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产品 151 到 200 共 257个

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  1. TC-S 7010 (Aurora A Inhibitor I)
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    TC-S 7010 (Aurora A Inhibitor I)

    Catalog No. A10100
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    Aurora A 抑制剂
    TC-S 7010 (Aurora A Inhibitor I)是Aurora A激酶（AurA）的有效和选择性抑制剂，IC50值为3.4 nM（Aurora A），对Aurora B具有极高的选择性1000倍； 用于研究Aurora A激酶的细胞作用的有用工具化合物。 了解更多
  2. CCT129202
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    CCT129202

    Catalog No. A10184
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    Aurora 抑制剂
    CCT129202是一种ATP竞争性的pan-Aurora抑制剂，作用于Aurora A，Aurora B和Aurora C时，IC50分别为0.042 μM，0.198 μM和0.227 μM，对FGFR3， GSK3β， PDGFRβ等作用效果稍弱。 了解更多
  3. GSK1070916
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    GSK1070916

    Catalog No. A11168
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    Aurora Kinase B/C 抑制剂
    GSK1070916是一种有效的Aurora B/C激酶抑制剂（IC50为3.5 nM/6.5 nM），在组织培养细胞和人肿瘤异种移植模型中具有广泛的抗肿瘤活性。 了解更多
  4. PF-03814735
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    PF-03814735

    Catalog No. A11171
    Aurora A/B Kinase 抑制剂
    PF-03814735是一种新颖，有效且可逆的Aurora A/B抑制剂，IC50为0.8 nM/5 nM，对Flt3，FAK，TrkA的效力较低，对Met和FGFR1的活性最低。 了解更多
  5. PHA-680632
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    PHA-680632

    Catalog No. A10714
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    Aurora 抑制剂
    PHA-680632是Aurora A，Aurora B和Aurora C的有效抑制剂，IC50分别为27 nM，135 nM和120 nM。对于FGFR1，FLT3，LCK，PLK1，STLK2和VEGFR2/3，它的IC50高10到200倍。 了解更多
  6. SNS-314
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    SNS-314

    Catalog No. A10851
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    Aurora 抑制剂
    SNS-314 Mesylate是Aurora A，Aurora B和Aurora C的有效和选择性抑制剂，IC50分别为9 nM，31 nM和3 nM。 它对Trk A/B，Flt4，Fms，Axl，c-Raf和DDR2的效力较低。 阶段1。 了解更多
  7. ZM-447439
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    ZM-447439

    Catalog No. A11009
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    Aurora Kinase 抑制剂
    ZM 447439是Aurora A和Aurora B的选择性和ATP竞争性抑制剂，IC50分别为110 nM和130 nM。它对Aurora A/B的选择性是MEK1，Src，Lck的8倍以上，对CDK1/2/4，Plk1，Chk1等的影响很小。 了解更多
  8. CYC116 (CYC-116)
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    CYC116 (CYC-116)

    Catalog No. A10248
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    Aurora Kinase 抑制剂
    CYC116 (CYC-116)是一种有效的Aurora A/B抑制剂，Ki为8.0 nM/9.2 nM，对VEGFR2(Ki为44 nM)作用稍弱。 了解更多
  9. XL-228
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    XL-228

    Catalog No. A13069
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    IGF-1R, Aurora, FGFR, ABL, SRC 抑制剂
    XL228是靶向IGF1R，AURORA激酶，FGFR1-3，ABL和SRC家族激酶的蛋白激酶抑制剂。XL228是一种Aurora A抑制剂（IC50，f3 nmol/L），对ABL1（Ki，5 nmol/L）以及BCR-ABL1 T315I（Ki，1.4 nmol/L）激酶显示出有效的生化活性。 了解更多
  10. MK-8745
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    MK-8745

    Catalog No. A13396
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    Aurora Kinase A 抑制剂
    MK-8745是一种新的极光特异性抑制剂。当在多种谱系的细胞系中进行体外试验时，它以p53依赖的方式诱导凋亡细胞死亡。 了解更多
  11. TC-A-2317 HCl
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    TC-A-2317 HCl

