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Cell Cycle

产品 51 到 100 共 257个

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  1. PD 0332991 Isethionate
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    PD 0332991 Isethionate

    Catalog No. A13811
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    CDK4/6 抑制剂
    PD 0332991 Isethionate是CDK4/6的高选择性抑制剂，IC50分别为11 nM/16 nM。 了解更多
  2. P276-00
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    P276-00

    Catalog No. A13547
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    CDK 抑制剂
    P276-00是一种新型CDK1，CDK4和CDK9抑制剂，IC50分别为79 nM，63 nM和20 nM。在第2/3阶段。 了解更多
  3. LEE011 (Ribociclib)
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    LEE011 (Ribociclib)

    Catalog No. A13549
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    CDK4/6 抑制剂
    LEE011 (Ribociclib)是一种可口服的细胞周期蛋白依赖性激酶（CDK）抑制剂，靶向细胞周期蛋白D1/CDK4和细胞周期蛋白D3/CDK6细胞周期途径，具有潜在的抗肿瘤活性。 了解更多
  4. LDC000067
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    LDC000067

    Catalog No. A14273
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    CDK 抑制剂
    LDC000067是一种高选择性CDK9抑制剂。 了解更多
  5. AMG-925
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    AMG-925

    Catalog No. A14025
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    Dual FLT3/CDK4 抑制剂
    AMG-925是一种有效，选择性和生物利用性的FLT3/细胞周期蛋白依赖性激酶4（CDK4）双激酶抑制剂。 了解更多
  6. CVT-313
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    CVT-313

    Catalog No. A15054
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    CDK2 抑制剂
    CVT-313是一种有效，选择性，可逆且具有ATP竞争性的CDK2抑制剂（对于Cdk2/A和Cdk2/E，IC50 = 0.5 uM；对于Cdk1/B为4.2 uM；对于Cdk4/D1为215 uM）。 了解更多
  7. Purvalanol A
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    Purvalanol A

    Catalog No. A15517
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    CDK 抑制剂
    Purvalanol A是一种有效的细胞渗透性细胞周期蛋白依赖性蛋白激酶（cdk）抑制剂。对于cdc2/cyclin B，cdk2/cyclin A，cdk2/cyclin E，cdk4/cyclin D1和cdk5-p35，IC50值分别为4、70、35、850和75 nM。 了解更多
  8. NVP-LCQ195
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    NVP-LCQ195

    Catalog No. A15196
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    CDK 抑制剂
    NVP-LCQ195是CDK1，CDK2，CDK3和CDK5的小分子杂环抑制剂，IC50为1-42 nM。 了解更多
  9. AG-024322
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    AG-024322

    Catalog No. A15485
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    CDK 抑制剂
    AG-24322是第二代CDK抑制剂。AG-024322是有效的CDK1，CDK2和CDK4抑制剂，可在临床前模型中产生细胞周期停滞和抗肿瘤活性。 了解更多
  10. NU2058
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    NU2058

    Catalog No. A15767
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    CDK 抑制剂
    NU2058是基于鸟嘌呤的CDK抑制剂，对CDK2和CDK1的IC50为17 uM和26 uM。 了解更多
  11. CDK8-IN-1
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    CDK8-IN-1

    Catalog No. A12961
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    CDK8 inhibitor
    CDK8-IN-1 is a potent and selective CDK8 inhibitor with an IC50 of 3 nM. 了解更多
  12. CDK-IN-2
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    CDK-IN-2

    Catalog No. A11353
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    CDK9 inhibitor
    CDK-IN-2 is a potent and specific CDK9 inhibitor with IC50 of <8 nM, extracted from reference 1, example 4. 了解更多
  13. Senexin A
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    Senexin A

    Catalog No. A21166
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    CDK8 inhibitor
    Senexin A is a CDK8 inhibitor with an IC50 of 280 nM. 了解更多
  14. Voruciclib hydrochloride
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    Voruciclib hydrochloride

    Catalog No. A21385
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    CDK inhibitor
    Voruciclib hydrochloride is a clinical stage orally active and selective CDK inhibitor with Ki values of 0.626 nM-9.1 nM. 了解更多
  15. PHA-767491 hydrochloride
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    PHA-767491 hydrochloride

