“alpha ergocryptine”的搜索结果

产品 51 到 100 共 642个

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  1. MRK-016

    Catalog No. A12046
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    GABAA α5 receptor agonist
    MRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多
  2. MAC glucuronide α-hydroxy lactone-linked SN-38

    Catalog No. A18407
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    Topoisomerase I inhibitor
    MAC glucuronide α-hydroxy lactone-linked SN-38 (Topoisomerase I inhibitor) is a stabilized lactone MAC glucuronide α-hydroxy lactone-linked SN-38 drug linker. 了解更多
  3. Alpha-Naphthoflavone

    Catalog No. A18474
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    aromatase inhibitor
    Alpha-Naphthoflavone is a synthetic flavonoid, acts as a potent and competitive aromatase inhibitor with an IC50 and a Ki of 0.5 and 0.2 μM, respectively. 了解更多
  4. PROTAC ERRα Degrader-2

    Catalog No. A18904
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    ERRa degrader
    PROTAC ERRalpha Degrader-2 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRalpha Degrader-2 is an estrogen-related receptor alpha (ERRa) degrader. 了解更多
  5. (+)-α-Tocopherol

    Catalog No. A17407
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    alpha-Tocopherol is one of the most abundant isoforms of vitamin E. alpha-Tocopherol is a biologically active liposoluble vitamin and potent antioxidant. 了解更多
  6. (+)-α-Lipoic acid

    Catalog No. A17343
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    Lipoic Acid, also known as R-(+)-alpha-Lipoic acid, is an organosulfur compound derived from octanoic acid. It is made in animals normally, and is essential for aerobic metabolism. It is also manufactured and is available as a dietary supplement in some countries where it is marketed as an antioxidant, and is available as a pharmaceutical drug in other countries. 了解更多
  7. Pifithrin-alpha

    Catalog No. A12451
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    p53 抑制剂
    Pifithrin-alpha是p53介导的细胞凋亡和p53依赖性基因转录(如细胞周期蛋白G,p21/waf1和mdm2表达)的可逆抑制剂。 了解更多
  8. 17 alpha-propionate

    Catalog No. A10009
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    Androgen 拮抗剂
    17 alpha-propionate是一种新型的局部和外周选择性雄激素拮抗剂。 了解更多
  9. EB-3D

    Catalog No. A22288
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    choline kinase α (ChoKα) inhibitor
    EB-3D is a potent and selective choline kinase α (ChoKα) inhibitor, with an IC50 of 1 μM for ChoKα1. 了解更多
  10. Estrone-N-O-C1-amido

    Catalog No. A19746
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    estrogen ligand
    Estrone-N-O-C1-amido (ERα ligand 1) is an Estrone-based estrogen ligand, which targets estrogen receptor α (ERα). Estrone-N-O-C1-amido (ERα ligand 1) binds to cIAP1 ligand Bestatin via a linker to form SNIPER. 了解更多
  11. 5α-Cholestan-3β-ol

    Catalog No. A19653
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    5α-Cholestan-3β-ol is a derivitized steroid compound, which is isolated from the testes of White Carneau pigeons. 了解更多
  12. N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride

    Catalog No. A19540
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    protease inhibitor
    N-alpha-Tosyl-L-lysine chloromethyl ketone (TLCK), a trypsin like protease inhibitor, sensitizes HeLa cells to Fas-mediated cell death. 了解更多
  13. NS11394

    Catalog No. A21425
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    GABA(A) receptor modulator
    NS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors. 了解更多
  14. Tesaglitazar

    Catalog No. A20891
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    PPAR alpha/gamma agonist
    Tesaglitazar is a dual peroxisome proliferator-activated receptor (PPAR) alpha/gamma agonist that is more potent on PPARγ than on PPARα, with EC50s of 13.4 μM and 3.6 μM for rat PPARα and human PPARα, respectively. 了解更多
  15. AGN 192836