    Catalog No. A13567
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    Aurora kinase A 抑制剂
    TC-A-2317 HCl是一种有效的Aurora激酶A抑制剂（Ki = 1.2 nM，而抑制Aurora激酶B则为101 nM）。选择性超过60种其他激酶（IC50值> 1000 nM）。表现出良好的细胞通透性和抗肿瘤活性。 了解更多
  12. AZD1152
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    AZD1152

    Catalog No. A15011
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    Aurora B 抑制剂
    AZD1152是一种前药，可在血清中迅速经历磷酸酶介导的裂解作用，释放出Barasertib-hQPA（一种选择性的Aurora B激酶抑制剂），在急性髓细胞性白血病（AML）患者的临床研究中显示出初步活性。 了解更多
  13. SCH-1473759
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    SCH-1473759

    Catalog No. A14059
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    Aurora A/B 抑制剂
    SCH-1473759是一种新型的亚纳摩尔Aurora A/B抑制剂，IC50分别为4 nM和13 nM。 了解更多
  14. HOI-07
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    HOI-07

    Catalog No. A15970
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    Aurora B 抑制剂
    HOI-07是有效的Aurora B激酶抑制剂。 了解更多
  15. LY3295668
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    LY3295668

    Catalog No. A16869
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    Aurora A 抑制剂
    LY3295668，也称为AK-01，是有效的Aurora-A激酶抑制剂。 了解更多
  16. CCT241736
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    CCT241736

    Catalog No. A21097
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    dual FLT3/Aurora kinase inhibitor
    CCT241736 is a potent and orally bioavailable dual FLT3 and Aurora kinase inhibitor. 了解更多
  17. SCH-1473759 hydrochloride
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    SCH-1473759 hydrochloride

    Catalog No. A21711
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    Aurora inhibitor
    SCH-1473759 hydrochloride is an aurora inhibitor with IC50s of 4 and 13 nM for aurora A and B, respectively. 了解更多
  18. Aurora Kinase Inhibitor 3
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    Aurora Kinase Inhibitor 3

    Catalog No. A19448
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    Aurora A kinase inhibitor
    Aurora Kinase Inhibitor 3 is a strong and selective Aurora A kinase inhibitor with an IC50 of 42 nM, and weakly inhibits EGFR with an IC50>10 μM. 了解更多
  19. Aurora inhibitor 1
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    Aurora inhibitor 1

    Catalog No. A19637
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    Aurora inhibitor
    Aurora inhibitor 1 is a potent Aurora inhibitor with an IC50 of ?? 4 nM and ??13 nM for Aurora A and Aurora B kinase, respectively. 了解更多
  20. LFM-A13
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    LFM-A13

    Catalog No. A16261
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    BTK 抑制剂
    LFM-A13是有效且选择性的Btk抑制剂，IC50为17.2 uM；也抑制PLK3，IC50为7.2 uM。 了解更多
  21. Y-27632 2HCl
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    Y-27632 2HCl

    Catalog No. A11001
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    ROCK 抑制剂
    Y-27632是一种Rho相关的线圈激酶（ROCK）抑制剂，可提高人类胚胎干细胞（hESCs）的克隆效率。比对其他激酶包括PKC，cAMP依赖性蛋白激酶，MLCK和PAK的作用强200多倍。 了解更多
  22. Fasudil HCl (HA-1077)
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    Fasudil HCl (HA-1077)

    Catalog No. A10381
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    ROCK 抑制剂
    Fasudil HCl (HA-1077)是一种环状核苷酸依赖性蛋白激酶抑制剂和Rho相关激酶抑制剂（IC50 = 10.7μM）。 了解更多
  23. GSK 269962
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    GSK 269962

    Catalog No. A12348
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    ROCK 抑制剂
    GSK 269962是一种强效Rho激酶(ROCK)抑制剂(重组人ROCK1和ROCK2的IC50值分别为1.6和4 nM)。 了解更多
  24. Thiazovivin
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    Thiazovivin

    Catalog No. A10928
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    ROCK 抑制剂
    Thiazovivin是一种Rho相关激酶（ROCK）的选择性抑制剂。 了解更多
  25. RKI-1313
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    RKI-1313

    Catalog No. A10899
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    ROCK 抑制剂
    RKI-1313是RKI-1447的阴性对照，RKI-1447是Rho相关的ROCK激酶的有效抑制剂，在乳腺癌中具有抗侵袭和抗肿瘤活性。 了解更多
  26. BMS-5
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    BMS-5