    Catalog No. A21395
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    dual Cdc7/Cdk9 inhibitor
    PHA-767491 hydrochloride is a dual Cdc7/Cdk9 inhibitor, with IC50s of 10 nM and 34 nM, respectively. 了解更多
  16. CDKI-73
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    CDKI-73

    Catalog No. A21467
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    CDK9 inhibitor
    CDKI-73 is a potent CDK9 inhibitor with Ki of 4 nM; shows selective toxicity to CLL cells(LD50=80 nM) versus normal B cell and normal CD34+ cell(LD50>20 uM). 了解更多
  17. CDK9-IN-1
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    CDK9-IN-1

    Catalog No. A21552
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    CDK9 inhibitor
    CDK9-IN-1 is a novel, selective CDK9 inhibitor for the treatment of HIV infection, with an IC50 of 39 nM for CDK9/CycT1, extracted from reference, compound 87. 了解更多
  18. (±)-BAY-1251152
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    (±)-BAY-1251152

    Catalog No. A21564
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    PTEF/CDK9 inhibitor
    (±)-BAY-1251152 is a racemic mixture of BAY-1251152. BAY-1251152 is a potent and highly selective PTEF/CDK9 inhibitor. 了解更多
  19. (-)-BAY-1251152
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    (-)-BAY-1251152

    Catalog No. A21570
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    PTEF/CDK9 inhibitor
    (-)-BAY-1251152 is an enanthiomer of BAY-1251152 with rotation (-). BAY-1251152 is a potent and highly selective PTEF/CDK9 inhibitor. 了解更多
  20. Lerociclib dihydrochloride
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    Lerociclib dihydrochloride

    Catalog No. A21577
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    CDK4/CDK6 inhibitor
    Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively. 了解更多
  21. LDC4297
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    LDC4297

    Catalog No. A21613
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    CDK7 inhibitor
    LDC4297 is a potent and selective CDK7 inhibitor with an IC50 of 0.13 nM. 了解更多
  22. BS-181 hydrochloride
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    BS-181 hydrochloride

    Catalog No. A21988
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    CDK7 inhibitor
    BS-181 hydrochloride is a highly selective CDK7 inhibitor with IC50 of 21 nM, and > 40-fold selective for CDK7 than CDK1, 2, 4, 5, 6, or 9. 了解更多
  23. SEL120-34A HCl
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    SEL120-34A HCl

    Catalog No. A21485
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    CDK8 inhibitor
    SEL120-34A HCl is a potent, selective, orally available, ATP-competitive CDK8 inhibitor, with IC50s of 4.4 nM and 10.4 nM for CDK8/CycC and CDK19/CycC, respectively, with antitumor activity. 了解更多
  24. NU6300
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    NU6300

    Catalog No. A21025
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    ATP-competitive CDK2 inhibitor
    NU6300 is the first covalent ATP-competitive CDK2 inhibitor. 了解更多
  25. Indirubin
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    Indirubin

    Catalog No. A10471
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    CDK & GSK-3β 抑制剂
    Indirubin是中国抗白血病药物的活性成分，是一种有效的细胞周期蛋白依赖性激酶和GSK-3β抑制剂，IC50约为5 μM和0.6 μM。 了解更多
  26. SNS-032 (BMS-387032)
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    SNS-032 (BMS-387032)

    Catalog No. A10850
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    CDK 抑制剂
    SNS-032（BMS-387032）是细胞周期蛋白依赖性激酶（Cdks）2、7和9的高度选择性和有效抑制剂，具有体外生长抑制作用，并具有诱导恶性B细胞凋亡的能力。 了解更多
  27. AT7519
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    AT7519

    Catalog No. A10093
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    CDK 抑制剂
    AT7519是多种细胞周期蛋白依赖性激酶（CDK）的抑制剂，可导致细胞周期停滞，诱导细胞凋亡和抑制肿瘤细胞增殖。作用于CDK1，2，4，6和9时，IC50为10-210 nM，对CDK3作用效果稍弱，对CDK7几乎没有抑制活性。 了解更多
  28. BS-181
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    BS-181

