Cell Metabolism
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Collagen proline hydroxylase inhibitor
Catalog No. A11371 -
LCI-699 (Osilodrostat)
Catalog No. A14013 11β-hydroxylase 抑制剂LCI-699 (Osilodrostat)是人11β-羟化酶和醛固酮合酶的有效抑制剂,IC50值分别为2.5和0.7 nM。 了解更多 -
4-Chloro-DL-phenylalanine
Catalog No. A16424 Tryptophan hydroxylase 抑制剂4-Chloro-DL-phenylalanine是色氨酸羟化酶的选择性和不可逆抑制剂,色氨酸羟化酶是5-羟色胺(5-羟色胺)生物合成中的限速酶。 了解更多 -
Fondaparinux Sodium
Catalog No. A17918 factor Xa inhibitorFondaparinux sodium is a factor Xa inhibitor to form the high affinity binding site for the anti-coagulant factor antithrombin III (ATIII). 了解更多 -
RWJ-445167
Catalog No. A12154 dual inhibitor of thrombin and factor XaRWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with Ki of 4.0 nM and 230 nM, respectively, exhibiting potent antithrombotic activity. 了解更多 -
BMS-654457
Catalog No. A21704 Factor XIa (FXIa) inhibitorBMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa), binding with human and rabbit FXIa with Kis of 0.2 and 0.42 nM, respectively. 了解更多 -
Apixaban (BMS-562247-01)
Catalog No. A10082 Factor Xa 抑制剂Apixaban (BMS-562247-01)是一种抗凝剂,用于预防静脉血栓栓塞和静脉血栓栓塞事件。 了解更多 -
BMS-740808
Catalog No. A10158 -
Rivaroxaban (Xarelto)
Catalog No. A10800 Factor Xa 抑制剂Rivaroxaban (Xarelto)是一种Factor Xa的直接抑制剂,无细胞试验中Ki和IC50分别为0.4 nM和0.7 nM。 了解更多 -
Otamixaban (FXV 673)
Catalog No. A11517 -
Letaxaban (TAK-442)
Catalog No. A12871 factor Xa 抑制剂Letaxaban (TAK-442)是一种有效的,选择性的,口服活性的Xa抑制剂,是一种四氢嘧啶-2(1H)-衍生物。TAK-442在贫血小板的人[半最大抑制浓度(IC(50)):53 nM,TAK-442]和大鼠(IC(50):32 nM,TAK-442)血浆中抑制内源性FXa活性。 了解更多 -
Betrixaban
Catalog No. A12518 FXa 抑制剂Betrixaban是一种抗凝血药,可作为直接Xa因子抑制剂。它具有强大的,口服活性和对因子Xa的高度选择性,由于其低hERG亲和力而从一组相似的化合物中选择。 了解更多 -
Edoxaban (tosylate Monohydrate)
Catalog No. A14317 Factor Xa 抑制剂Edoxaban (tosylate Monohydrate)是选择性Factor Xa抑制剂,Ki为0.561 nM。 了解更多 -
5-R-Rivaroxaban
Catalog No. A14979 Factor Xa 抑制剂5-R-Rivaroxaban是利伐沙班的(R)对映异构体。利伐沙班是一种新型的口服直接Xa因子抑制剂,在晚期开发中用于预防和治疗血栓栓塞性疾病。 了解更多 -
Edoxaban tosylate
Catalog No. A15076 -
Rasagiline
Catalog No. A11111 -
Hordenine
Catalog No. A10454 -
Quercetin (Sophoretin)
Catalog No. A10766 MAO-B 抑制剂Quercetin (Sophoretin)抑制许多酶系统,包括酪氨酸蛋白激酶,磷脂酶A2,磷酸二酯酶,线粒体ATPase,PI 3-激酶和蛋白激酶C。 了解更多 -
Quercetin dihydrate (Sophoretin)
Catalog No. A10765 MAO-B 抑制剂Quercetin dihydrate (Sophoretin)抑制许多酶系统,包括酪氨酸蛋白激酶,磷脂酶A2,磷酸二酯酶,线粒体ATPase,PI 3-激酶和蛋白激酶C。 了解更多 -
Olodaterol
Catalog No. A15761 MAO 抑制剂Olodaterol是一种长效的β肾上腺素受体激动剂,由Boehringer-Ingelheim生产,用于吸入治疗慢性阻塞性肺疾病(COPD)患者。 了解更多 -
Pargyline hydrochloride
Catalog No. A17288 MAO inhibitorPargyline hydrochloride is an irreversible inhibitor of monoamine oxidase (MAO) that is used clinically to treat moderate hypertension. 了解更多 -
Iproniazid