    Catalog No. A13013
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    α2 adrenergic agonist
    AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. 了解更多
  16. Vitamin E Acetate

    Catalog No. A17284
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    D-α-Tocopherol acetate (D-Vitamin E acetate) can be hydrolyzed to d-alpha-tocopherol (VE) and absorbed in the small intestine. 了解更多
  17. α-Estradiol

    Catalog No. A17082
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    Alpha-Estradiol是一种内源性雌激素受体配体(ERα和ERβ受体的Ki值分别为0.2和1.2 nM)。 了解更多
  18. 18α-Glycyrrhetinic acid

    Catalog No. A12199
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    The aglycone of glycyrrhizin
    18α-Glycyrrhetinic acid是甘草中发现的一种生物活性三萜类化合物。它显示对11-hs D1(11-羟基类固醇脱氢酶1)的选择性抑制。 了解更多
  19. TNF alpha human

    Catalog No. AP5560
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    Tumor Necrosis Factor-Alpha Human Recombinant 了解更多
  20. IL 1 alpha Rat, His

    Catalog No. AP5482
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    Interleukin-1 alpha Rat Recombinant, His Tag 了解更多
  21. IL 1 alpha Mouse, His

    Catalog No. AP5463
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    Interleukin-1 alpha Mouse Recombinant, His Tag 了解更多
  22. IL 1 alpha Rhesus Macaque

    Catalog No. AP5454
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    Interleukin-1 alpha Rhesus Macaque Recombinant 了解更多
  23. IL 1 alpha Mouse

    Catalog No. AP5400
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    Interleukin-1 alpha Mouse Recombinant 了解更多
  24. IL 1 alpha Human, His

    Catalog No. AP5385
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    Interleukin-1 alpha Human Recombinant, His Tag 了解更多
  25. IL 1 alpha Porcine

    Catalog No. AP5375
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    Interleukin-1 alpha Porcine Recombinant 了解更多
  26. IL 1 alpha Rat

    Catalog No. AP5366
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    Interleukin-1 alpha Rat Recombinant 了解更多
  27. IL 1 alpha Human

    Catalog No. AP5341
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    Interleukin-1 alpha Human Recombinant 了解更多
  28. PKAR-I alpha Human

    Catalog No. AP4568
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    Protein Kinase A regulatory subunit-1 alpha Human Recombinant 了解更多
  29. Inhibin alpha A Chain Human

    Catalog No. AP3262
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    Inhibin-Alpha A Chain Human Recombinant 了解更多
  30. HSP90 Alpha Antibody

    Catalog No. AP2838
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    Heat shock protein HSP 90-alpha, Mouse Anti Human 了解更多
  31. CEBP Alpha Human

    Catalog No. AP1883
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    CCAAT/enhancer binding protein CEBP Alpha Human Recombinant 了解更多
  32. Gliadin Alpha Wheat

    Catalog No. AP1395
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    Gliadin Alpha Wheat Recombinant 了解更多
  33. HSP90 Alpha Human

    Catalog No. AP0084
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    Heat Shock Protein-90 Alpha Human Recombinant 了解更多
  34. PI3K-alpha inhibitor 1

    Catalog No. A16274
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    PI3Kα 抑制剂
    PI3K-alpha inhibitor 1 是从专利US/20120088764A1中提取的PI3Kα抑制剂,化合物243,IC50 <0.1uM,PI3Kα抑制剂1还抑制HDAC(0.1uM≤IC50≤1uM)。 了解更多
  35. Cimigenol-3-O-alpha-L-arabinoside

    Catalog No. A15407
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    Cimigenol-3-O-alpha-L-阿拉伯糖苷是从Cimicifuga foetida L.干燥的根茎中提取的。 了解更多
  36. alpha-hederin

    Catalog No. A15399
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    alpha-hederin一种从常春藤提取的皂苷。 了解更多
  37. alpha-Hederin