    Catalog No. A10163
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    CDK 抑制剂
    BS-181 是作为CDK7抑制剂的潜在抗肿瘤剂。 了解更多
  29. Flavopiridol HCl
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    Flavopiridol HCl

    Catalog No. A11045
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    CDK 抑制剂
    Flavopiridol HCl是细胞周期蛋白依赖性激酶的抑制剂。（-）-顺式形式诱导特定肿瘤细胞的凋亡。 了解更多
  30. JNJ-7706621
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    JNJ-7706621

    Catalog No. A10494
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    CDK/Aurora A/B 抑制剂
    JNJ-7706621是对CDK1/2具有最高效力的pan-CDK抑制剂，IC50为9 nM/4 nM，并且在无细胞分析中对CDK1/2的选择性是CDK3/4/6的6倍以上。它还能有效抑制极光A/B，对Plk1和Wee1没有活性。 了解更多
  31. PHA-848125 (Milciclib)
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    PHA-848125 (Milciclib)

    Catalog No. A11047
    CDK 抑制剂
    PHA-848125 (Milciclib)是一种有效的，ATP竞争性CDK抑制剂，作用于CDK2，IC50为45 nM，作用于CDK2比作用于CDK1，2，4，5和7选择性高3倍以上。 了解更多
  32. AZD5438
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    AZD5438

    Catalog No. A11105
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    CDK 抑制剂
    AZD5438是有效的细胞周期蛋白依赖性激酶（CDK）1、2和9抑制剂（IC50值分别为16、6和20 nM）。 了解更多
  33. BMS-265246
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    BMS-265246

    Catalog No. A11154
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    CDK 抑制剂
    BMS-265246是cdk2/cyclin E和cdk1/cyclin B以及cdk4/cyclin D的强新吡唑并吡啶抑制剂。 了解更多
  34. R547
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    R547

    Catalog No. A11190
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    CDK 抑制剂
    R547是一种新型的细胞周期和转录周期依赖性激酶（CDKs）选择性抑制剂（CDK1，CDK2和CDK4分别为Ki = 1、3和1 nM），具有出色的体外细胞效价，可抑制各种细胞的生长。人肿瘤细胞系。 了解更多
  35. AT7519 HCl
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    AT7519 HCl

    Catalog No. A11313
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    CDK 抑制剂
    AT7519是多种细胞周期蛋白依赖性激酶（CDK）的抑制剂，可导致细胞周期停滞，诱导细胞凋亡和抑制肿瘤细胞增殖。 了解更多
  36. CGP60474
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    CGP60474

    Catalog No. A11347
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    CDK 抑制剂
    CGP60474是细胞周期蛋白依赖性激酶(CDK)的有效抑制剂。 了解更多
  37. Purvalanol B
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    Purvalanol B

    Catalog No. A12352
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    CDK 抑制剂
    Purvalanol B是一种细胞周期蛋白依赖性激酶抑制剂。对于cdc2/cyclin B，cdk2/cyclin A，cdk2/cyclin E，cdk4/cyclin D1和cdk5-p35的ic50值分别为6、6、9、> 10，000和6 nm。对一系列其他蛋白激酶具有选择性(IC50 > 10，000 nM)。 了解更多
  38. NU 6102
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    NU 6102

    Catalog No. A12438
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    CDK 抑制剂
    NU 6102与CDK4/D1（IC50 = 1.6μM），DYRK1A（IC50 = 0.9μM），PDK1（IC50 = 0.8μM）和ROCKII（IC50 = 0.6μM）相比，NU6102对CDK1和CDK2具有选择性。 了解更多
  39. Wogonin
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    Wogonin

    Catalog No. A12216
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    CDK9 抑制剂
    Wogonin是抗炎剂和CDK9抑制剂，并且在抑制CDK9活性的剂量下不抑制CDK2, CDK4和CDK6也抑制N-乙酰转移酶。 了解更多
  40. TG003
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    TG003

    Catalog No. A13721
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    Clk 抑制剂
    TG003是Cdc2样激酶（Clk）的有效，特异性，可逆和ATP竞争性抑制剂。 了解更多
  41. THZ1
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    THZ1

