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￥ 0.00 Cell Metabolism
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Quercetin (Sophoretin)
Catalog No. A10766 MAO-B 抑制剂Quercetin (Sophoretin)抑制许多酶系统，包括酪氨酸蛋白激酶，磷脂酶A2，磷酸二酯酶，线粒体ATPase，PI 3-激酶和蛋白激酶C。 了解更多 -
Quercetin dihydrate (Sophoretin)
Catalog No. A10765 MAO-B 抑制剂Quercetin dihydrate (Sophoretin)抑制许多酶系统，包括酪氨酸蛋白激酶，磷脂酶A2，磷酸二酯酶，线粒体ATPase，PI 3-激酶和蛋白激酶C。 了解更多 -
Olodaterol
Catalog No. A15761 MAO 抑制剂Olodaterol是一种长效的β肾上腺素受体激动剂，由Boehringer-Ingelheim生产，用于吸入治疗慢性阻塞性肺疾病（COPD）患者。 了解更多 -
Pargyline hydrochloride
Catalog No. A17288 MAO inhibitorPargyline hydrochloride is an irreversible inhibitor of monoamine oxidase (MAO) that is used clinically to treat moderate hypertension. 了解更多 -
Iproniazid
Catalog No. A17445 MAO inhibitorIproniazid is a non-selective, irreversible monoamine oxidase (MAO) inhibitor (MAOI) that is used as an antidepressive agent. 了解更多 -
Molindone hydrochloride
Catalog No. A17647 MAO inhibitorMolindone HCl is a D2 dopamine receptor antagonist. It also acts as a MAO inhibitor. 了解更多 -
Minaprine dihydrochloride
Catalog No. A17722 MAO-A inhibitorMinaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression. 了解更多 -
Toloxatone
Catalog No. A18043 MAO-A inhibitorToloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor. Antidepressant. 了解更多 -
Iproniazid phosphate
Catalog No. A18135 MAO inhibitorIproniazid phosphate is an irreversible inhibitor of monoamine oxidase types A and B that is used as an antidepressive agent. It has also been used as an antitubercular agent, but its use is limited by its toxicity. 了解更多 -
Salsolidine
Catalog No. A12969 MAO-A inhibitorSalsolidine is a tetrahydroisoquinoline alkaloid, acts as a stereoselective competitive MAO A inhibitor. 了解更多 -
Lazabemide
Catalog No. A21270 MAO-B inhibitorLazabemide(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). 了解更多 -
Ro 41-1049 hydrochloride
Catalog No. A21672 inhibitor of monoamine oxidase-A (MAO-A)Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (MAO-A). 了解更多 -
Brofaromine
Catalog No. A21777 MAO inhibitorBrofaromine (CGP 11305A) is a monoamine oxidase (MAO) inhibitor with IC50 of 0.2?μM for MAO-A. 了解更多 -
Apixaban (BMS-562247-01)
Catalog No. A10082 Factor Xa 抑制剂Apixaban (BMS-562247-01)是一种抗凝剂，用于预防静脉血栓栓塞和静脉血栓栓塞事件。 了解更多 -
BMS-740808
Catalog No. A10158 -
Rivaroxaban (Xarelto)
Catalog No. A10800 Factor Xa 抑制剂Rivaroxaban (Xarelto)是一种Factor Xa的直接抑制剂，无细胞试验中Ki和IC50分别为0.4 nM和0.7 nM。 了解更多 -
Otamixaban (FXV 673)
Catalog No. A11517 -
Letaxaban (TAK-442)
Catalog No. A12871 factor Xa 抑制剂Letaxaban (TAK-442)是一种有效的，选择性的，口服活性的Xa抑制剂，是一种四氢嘧啶-2（1H）-衍生物。TAK-442在贫血小板的人[半最大抑制浓度（IC（50））：53 nM，TAK-442]和大鼠（IC（50）：32 nM，TAK-442）血浆中抑制内源性FXa活性。 了解更多 -
