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￥ 0.00 “glucagon receptor”的搜索结果
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JNJ-63576253
Catalog No. A22530 TRC253, also known as JNJ63576253, is a potent and orally active androgen receptor antagonist. 了解更多 -
MK-212 HCl
Catalog No. A22531 MK 212 hydrochloride is a 5-HT receptor agonist; displays selectivity for 5-HT2C over 5-HT2A (IC50 values are 0.028 and 0.42 μM for human 5-HT2C and 5-HT2A receptors expressed in HEK293 cells respectively). 了解更多 -
JNJ-10198409
Catalog No. A22554 PDGFRα/PDGFRβ inhbitorJNJ 10198409 is a potent platelet-derived growth factor receptor (PDGFR) inhibitor (IC50 values are 4.2 and 45 nM for PDGFRβ and PDGFRα, respectively). Also inhibits c-Abl, Lck, c-Src and Fyn kinases (IC50 values are 22, 100, 185 and 378 nM respectively). 了解更多 -
M8-B (hydrochloride)
Catalog No. A22607 TRPM8 antagonistM8-B is an antagonist of transient receptor potential melastatin 8 (TRPM8) that blocks activation by cold, icilin (Item No. 10137), or menthol in vitro (IC50s = 7.8, 26.9, and 64.3 nM, respectively). 了解更多 -
Triptorelin
Catalog No. A22621 GnRH peptide agonistTriptorelin is a synthetic gonadotropin-releasing hormone (GnRH) peptide agonist that binds to the GnRH receptor. It inhibits the growth of DU145, LNCaP, and PC3 prostate and OVCAR-3 ovarian cancer cells. 了解更多 -
BLT-1
Catalog No. A22704 type 1 (SR-BI) inhibitorBLT-1, a thiosemicarbazone copper chelator, is a selective scavenger receptor B, type 1 (SR-BI) inhibitor. BLT-1 inhibits the transfer of lipids between high-density lipoproteins (HDL) and cells mediated by SR-BI. BLT-1 is a potent HCV entry inhibitor. 了解更多 -
NSC-703786 (5F-203)
Catalog No. A22708 NSC-703786 (5F-203) is a cytotoxic molecule that forms DNA adducts leading to cell death. NSC-703786 induces aryl hydrocarbon receptor signaling, and elevates expression of CYP1A1. Treatment of cells with NSC-703786 also leads to elevation of reactive oxygen species and activation of p38, JNK and ERK. 了解更多 -
Tyrphostin AG1296
Catalog No. A16773 PDGFR inhibitorTyrphostin AG1296 is a potent and selective inhibitor of platelet-derived growth factor receptor (PDGFR), with an IC50 of 0.8 μM. 了解更多 -
Avobenzone
Catalog No. A11818 estrogen agonistAvobenzone, a dibenzoylmethane compound, is one of the most widely used filters in sunscreens for skin photoprotection in the UVA band. Avobenzone is an endocrine disruptor that directly binds to estrogen receptor β and acts as an estrogen agonist. 了解更多 -
Blarcamesine (AVex-73)
Catalog No. A21095 muscarinic M1 agonistBlarcamesine, also known as AVex-73 and AE-37, is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease. It is an σ receptor ligand. 了解更多 -
Pridopidine
Catalog No. A22009 D2R antagonistPridopidine, a dopamine (DA) stabilizer, acts as a low affinity dopamine D2 receptor (D2R) antagonist. 了解更多 -
Calcitriol Impurities D
Catalog No. A20825 impurity of CalcitriolCalcitriol Impurities D is the impurity of Calcitriol, Calcitriol is the hormonally active form of vitamin D, Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor (VDR). 了解更多 -
GSK2798745
Catalog No. A20799 TRPV4 ion channel blockerGSK2798745 is a first-in-class, highly potent, selective, orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively. 了解更多 -
WAY-204688
Catalog No. A20757 NF-κB inhibitorWAY-204688 is an estrogen receptor (ER-α) selective, orally active inhibitor of NF-κB transcriptional activity with an IC50 of 122?±?30 nM for NF-κB-luciferase (NF-κB-luc) in HAECT-1 cells. 了解更多 -
GSK180736A
Catalog No. A20736 GRK2 inhibitorGSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM. 了解更多 -
Fezolinetant
Catalog No. A20706 NK3R antagonistFezolinetant is an antagonist of the neurokinin 3 receptor (NK3R), used for the treatment of menopausal hot flushes. 了解更多 -
Setmelanotide
Catalog No. A20689 MC4R agonistSetmelanotide (RM-493; BIM-22493; IRC-022493) is a selective melanocortin 4 receptor (MC4R) agonist with EC50s of 0.27 nM and 0.28 nM for human and rat MC4R, respectively. 了解更多 -
CCR2-RA-[R]
Catalog No. A20644 CCR2 antagonistCCR2-RA-[R] is an allosteric antagonist of the C-C chemokine receptor type 2 (CCR2) with an IC50 of 103 nM. 了解更多 -
Saroglitazar
Catalog No. A20636 PPAR agonistSaroglitazar is a novel peroxisome proliferator-activated receptor (PPAR) agonist with predominant PPARα and moderate PPARγ activity with EC50 values of 0.65 pM and 3 nM in HepG2 cells, respectively. 了解更多 -
Calcitriol Impurities A
Catalog No. A20633 Calcitriol Impurities A is the impurity of Calcitriol, Calcitriol is the hormonally active form of vitamin D, Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor (VDR). 了解更多 -
Azeliragon
Catalog No. A20622 RAGE inhibitorAzeliragon (TTP488) is an orally bioavailable inhibitor of the receptor for advanced glycation end products (RAGE) in development as a potential treatment to slow disease progression in patients with mild Alzheimer??s disease (AD). Azeliragon also can cross the blood-brain barrier (BBB). 了解更多 -
GSK682753A
Catalog No. A20519 EBI2 inverse agonistGSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2) with an IC50 of 53.6 nM. 了解更多 -
Mivotilate
Catalog No. A20504 AhR activatorMivotilate is a nontoxic, potent activator of the aryl hydrocarbon receptor (AhR), and acts as a hepatoprotective agent. 了解更多 -
Agmatine sulfate
Catalog No. A20485 NO synthase inhibitorAgmatine sulfate exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide synthesis. It is an endogenous agonist at imidazoline receptor and a NO synthase inhibitor. 了解更多 -
CCR2 antagonist 3
Catalog No. A20467 -
(-)-(S)-Equol
Catalog No. A20465 (-)-(S)-Equol is a high affinity ligand for estrogen receptor β with a Ki of 0.73 nM. 了解更多 -
Trifarotene
Catalog No. A20458 RAR agonistTrifarotene (CD5789) is a retinoic acid receptor (RAR) agonist with Kdapp of 2, 15 and 500 nM for RARγ, RARβ and RARα, respectively. 了解更多 -
TCS-OX2-29
Catalog No. A20457 OX2R antagonistTCS-OX2-29 is a potent, high affinities and selective orexin-2 receptor (OX2R) antagonist with an IC50 value of 40 nM and a pKI value of 7.5. TCS-OX2-29 displays ~250-fold selectivity for OX2 over OX1. 了解更多
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