepine

    Catalog No. A12333
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    muscarinic receptor inhibitor
    Darenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多
  49. MRK-016

    Catalog No. A12046
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    GABAA α5 receptor agonist
    MRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多
  50. Tecadenoson

    Catalog No. A13302
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    A1 adenosine receptor agonist
    Tecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. 了解更多

产品 551 到 600 共 1712个

每页
页面:
  1. 10
  2. 11
  3. 12
  4. 13
  5. 14

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