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Lu AF21934
Catalog No. A12140 mGlu4 receptor modulatorLu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多 -
Beperidium iodide
Catalog No. A12382 competitive antagonistic effect against acetylcholine receptorBeperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93. 了解更多 -
GSK1059865
Catalog No. A12401 -
Dexamethasone palmitate
Catalog No. A18453 Dexamethasone palmitate (DXP) is a prodrug of Dexamethasone, which is a glucocorticoid receptor agonist. Dexamethasone palmitate (DXP) has a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Anti-inflammatory agent. 了解更多 -
ROR agonist-1
Catalog No. A18569 ROR 激动剂ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多 -
PROTAC ERRα Degrader-2
Catalog No. A18904 ERRa degraderPROTAC ERRalpha Degrader-2 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRalpha Degrader-2 is an estrogen-related receptor alpha (ERRa) degrader. 了解更多 -
PROTAC ERRα Degrader-1
Catalog No. A18910 ERRα DegraderPROTAC ERRα Degrader-1 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRα Degrader-1 is an estrogen-related receptor alpha (ERRa) degrader. 了解更多 -
AZD2906
Catalog No. A18936 glucocorticoid receptor agonistAZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. 了解更多 -
PF-05231023
Catalog No. A18949 FGF21-receptor agonistPF-05231023, a long-acting fibroblast growth factor 21 (FGF21) analog, is a FGF21-receptor agonist, suitable for development as a potential treatment for T2DM. 了解更多 -
GSK1521498 free base
Catalog No. A18994 μ-opioid receptor antagonistGSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多 -
Asoprisnil
Catalog No. A19030 Progesterone receptor modulatorAsoprisnil (J867), a selective progesterone receptor modulator, exhibits mixed progesterone agonist and antagonist effects on various progesterone targeted tissues in animal and human. 了解更多 -
Apelin agonist 1
Catalog No. A19035 apelin agonistApelin agonist 1 is an oral selective apelin agonist AM-2995, a agonist of the APJ (APLNR, angiotensin receptor like-1) receptor, may be used in the treatment of cardiovascular conditions. 了解更多 -
STING agonist-4
Catalog No. A19074 STING receptor agonistSTING agonist-4 is an stimulator of Interferon Genes (STING) receptor agonist with an apparent inhibitory constant (IC50) of 20 nM. 了解更多 -
S18-000003
Catalog No. A19105 RORγt 抑制剂S18-000003 is a potent orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t (RORγt) inhibitor with an IC50 of 29 nM. S18-000003 inhibits IL-17 production. 了解更多 -
Balovaptan
Catalog No. A19373 hV1a receptor antagonistBalovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism. 了解更多 -
Alosetron (Hydrochloride(1:X))
Catalog No. A11309 Serotonin 5HT3-receptor antagonistAlosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多 -
JTE-952
Catalog No. A18391 CSF-1R 抑制剂TE-952 is a potent, oral active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), with IC50 values of 13 nM and 261 nM for CSF1R and TrkA , respectively. Effective against a mouse collagen-induced model of arthritis. 了解更多 -
Dexloxiglumide
Catalog No. A18541 CCKA receptor antagonistDexloxiglumide is a selective cholecystokinin type A (CCKA) receptor antagonist. Dexloxiglumide, the active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). 了解更多 -
BTRX-335140
Catalog No. A18583 κ opioid receptor antagonistBTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. 了解更多 -
FGFR1/DDR2 inhibitor 1
Catalog No. A18716 FGFR1/DDR2 inhibitorFGFR1/DDR2 inhibitor 1 is an inhibitor of fibroblast growth factor receptor 1 (FGFR1) and discoindin domain receptor 2 (DDR2), with IC50 values of 31.1 nM, 108.4 nM and 3.2 nM for FGFR1, KG-1, and DDR2, respectively. 了解更多 -
PF-06256142
Catalog No. A18872 D1 receptor agonistPF-06256142 is a potent and selective orthosteric agonist of the D1 receptor, with D1 EC50=30 nM and D1 binding Ki = 12 nM. 了解更多 -
Tulobuterol hydrochloride
Catalog No. A18226 β2-adrenergic receptor agonistTulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多 -
Glycerol phenylbutyrate
Catalog No. A18201 sigma-2 (σ2) receptor ligandGlycerol phenylbutyrate is a sigma-2 (σ2) receptor ligand, with a pKi of 8.02. 了解更多 -
Lofexidine
Catalog No. A18151 α2-receptor agonistLofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal. 了解更多 -
Lasofoxifene Tartrate
Catalog No. A18097 selective Estrogen receptor modulatorLasofoxifene tartrate is a third-generation selective estrogen receptor modulator. 了解更多 -
Lusutrombopag
Catalog No. A18089 thrombopoietin (TPO) receptor agonistLusutrombopag, also known as S-888711, is an orally bioavailable, small molecule thrombopoietin (TPO) receptor agonist being developed by Shionogi for chronic liver disease (CLD) patients with thrombocytopenia prior to elective invasive surgery. 了解更多 -
Metipranolol hydrochloride
Catalog No. A18064 β-adrenergic receptor antagonistMetipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多 -
Mebhydrolin napadisylate
Catalog No. A17997 -
Leuprorelin Acetate
Catalog No. A17986 GnRH/LHRH receptor agonistLeuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. 了解更多
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