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￥ 0.00 “glucagon receptor”的搜索结果
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GSK189254A
Catalog No. A22005 histamine H3 receptor antagonistGSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. 了解更多 -
Aripiprazole (D8)
Catalog No. A22004 human 5-HT1A receptor partial agonistAripiprazole D8 (OPC-14597 D8) is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. 了解更多 -
Carotegrast
Catalog No. A21997 α4 integrin receptor inhibitorCarotegrast is an orally available α4 integrin receptor inhibitor with anti-inflammatories activities. 了解更多 -
Amisulpride hydrochloride
Catalog No. A21994 dopamine D2/D3 receptor antagonistAmisulpride hydrochloride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively. 了解更多 -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. 了解更多 -
Ziprasidone D8
Catalog No. A21989 5-HT / dopamine receptor antagonistZiprasidone D8 is deuterium labeled Ziprasidone, which is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多 -
Eplivanserin mixture
Catalog No. A21987 serotonin reuptake inhibitor/5-HT2A receptor antagonistEplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多 -
Ro 10-5824 dihydrochloride
Catalog No. A21986 dopamine D4 receptor partial agonistRo 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多 -
Niperotidine
Catalog No. A21981 histamine H2-receptor antagonistNiperotidine is a histamine H2-receptor antagonist. 了解更多 -
Ritanserin
Catalog No. A21976 5-HT2 receptor antagonistRitanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. 了解更多 -
Haloperidol D4'
Catalog No. A21971 dopamine D2 receptor antagonistHaloperidol D4' is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. 了解更多 -
Atenolol
Catalog No. A21962 -
Haloperidol D4
Catalog No. A21961 dopamine D2 receptor antagonistHaloperidol D4 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. 了解更多 -
Mapracorat
Catalog No. A21953 glucocorticoid receptor agonistMapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. 了解更多 -
MT-7716 free base
Catalog No. A21928 non-peptide nociceptin receptor (NOP) agonistMT-7716 free base (W-212393) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. 了解更多 -
SB-224289 hydrochloride
Catalog No. A21920 5-HT1B receptor antagonistSB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. 了解更多 -
AR-M 1000390 hydrochloride
Catalog No. A21911 δ opioid receptor agonistAR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多 -
Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多 -
Olcegepant hydrochloride
Catalog No. A21900 CGRP1 receptor antagonistOlcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. 了解更多 -
Methoxy-PEPy
Catalog No. A21899 mGlu5 receptor antagonistMethoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM. 了解更多 -
SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
Catalog No. A21897 NMDA receptor antagonistSDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多 -
SB-269970 hydrochloride
Catalog No. A21889 5-HT7 receptor antagonistSB269970 hydrochloride (SB-269970A) is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with the pKi of 8.3, exhibits >50-fold selectivity against other receptors. 了解更多 -
Timapiprant sodium
Catalog No. A21883 D prostanoid receptor 2 antagonistTimapiprant sodium (OC000459 sodium) is a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist. 了解更多 -
LDN193189 Tetrahydrochloride
Catalog No. A21881 BMP type I receptor inhibitorLDN193189 Tetrahydrochloride is a selective BMP type I receptor inhibitor, which efficiently inhibits ALK2 and ALK3 (IC50=5 nM and 30 nM, respectively), with weaker effects on ALK4, ALK5 and ALK7 (IC50??500 nM). 了解更多 -
7-Chlorokynurenic acid sodium salt
Catalog No. A21879 NMDA receptor antagonist7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多 -
Vilazodone D8
Catalog No. A21876 SSR inhibitor / 5-HT1A receptor partial agonistVilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多 -
SKF 82958
Catalog No. A21866 -
Macitentan (n-butyl analogue)
Catalog No. A21845 endothelin ETA and ETB receptor antagonistMacitentan n-butyl analogue is a n-butyl analogue of Macitentan. Macitentan is an orally active, non-peptide dual endothelin ETA and ETB receptor antagonist for the potential treatment of idiopathic pulmonary fibrosis (IPF) and pulmonary arterial hypertension (PAH). 了解更多 -
Enclomiphene citrate
Catalog No. A21830 oestrogen receptor antagonistEnclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property. 了解更多 -
Nomegestrol acetate
Catalog No. A21829 progesterone receptor agonistNomegestrol acetate is a potent, highly selective progestogen, which is characterized as a full agonist at the progesterone receptor, with no or minimal binding to other steroid receptors, including the androgen and glucocorticoid receptors. 了解更多 -
DDR1-IN-1 dihydrochloride
Catalog No. A21813 DDR1 receptor tyrosine kinase inhibitorDDR1-IN-1 dihydrochloride is a potent and selective DDR1 receptor tyrosine kinase inhibitor with an IC50 of 105 nM; 4-fold less potent for DDR2 (IC50 = 413 nM). 了解更多 -
Mavoglurant racemate
Catalog No. A21799 mGlu5 receptor antagonistMavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. 了解更多 -
GSK1521498 free base (hydrochloride)
Catalog No. A21792 μ-opioid receptor (MOR) antagonistGSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多 -
PF-5190457
Catalog No. A21784 ghrelin receptor inverse agonistPF-5190457 is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36. 了解更多 -
SKF-82958 hydrobromide
Catalog No. A21763 D1/D5 receptor full agonistSKF-82958 hydrobromide is a D1/D5 receptor full agonist. 了解更多 -
Eprotirome
Catalog No. A21743 thyroid hormone receptor agonistEprotirome is a liver-selective thyroid hormone receptor agonist. 了解更多 -
LY 344864 S-enantiomer
Catalog No. A21742 5-HT1F receptor agonistLY 344864 S-enantiomer is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist. 了解更多 -
MCOPPB triHydrochloride
Catalog No. A21722 nociceptin receptor agonistMCOPPB 3Hcl is a nociceptin receptor agonist with pKi of 10.07; weaker activity at other opioid receptors. 了解更多 -
Pipequaline hydrochloride
Catalog No. A21712 partial benzodiazepine receptor agonistPipequaline hydrochloride (PK-8165 hydrochloride) is a partial benzodiazepine receptor agonist with anxiolytic activity. 了解更多 -
Taranabant ((1R,2R)stereoisomer)
Catalog No. A21705 CB1 receptor inverse agonistTaranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多 -
diABZI STING agonist-1 trihydrochloride
Catalog No. A21694 STING receptor agonistdiABZI STING agonist-1 (trihydrochloride) is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 for human PBMCs. 了解更多 -
diABZI STING agonist-1
Catalog No. A21688 STING receptor agonistdiABZI STING agonist-1 is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 nM for human PBMCs. 了解更多 -
SAG hydrochloride
Catalog No. A21678 Smo receptor agonistSAG (hydrochloride) is a potent Smo receptor agonist, and activates the Hedgehog signaling pathway, with a Kd of 59 nM. 了解更多
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