Betrixaban
Catalog No. A12518 FXa 抑制剂Betrixaban是一种抗凝血药，可作为直接Xa因子抑制剂。它具有强大的，口服活性和对因子Xa的高度选择性，由于其低hERG亲和力而从一组相似的化合物中选择。 了解更多 -
Edoxaban (tosylate Monohydrate)
Catalog No. A14317 Factor Xa 抑制剂Edoxaban (tosylate Monohydrate)是选择性Factor Xa抑制剂，Ki为0.561 nM。 了解更多 -
5-R-Rivaroxaban
Catalog No. A14979 Factor Xa 抑制剂5-R-Rivaroxaban是利伐沙班的（R）对映异构体。利伐沙班是一种新型的口服直接Xa因子抑制剂，在晚期开发中用于预防和治疗血栓栓塞性疾病。 了解更多 -
Edoxaban tosylate
Catalog No. A15076 -
Fondaparinux Sodium
Catalog No. A17918 factor Xa inhibitorFondaparinux sodium is a factor Xa inhibitor to form the high affinity binding site for the anti-coagulant factor antithrombin III (ATIII). 了解更多 -
RWJ-445167
Catalog No. A12154 dual inhibitor of thrombin and factor XaRWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with Ki of 4.0 nM and 230 nM, respectively, exhibiting potent antithrombotic activity. 了解更多 -
BMS-654457
Catalog No. A21704 Factor XIa (FXIa) inhibitorBMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa), binding with human and rabbit FXIa with Kis of 0.2 and 0.42 nM, respectively. 了解更多 -
Nepicastat HCl
Catalog No. A11172 -
Tetrahydropapaverine HCl
Catalog No. A10920 Hydroxylase 抑制剂Tetrahydropapaverine HCl是TIQs的一种，是Salsolinol和Tetrahydropapaveroline的类似物，对多巴胺神经元具有神经毒性作用。 了解更多 -
LX 1606 Hippurate
Catalog No. A10542 Hydroxylase 抑制剂LX 1606 hippurate是一种口服生物可利用的小分子色氨酸羟化酶(TPH)抑制剂，具有潜在的抗旋转能活性。 了解更多 -
Nepicastat (free base) (SYN-117)
Catalog No. A10637 dopamine beta-hydroxylase 抑制剂Nepicastat (free base) (SYN-117)是多巴胺β-羟化酶的抑制剂，该酶催化多巴胺向去甲肾上腺素的转化。 了解更多 -
LX 1606 (Telotristat)
Catalog No. A11785 Serotonin synthesis 抑制剂LX 1606 (Telotristat)是一种口服生物可利用的小分子色氨酸羟化酶（TPH）抑制剂，具有潜在的抗血清素活性。 了解更多 -
Ro 61-8048
Catalog No. A12833 Hydroxylase 抑制剂Ro 61-8048是有效的竞争性犬尿氨酸3-羟化酶抑制剂（Ki = 4.8 nM，IC50 = 37 nM）。 了解更多 -
Collagen proline hydroxylase inhibitor
Catalog No. A11371 -
LCI-699 (Osilodrostat)
Catalog No. A14013 11β-hydroxylase 抑制剂LCI-699 (Osilodrostat)是人11β-羟化酶和醛固酮合酶的有效抑制剂，IC50值分别为2.5和0.7 nM。 了解更多 -
4-Chloro-DL-phenylalanine
Catalog No. A16424 Tryptophan hydroxylase 抑制剂4-Chloro-DL-phenylalanine是色氨酸羟化酶的选择性和不可逆抑制剂，色氨酸羟化酶是5-羟色胺（5-羟色胺）生物合成中的限速酶。 了解更多 -
17-AAG (KOS953)
Catalog No. A10010 HSP90 抑制剂17-AAG (KOS953)是一种有效的HSP90抑制剂，无细胞试验中IC50为5 nM，作用于来自肿瘤细胞的HSP90比作用于来自正常细胞HSP90结合亲和力高100倍。 了解更多 -
AUY922 (Luminespib, NVP-AUY922)
Catalog No. A10659 HSP90 抑制剂AUY922 (Luminespib,NVP-AUY922)是一种高效的HSP90抑制剂，在Hsp90 FP结合测定中的IC50 = 21 nM，并在体外抑制多种人类癌细胞系的增殖，GI50平均为9 nM。Luminespib (AUY-922, NVP-AUY922)是一种高效的HSP90抑制剂，无细胞试验中作用于HSP90α/β的IC50为13 nM /21 nM，对HSP90家族成员GRP94和TRAP-1具有稍弱的作用，与任何小分子HSP90配体均可紧密结合。 了解更多 -
NVP-BEP800
Catalog No. A10660 HSP90 抑制剂NVP-BEP800是一种新型的，完全合成的，口服可生物利用的抑制剂，可与Hsp90的NH2末端ATP结合袋结合。 了解更多
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