Catalog No. A17445 MAO inhibitorIproniazid is a non-selective, irreversible monoamine oxidase (MAO) inhibitor (MAOI) that is used as an antidepressive agent. 了解更多 -
Molindone hydrochloride
Catalog No. A17647 MAO inhibitorMolindone HCl is a D2 dopamine receptor antagonist. It also acts as a MAO inhibitor. 了解更多 -
Minaprine dihydrochloride
Catalog No. A17722 MAO-A inhibitorMinaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression. 了解更多 -
Toloxatone
Catalog No. A18043 MAO-A inhibitorToloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor. Antidepressant. 了解更多 -
Iproniazid phosphate
Catalog No. A18135 MAO inhibitorIproniazid phosphate is an irreversible inhibitor of monoamine oxidase types A and B that is used as an antidepressive agent. It has also been used as an antitubercular agent, but its use is limited by its toxicity. 了解更多 -
Salsolidine
Catalog No. A12969 MAO-A inhibitorSalsolidine is a tetrahydroisoquinoline alkaloid, acts as a stereoselective competitive MAO A inhibitor. 了解更多 -
Lazabemide
Catalog No. A21270 MAO-B inhibitorLazabemide(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). 了解更多 -
Ro 41-1049 hydrochloride
Catalog No. A21672 inhibitor of monoamine oxidase-A (MAO-A)Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (MAO-A). 了解更多 -
Brofaromine
Catalog No. A21777 MAO inhibitorBrofaromine (CGP 11305A) is a monoamine oxidase (MAO) inhibitor with IC50 of 0.2?μM for MAO-A. 了解更多 -
Safinamide Mesylate (FCE28073)
Catalog No. A10818 -
Rasagiline mesylate
Catalog No. A11722 Monoamine oxidase 抑制剂Rasagiline mesylate是一种不可逆的单胺氧化酶抑制剂,在早期帕金森氏病中用作单一疗法,在较晚期的病例中用作辅助疗法。对于B型MAO,它对A型的选择性是14倍。 了解更多 -
SL251188
Catalog No. A11777 -
Moclobemide
Catalog No. A11885 -
Bifemelane HCl
Catalog No. A13353 -
Tranylcypromine hydrochloride
Catalog No. A13358 LSD1/BHC110 & MAO 抑制剂Tranylcypromine hydrochloride是一种非选择性的MAO-A/B抑制剂。 了解更多 -
Safinamide
Catalog No. A13294 -
Clorgyline hydrochloride
Catalog No. A17357 monoamine oxidase A inhibitorClorgyline hydrochloride is an irreversible and selective inhibitor of monoamine oxidase A (MAO-A) that is used in scientific research; structurally related to Pargyline. 了解更多 -
Isocarboxazid
Catalog No. A17887 monoamine oxidase inhibitorIsocarboxazid is a non-selective and irreversible inhibitor of monoamine oxidase, with an IC50 of 4.8 μM for rat brain monoamine oxidase in vitro. 了解更多 -
Rasagiline 13C3 mesylate racemic
Catalog No. A21350 Monoamine oxidase inhibitorRasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible inhibitor of monoamine oxidase. 了解更多 -
PAT-1251 Hydrochloride
Catalog No. A21969 LOXL2 inhibitorPAT-1251 Hydrochloride is a potent, selective and oral lysyl oxidase-like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively). 了解更多