Cell Metabolism
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Methotrexate (Abitrexate)
Catalog No. A10021 -
Pemetrexed
Catalog No. A12668 -
NSC 131463 (DAMPA)
Catalog No. A10655 -
Pralatrexate
Catalog No. A11522 -
Diaveridine
Catalog No. A17000 DHFR 抑制剂Diaveridine(EGIS-5645)是一种二氢叶酸还原酶(DHFR)抑制剂,其野生型DHFR的Ki值为11.5 nM,同时也是一种抗菌剂。 了解更多 -
CAY10566
Catalog No. A16936 -
Ammonium Glycyrrhizinate (AMGZ)
Catalog No. A10070 -
Mycophenolate mofetil (CellCept)
Catalog No. A10613 IMPDH 抑制剂Mycophenolate mofetil (CellCept)是嘌呤生物合成(特别是鸟嘌呤合成)中肌苷单磷酸脱氢酶(IMPDH)的可逆抑制剂,对T细胞和B细胞的生长是必需的。 了解更多 -
Leflunomide
Catalog No. A10521 Dehydrogenase 抑制剂Leflunomide是一种嘧啶合成抑制剂,属于DMARD类药物。来氟米特用于缓解类风湿性关节炎引起的症状,如炎症、肿胀、僵硬和关节痛。 了解更多 -
CPI-613 (Devimistat)
Catalog No. A11786 Dehydrogenase 抑制剂CPI-613是合成的α-硫辛酸硫辛酸类似物的对映异构体的外消旋混合物,具有潜在的化学预防和抗肿瘤活性。 了解更多 -
CGP 3466B maleate
Catalog No. A12385 -
Vidofludimus (4SC-101)
Catalog No. A12997 -
AZD4017
Catalog No. A13542 -
MK-8245 Trifluoroacetate
Catalog No. A15170 Liver-targeting SCD 抑制剂?MK-8245 Trifluoroacetate是硬脂酰辅酶A去饱和酶(SCD)的肝靶向抑制剂,对人SCD1的IC50为1 nM,对大鼠SCD1和小鼠SCD1的IC50为3 nM,具有抗糖尿病和抗血脂异常的功效。 了解更多 -
NCT-501
Catalog No. A15892 -
AG-120
Catalog No. A15869 -
Fomepizole
Catalog No. A16164 -
CBR 5884
Catalog No. A16176 -
UK-383367
Catalog No. A10959 -
Ethoxzolamide
Catalog No. A17359 Carbonic anhydrase inhibitorEthoxzolamide is a carbonic anhydrase inhibitor with Ki of 1 nM. 了解更多 -
Dorzolamide HCL
Catalog No. A10333 carbonic anhydrase 抑制剂Dorzolamide HCl是一种碳酸酐酶抑制剂。它是一种抗青光眼剂,以滴眼剂的形式局部使用。盐酸度尔佐胺用于降低开角型青光眼和高眼压患者的眼内压升高。 了解更多 -
Tioxolone
Catalog No. A11673 -
Brinzolamide
Catalog No. A11765 -
Diclofenamide
Catalog No. A10303 -
Indisulam (E7070)
Catalog No. A12325 Carbonic anhydrase inhbitorIndisulam (E7070)是一种碳酸酐酶抑制剂,也是一种靶向细胞周期G1期的新型合成磺酰胺。 了解更多 -
Punicalagin
Catalog No. A12105 Carbonic anhydrase 抑制剂Punicalagin是一种鞣花单宁,一种酚类化合物。它是一种高活性碳酸酐酶抑制剂。 了解更多 -
U-104
Catalog No. A14959 -
Acetazolamide
Catalog No. A15859 Carbonic Anhydrase 抑制剂Acetazolamide是一种有效的碳酸酐酶(CA)抑制剂,在临床实践中通常用作迅速降低眼内压(IOP)的直接且容易获得的选择。 了解更多 -
Benzenesulfonamide
Catalog No. A13594 -
URB597
Catalog No. A11049 -
PF-04457845
Catalog No. A15209 -
FAAH inhibitor 1
Catalog No. A21841 FAAH inhibitorFAAH inhibitor 1 (Benzothiazole analog 3) is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18??8 nM. 了解更多 -
PF-3845
Catalog No. A11183 -
LY 2183240
Catalog No. A11960 FAAH 抑制剂LY 2183240既可作为内源性大麻素再摄取的有效抑制剂,IC50为270 pM,又可作为脂肪酸酰胺水解酶(FAAH)的抑制剂,IC50为12.4 nM,而脂肪酸酰胺水解酶是负责降解花生四烯酸的主要酶。 了解更多 -
JNJ 1661010
Catalog No. A12420 -
Glycyrrhetinic acid (Enoxolone)
Catalog No. A10353