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￥ 0.00 “AG 013736”的搜索结果
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GSK1521498
Catalog No. A20649 μ-opioid receptor (MOR) antagonistGSK1521498 is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多 -
Adomeglivant
Catalog No. A20647 glucagon receptor antagonistAdomeglivant is a potent and selective glucagon receptor antagonist that is used in clinical trial for type 2 diabetes mellitus. 了解更多 -
6-Amino-5-nitropyridin-2-one
Catalog No. A20646 6-Amino-5-nitropyridin-2-one is a pyridine base and used as a nucleobase of hachimoji DNA, in which it pairs with 5-aza-7-deazaguanine. 了解更多 -
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CCR2-RA-[R]
Catalog No. A20644 CCR2 antagonistCCR2-RA-[R] is an allosteric antagonist of the C-C chemokine receptor type 2 (CCR2) with an IC50 of 103 nM. 了解更多 -
BMS-779788
Catalog No. A20640 LXR partial agonistBMS-779788 is a LXR partial agonist with IC50 values of 68 nM for LXRα and 14 nM for LXRβ. 了解更多 -
Saroglitazar
Catalog No. A20636 PPAR agonistSaroglitazar is a novel peroxisome proliferator-activated receptor (PPAR) agonist with predominant PPARα and moderate PPARγ activity with EC50 values of 0.65 pM and 3 nM in HepG2 cells, respectively. 了解更多 -
PF-06291874
Catalog No. A20635 glucagon receptor antagonistPF-06291874 (Glucagon receptor antagonists-4) is a highly potent and orally active glucagon receptor antagonist. It displays low in vivo clearance in both rats and dogs. 了解更多 -
Azetidine-2-carboxylic acid
Catalog No. A20628 Azetidine-2-carboxylic acid is a non proteinogenic amino acid homologue of proline. Found in common beets. Azetidine-2-carboxylic acid can be misincorporated into proteins in place of proline in many species, including humans. Toxic and teratogenic agent. 了解更多 -
Zaurategrast ethyl ester
Catalog No. A20624 α4β1/α4β7 integrin antagonistZaurategrast ethyl ester (CDP323), the ethyl ester prodrug of CT7758, is a α4β1/α4β7 integrin antagonist used for the treatment of inflammatory and autoimmune disorders. 了解更多 -
Azeliragon
Catalog No. A20622 RAGE inhibitorAzeliragon (TTP488) is an orally bioavailable inhibitor of the receptor for advanced glycation end products (RAGE) in development as a potential treatment to slow disease progression in patients with mild Alzheimer??s disease (AD). Azeliragon also can cross the blood-brain barrier (BBB). 了解更多 -
TAK-220
Catalog No. A20618 -
Asparagusic acid
Catalog No. A20607 Asparagusic acid (1,2-dithiolane-4-carboxylic acid) is unique to asparagus. The compound is responsible for the odorous urine excreted after eating asparagus. Its derivatives ihydroasparagusic acid have anti-inflammatory effect. 了解更多 -
3-Bromopyruvic acid
Catalog No. A20605 hexokinase II inhibitor3-Bromopyruvic acid is a hexokinase II inhibitor, is an effective antitumor agent on the hepatoma cells. 了解更多 -
Taprenepag isopropyl
Catalog No. A20604 EP2 receptor agonistTaprenepag isopropyl is a highly selective EP2 receptor agonist. 了解更多 -
10-Deacetyl-7-xylosyl paclitaxel
Catalog No. A20602 10-Deacetyl-7-xylosyl paclitaxel is a Paclitaxel (a microtubule stabilizing agent; enhances tubulin polymerization) derivative with improved pharmacological features. 了解更多 -
LX2761