    Catalog No. A14614
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    alpha-Hederin提取自海葵银莲花。 了解更多
  38. alpha-Amyloid Precursor Protein Modulator

    Catalog No. A13094
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    α-淀粉样前体蛋白调节剂是细胞可渗透的苯并内酰胺衍生的PKC激活剂(PKCα的Ki = 11.9 nM),即使在人类原纤维中为100 nM时,也能有效增强淀粉样前体蛋白(APP)的非淀粉样生成性α-加工。 了解更多
  39. MN58b

    Catalog No. A22129
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    choline kinase α (CHKα) inhibitor
    MN58b is a selective choline kinase α (CHKα) inhibitor, and results in inhibition of phosphocholine synthesis. 了解更多
  40. Cholesterol

    Catalog No. A22211
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    endogenous estrogen-related receptor α (ERRα) agonist
    Cholesterol is also an endogenous estrogen-related receptor α (ERRα) agonist. 了解更多
  41. Zaurategrast ethyl ester

    Catalog No. A20624
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    α4β1/α4β7 integrin antagonist
    Zaurategrast ethyl ester (CDP323), the ethyl ester prodrug of CT7758, is a α4β1/α4β7 integrin antagonist used for the treatment of inflammatory and autoimmune disorders. 了解更多
  42. N-Nonyldeoxynojirimycin

    Catalog No. A19963
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    alpha-glucosidase/alpha-1,6-glucosidase inhibitor
    N-Nonyldeoxynojirimycin (NN-DNJ) is a potent inhibitor of alpha-glucosidase and alpha-1,6-glucosidase (IC50s, 0.42, 8.4 μM, respectively), inhibits glycogen breakdown. 了解更多
  43. M1001

    Catalog No. A19443
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    HIF-2α agonist
    M1001 is a weak agonist of HIF-2α, directly binds to the HIF-2α PAS-B domain, with a Kd of 667 nM. M1001 enhances the stabilities of HIF-2α-ARNT complex. 了解更多
  44. Pozanicline

    Catalog No. A21318
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    Pozanicline (ABT-089) selectively activate neuronal nicotinic acetylcholine receptor (nAChR) subtypes, is a novel cholinergic agent that is a partial agonist at α4β2* nAChRs (Ki=16 nM) and shows high selectivity for α6β2* and α4α5β2 nAChR subtypes, the binding affinity (Ki, rat) for Pozanicline to [3H] cytisine sites is 16.7 nM. 了解更多
  45. CCMI

    Catalog No. A21534
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    α7 nAChR-positive allosteric modulator
    CCMI is a potent and selective α7 nAChR-positive allosteric modulator, does not bind to or activate α7 nAChRs via the orthosteric site, and causes significant positive modulation of agonist-induced currents at α7 nAChRs. 了解更多
  46. Asenapine

    Catalog No. A18010
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    adrenergic receptor inhibitor
    Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. 了解更多
  47. (+)-Cloprostenol

    Catalog No. A12979
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    prostaglandin F2α (PGF2α) analogue
    (+)-Cloprostenol is a prostaglandin F2α (PGF2α) analogue, and shows selective agonistic activity at the prostaglandin receptor. 了解更多
  48. Medetomidine

    Catalog No. A11494
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    α2-adrenoceptor agonist
    Medetomidine(Domtor) is a potent, highly selective α2-adrenoceptor agonist (Ki values are 1.08 and 1750 nM for α2- and α1-adrenoceptors respectively). 了解更多
  49. OPC-28326

    Catalog No. A12762
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    α2-adrenergic receptor angatonist
    OPC-28326 is a selective peripheral vasodilator and an angatonist of α2-adrenergic receptor, with Ki of 2040, 285, and 55?nM for α2A-, α2B- and α2C-adrenoceptors, respectively. 了解更多
  50. TPA 023

    Catalog No. A20140
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    GABAA α2/α3 agonist
    TPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM. 了解更多

产品 51 到 100 共 642个

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