    Catalog No. A12839
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    LIMK 抑制剂
    BMS-5是一种有效的LIMK抑制剂，对LIMK1和LIMK2的IC50分别为7 nM和8 nM。 了解更多
  27. BDP5290
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    BDP5290

    Catalog No. A16966
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    ROCK and MRCK 抑制剂
    BDP5290是ROCK和MRCK的有效抑制剂，对ROCK1，ROCK2，MRCKα和MRCKβ的IC50分别为5 nM，50 nM，10 nM和100 nM。 了解更多
  28. R-10015
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    R-10015

    Catalog No. A18806
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    LIMK inhibitor
    R-10015, a broad-spectrum antiviral compound for HIV infection, acts as a potent and selective inhibitor of LIM domain kinase (LIMK) and binds to the ATP-binding pocket, with an IC50 of 38 nM for human LIMK1. 了解更多
  29. ROCK inhibitor-2
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    ROCK inhibitor-2

    Catalog No. A18912
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    ROCK1/ROCK2 inhibitor
    ROCK inhibitor-2 is a selective dual ROCK1 and ROCK2 inhibitor with IC50s of 17 nM and 2 nM, respectively. 了解更多
  30. T56-LIMKi
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    T56-LIMKi

    Catalog No. A12266
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    LIMK2 inhibitor
    T56-LIMKi is a selective inhibitor of LIMK2; inhibits the growth of Panc-1 cells with an IC50 of 35.2 μM. 了解更多
  31. Y-33075 dihydrochloride
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    Y-33075 dihydrochloride

    Catalog No. A11611
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    ROCK inhibitor
    Y-33075 dihydrochloride is a selective ROCK inhibitor with an IC50 of 3.6 nM. 了解更多
  32. Y-27632
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    Y-27632

    Catalog No. A21448
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    ROCK-I/ROCK-II inhibitor
    Y-27632 is an ATP-competitive inhibitor of ROCK-I and ROCK-II, with Ki of 220 nM and 300 nM for ROCK-I and ROCK-II, respectively. 了解更多
  33. Fasudil
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    Fasudil

    Catalog No. A21628
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    ROCK inhibitor
    Fasudil (HA-1077; AT877), is a nonspecific ROCK inhibitor and also has inhibitory effect on protein kinases. 了解更多
  34. BMS-3
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    BMS-3

    Catalog No. A20999
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    LIMK inhibitor
    BMS-3 is a potent LIMK inhibitor with IC50s of 5 nM and 6 nM for LIMK1 and LIMK2, respectively. 了解更多
  35. GSK429286A
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    GSK429286A

    Catalog No. A10441
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    ROCK 抑制剂
    GSK429286A是含有蛋白激酶(ROCK)的Rho相关卷曲螺旋的细胞渗透性选择性小分子抑制剂。 了解更多
  36. HA-1077 dihydrochloride
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    HA-1077 dihydrochloride

    Catalog No. A13785
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    ROCK 抑制剂
    HA-1077 dihydrochloride通过充当细胞内Ca2+拮抗剂来抑制血管平滑肌收缩。 了解更多
  37. RKI-1447
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    RKI-1447

    Catalog No. A13067
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    ROCK1/ROCK2 抑制剂
    RKI-1447是Rho相关ROCK激酶的有效抑制剂，在乳腺癌中具有抗侵袭和抗肿瘤活性。 了解更多
  38. Y-33075
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    Y-33075

    Catalog No. A11610
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    ROCK 抑制剂
    Y-33075是ROCK（Rho相关的卷曲螺旋形成蛋白激酶）抑制剂。 了解更多
  39. AT13148
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    AT13148

    Catalog No. A12464
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    multi-AGC kinase 抑制剂
    AT13148是一种新型多AGC激酶抑制剂，具有强大的药效和抗肿瘤活性，与其他AKT抑制剂相比，具有独特的作用机理。 了解更多
  40. chroman 1
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    chroman 1

    Catalog No. A15045
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    ROCK 抑制剂
    Chroman 1 是一种高效且选择性的ROCK II抑制剂。 了解更多
  41. H-1152
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    H-1152