Catalog No. A20597 SGLT1/SGLT2 inhibitorLX2761 is chemically stable and potent inhibitor against sodium-dependent glucose cotransporter 1 (SGLT1) and SGLT2 in vitro with IC50s of 2.2 nM and 2.7nM for hSGLT1 and hSGLT2, but displays specific SGLT1 inhibition in the gastrointestinal (GI) tract. 了解更多 -
L-Cysteinesulfinic acid
Catalog No. A20585 metabotropic glutamate receptors agonistL-Cysteinesulfinic acid is a potent agonist at several rat metabotropic glutamate receptors (mGluRs) with pEC50s of 3.92±0.03, 4.6±0.2, 3.9±0.2, 2.7±0.2, 4.0±0.2, and 3.94±0.08 for mGluR1, mGluR5, mGluR2, mGluR4, mGluR6, and mGluR8, respectively. 了解更多 -
Bicyclomycin benzoate
Catalog No. A20581 Bicyclomycin benzoate is an antibiotic exhibiting activity against a broad spectrum of Gram-negative bacteria and against the Gram-positive bacterium. 了解更多 -
Quinolinic acid
Catalog No. A20575 NMDA receptor agonistQuinolinic acid is an endogenous N-methyl-D-aspartate (NMDA) receptor agonist synthesized from L-tryptophan via the kynurenine pathway and thereby has the potential of mediating N-methyl-D-aspartate neuronal damage and dysfunction. 了解更多 -
Dansyl glutathione
Catalog No. A20573 Dansyl glutathione is a trapping agent for the quantitative estimation and identification of reactive metabolites. 了解更多 -
Allopurinol riboside
Catalog No. A20572 Allopurinol riboside, a metabolite of allopurinol, shows potent activities against parasites. 了解更多 -
sulfo-SPDB-DM4
Catalog No. A20566 sulfo-SPDB-DM4 is a drug-linker conjugate for ADC by using the maytansinebased payload (DM4, an antitubulin agent) via the sulfo-SPDB linker. 了解更多 -
Isoguvacine hydrochloride
Catalog No. A20563 -
JNJ16259685
Catalog No. A20545 mGlu1 receptor antagonistJNJ16259685 is a selective antagonist of mGlu1 receptor, and inhibits the synaptic activation of mGlu1 in a concentration-dependent manner with IC50 of 19 nM. 了解更多 -
Naltrindole hydrochloride
Catalog No. A20541 δ opioid receptor antagonistNaltrindole hydrochloride is a highly potent and selective non-peptide δ opioid receptor antagonist with a Ki of 0.02 nM. 了解更多 -
MMAF-OMe
Catalog No. A20540 -
DREADD agonist 21
Catalog No. A20534 hM3Dq agonist.DREADD agonist 21 is a potent human muscarinic acetylcholine M3 receptors (hM3Dq) agonist(EC50=1.7 nM). 了解更多 -
Nicotinamide N-oxide
Catalog No. A20532 CXCR2 receptor antagonistNicotinamide N-oxide, an in vivo nicotinamide metabolite, is a potent, and selective antagonist of the CXCR2 receptor. 了解更多 -
Linaprazan
Catalog No. A20526 Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding. (IC50: 1.0 ± 0.2 μM) It is a acid-suppressing agents with rapid onset of action and potent acid inhibition. 了解更多 -
GSK682753A
Catalog No. A20519 EBI2 inverse agonistGSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2) with an IC50 of 53.6 nM. 了解更多 -
Mivotilate
Catalog No. A20504 AhR activatorMivotilate is a nontoxic, potent activator of the aryl hydrocarbon receptor (AhR), and acts as a hepatoprotective agent. 了解更多 -
Sarmazenil
Catalog No. A20487 benzodiazepine receptor antagonistSarmazenil is a benzodiazepine receptor antagonist. 了解更多 -
Oxaquin
Catalog No. A20486 Oxaquin (MCB-3837) is a water-soluble, injectable prodrug that is rapidly converted to the active sub-stance MCB3681 in vivo following intravenous (i.v.) administration, active against Gram-positive bacterial species. Oxaquin (MCB-3837) itself has no antimicrobial effects. 了解更多
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