    Catalog No. A14192
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    CDK7 抑制剂
    THZ1是一种新型的选择性强效共价CDK7抑制剂，IC50（结合亲和力）为3.2 nM。抑制Jurkat细胞的增殖，IC50为50 nM。 了解更多
  42. TG-02 (SB1317)
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    TG-02 (SB1317)

    Catalog No. A11962
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    FLT3 抑制剂
    TG-02 (SB1317)是一种新型的小分子有效CDK/JAK2/FLT3抑制剂。 了解更多
  43. NU6027
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    NU6027

    Catalog No. A14136
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    ATR/CDK 抑制剂
    NU6027是一种有效的细胞ATR活性抑制剂（IC（50）=6.7μM），并以ATR依赖的方式增强羟基脲和顺铂的细胞毒性。 了解更多
  44. ML167
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    ML167

    Catalog No. A14297
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    Clk4 抑制剂
    ML167是一种高度选择性的Cdc2样激酶4（Clk4）抑制剂。 了解更多
  45. SU9516
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    SU9516

    Catalog No. A14318
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    CDK2 抑制剂
    SU9516是一种有效的选择性cdk2抑制剂。它抑制pRb磷酸化，导致增强的pRB/E2F复合物形成，并诱导G1和G2-M细胞周期停滞。 了解更多
  46. Voruciclib
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    Voruciclib

    Catalog No. A14392
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    CDK 抑制剂
    Voruciclib是一种黄酮和细胞周期蛋白依赖性激酶（CDK）抑制剂，具有潜在的抗肿瘤活性。 了解更多
  47. CA-224
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    CA-224

    Catalog No. A14414
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    CDK4 抑制剂
    CA-224是有效的CDK4抑制剂，也是fascaplysin的非平面类似物，在体外特异性抑制Cdk4-cyclin D1。 了解更多
  48. Ro 3306
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    Ro 3306

    Catalog No. A14437
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    CDK1 抑制剂
    Ro 3306是一种具有ATP竞争能力的有效细胞周期蛋白依赖性激酶（cdk）1抑制剂（cdk1/cyclin B1和cdk1/cyclin A的Ki值分别为35和110 nM。 了解更多
  49. PHA690509
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    PHA690509

    Catalog No. A13550
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    CDK 抑制剂
    PHA690509是ATP竞争性CDK抑制剂。 了解更多
  50. AZD5597
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    AZD5597

    Catalog No. A13506
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    CDK 抑制剂
    AZD5597是有效的CDK抑制剂，对一系列癌细胞具有体外抗增殖作用。 了解更多

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分类
  1. Chk (38)
  2. CDK (97)
  3. Aurora Kinase (37)
  4. PLK (14)
  5. ROCK (33)
  6. c-Myc (5)
  7. Wee1 (2)
  8. Ras (38)
  9. DYRK (11)
  10. G-quadruplex (3)
  11. RAD51 (3)
作用机制
  1. Inhibitor (抑制剂) (250)
  2. Agonist (激动剂) (1)
  3. Antagonist (拮抗剂) (1)
  4. Activator (激活剂) (2)
  5. Degrader (降解剂) (1)
靶点
  1. A3 adenosine receptor (1)
  2. Abl (3)
  3. Aurora A (28)
  4. Aurora B (22)
  5. Aurora C (11)
  6. Bcr-Abl (1)
  7. CDK (3)
  8. CDK2 (1)
  9. CDK4 (2)
  10. Chk2 (1)
  11. CYP3A4 (1)
  12. FAK (1)
  13. FGFR1 (4)
  14. FGFR2 (1)
  15. FGFR3 (1)
  16. FLT3 (6)
  17. IGF1R (1)
  18. JAK2 (4)
  19. JAK3 (1)
  20. Lck (1)
  21. MEK1 (2)
  22. MEK2 (1)
  23. PDE3 (1)
  24. PDGFRβ (1)
  25. RET (1)
  26. Src (3)
  27. TrkA (2)
  28. VEGFR2 (FLK1) (2)
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