    Catalog No. A15101
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    ROCK 抑制剂
    H-1152是一种异喹啉磺酰胺衍生物，是Rho激酶的一种更特异，更强且可透过膜的抑制剂，Ki值为1.6 nM，但对其他丝氨酸/苏氨酸激酶的抑制作用较差。 了解更多
  42. Glycyl-H 1152 2HCl
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    Glycyl-H 1152 2HCl

    Catalog No. A13659
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    ROCK 抑制剂
    Glycyl-H 1152 2HCl是一种选择性有效的ROCK抑制剂（ROCKII，Aurora A，CAMKII，PKG，PKA和PKC的IC50值分别为0.0118、2.35、2.57、3.26，> 10和> 10 uM。） 了解更多
  43. H-1152 dihydrochloride
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    H-1152 dihydrochloride

    Catalog No. A15102
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    ROCK 抑制剂
    H-1152 dihydrochloride是一种异喹啉磺酰胺衍生物，是Rho激酶的一种更特异，更强且可透过膜的抑制剂，Ki值为1.6 nM，但对其他丝氨酸/苏氨酸激酶的抑制作用较弱。 了解更多
  44. SLx-2119 (KD025)
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    SLx-2119 (KD025)

    Catalog No. A15239
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    ROCK2 抑制剂
    SLx-2119 (KD025)是ROCK2的小分子和选择性抑制剂，IC50为105 nM。在ROCK1上的选择性> 200倍（IC50 = 24 uM）。 了解更多
  45. SAR407899 HCl
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    SAR407899 HCl

    Catalog No. A15921
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    ROCK 抑制剂
    SAR407899是一种有效且选择性的Rho激酶抑制剂，具有良好的抗高血压活性。 了解更多
  46. Ripasudil
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    Ripasudil

    Catalog No. A15888
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    ROCK inhibitor
    Ripasudil (K-115) is potent ROCK inhibitor with IC50 of 51 nM and 19 nM for ROCK1 and ROCK2, respectively, used for the treatment of glaucoma and ocular hypertension. 了解更多
  47. LX7101
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    LX7101

    Catalog No. A16211
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    LIMK2 抑制剂
    LX7101是基于吡咯并嘧啶的局部递送的LIM域激酶2（LIMK2）抑制剂，LIM域激酶2是与眼内压调节相关的激酶。 了解更多
  48. ROCK inhibitor-1
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    ROCK inhibitor-1

    Catalog No. A15226
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    ROCK 抑制剂
    N/A 了解更多
  49. ROCK inhibitor
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    ROCK inhibitor

    Catalog No. A15225
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    ROCK 抑制剂
    ROCK inhibitor是人类ROCK-1和ROCK-2同工酶的高效抑制剂，IC50值分别为0.6和1.1 nM。 了解更多
  50. Narciclasine
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    Narciclasine

    Catalog No. A15178
    ROCK activator
    Narciclasine是Rho/Rho激酶/ LIM激酶/ cofilin信号通路激活剂。 了解更多

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  1. Chk (38)
  2. CDK (97)
  3. Aurora Kinase (37)
  4. PLK (14)
  5. ROCK (33)
  6. c-Myc (5)
  7. Wee1 (2)
  8. Ras (38)
  9. DYRK (11)
  10. G-quadruplex (3)
  11. RAD51 (3)
作用机制
  1. Inhibitor (抑制剂) (250)
  2. Agonist (激动剂) (1)
  3. Antagonist (拮抗剂) (1)
  4. Activator (激活剂) (2)
  5. Degrader (降解剂) (1)
靶点
  1. A3 adenosine receptor (1)
  2. Abl (3)
  3. Aurora A (28)
  4. Aurora B (22)
  5. Aurora C (11)
  6. Bcr-Abl (1)
  7. CDK (3)
  8. CDK2 (1)
  9. CDK4 (2)
  10. Chk2 (1)
  11. CYP3A4 (1)
  12. FAK (1)
  13. FGFR1 (4)
  14. FGFR2 (1)
  15. FGFR3 (1)
  16. FLT3 (6)
  17. IGF1R (1)
  18. JAK2 (4)
  19. JAK3 (1)
  20. Lck (1)
  21. MEK1 (2)
  22. MEK2 (1)
  23. PDE3 (1)
  24. PDGFRβ (1)
  25. RET (1)
  26. Src (3)
  27. TrkA (2)
  28. VEGFR2 (FLK1) (2)
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