微信关注
China
Total item
Cart Subtotal
￥ 0.00 Cell Metabolism
-
Clarithromycin
Catalog No. A10225 cytochrome P4503A4 抑制剂Clarithromycin是一种大环内酯类抗生素。它通过干扰细菌的蛋白质合成来防止细菌生长。 了解更多 -
Haloperidol (Haldol)
Catalog No. A10446 -
Talarozole R enantiomer
Catalog No. A13113 Cytochrome P450 抑制剂Talarozole R enantiomer 通过阻断细胞色素P450酶同工酶CYP26（一种视黄酸羟化酶）来抑制视黄酸的代谢。 了解更多 -
Efavirenz
Catalog No. A15826 -
Sulfaphenazole
Catalog No. A17283 CYP2C9 inhibitorSulfaphenazole is a specific inhibitor of CYP2C9 which blocks atherogenic and pro-inflammatory effects of linoleic acid (increase in oxidative stress and activation of AP-1) mediated by CYP2C9. 了解更多 -
CYP17-IN-1
Catalog No. A12622 CYP17 inhibitorCYP17-IN-1 (compound 9c) is a potent and orally active CYP17 inhibitor against rat and human CYP17 with IC50s of 15.8 and 20.1 nM. 了解更多 -
Liarozole dihydrochloride
Catalog No. A21853 CYP450 dependent inhibitorLiarozole dihydrochloride (R75251; R85246) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase). 了解更多 -
Seviteronel
Catalog No. A20996 CYP17 lyase inhibitorSeviteronel (VT-464) is a potent CYP17 lyase inhibitor(h-Lyase IC50=69 nM) that demonstrated both exceptional in vitro lyase/hydroxylase selectivity (~10-fold) and oral activity in a hamster model of androgen biosynthesis inhibition. 了解更多 -
TAK-700 (Orteronel)
Catalog No. A11044 -
Voriconazole (Vfend)
Catalog No. A10978 -
Abiraterone (CB-7598)
Catalog No. A10020 -
Abiraterone Acetate (CB7630)
Catalog No. A11058 -
Avasimibe (CI-1011)
Catalog No. A10102 CYP17 抑制剂Avasimibe (CI-1011)是口服可生物利用的酰基辅酶A：胆固醇O-酰基转移酶（ACAT）抑制剂，IC50分别为2.9 μM， 13.9 μM和26.5 μM。 了解更多 -
TOK-001 (Galeterone)
Catalog No. A11138 -
Posaconazole
Catalog No. A10744 CYP3A4 抑制剂Posaconazole主要是CYP3A4的抑制剂，但不抑制其他CYP酶的活性。也是甾醇C14+脱甲基酶抑制剂的抑制剂，IC50为0.25μM。泊沙康唑的终末消除半衰期中位数为15-35小时。 了解更多 -
Ketoconazole
Catalog No. A10498 -
Cobicistat (GS-9350)
Catalog No. A11277 CYP3A 抑制剂Cobicistat (GS-9350)是有效，选择性的细胞色素酶P450 3A (CYP3A)抑制剂，包括重要的cyp3a4亚型。它还抑制肠道转运蛋白，增加几种hiv药物的整体吸收，包括atazanavir、darunavir和tenofovir alafenamide延胡索酸盐。 了解更多 -
PF 4981517
Catalog No. A12544 CYP3A4 抑制剂PF 4981517是一种有效且选择性的CYP3A4抑制剂（CYP3A4，CYP3A5和CYP3A7的IC50值分别为0.03、17和70 μM）。 了解更多 -
Ozagrel(OKY-046)
Catalog No. A10688 -
TAK-700 Salt (Orteronel Salt)
Catalog No. A13515 CYP17A1/androgen synthesis 抑制剂TAK-700 Salt (Orteronel Salt)是一种雄激素合成抑制剂。它选择性地抑制在睾丸，肾上腺和前列腺肿瘤组织中表达的酶CYP17A。 了解更多 -
Choline Fenofibrate
Catalog No. A15044 -
Azathramycin
Catalog No. A15010 -
Benzbromarone
Catalog No. A16201 -
Cilostamide
Catalog No. A13596 -
GSK256066 2,2,2-trifluoroacetic acid
Catalog No. A15097 PDE 抑制剂GSK256066是一种选择性PDE4B（与A-D型同等亲和力）抑制剂，IC50为3.2 pM，对PDE1/2/3/5/6的选择性> 380,000倍，对PDE4B与PDE7的选择性> 2500倍。 了解更多 -
Nortadalafil
Catalog No. A15191 PDE5 抑制剂Nortadalafil是去甲基他达拉非，它是一种PDE5抑制剂，目前以药丸形式销售，用于治疗勃起功能障碍（ED），名称为Cialis。并以Adcirca为名，用于治疗肺动脉高压。 了解更多 -
Olprinone Hydrochloride
Catalog No. A15198 -
TAK-063
Catalog No. A15799 -
Sildenafil
Catalog No. A12631 PDE5 抑制剂Sildenafil是选择性磷酸二酯酶5（PDE5）抑制剂之一（IC50 = 5.22 nM），被认为是治疗勃起功能障碍的最佳方法。 了解更多 -
PDE-9 inhibitor
Catalog No. A11532 -
AN3199
Catalog No. A12228 -
PF-05180999
Catalog No. A13006 PDE2A inhibitorPF-05180999 is a phosphodiesterase 2A (PDE2A) inhibitor, with an IC50 of 1.6 nM. 了解更多 -
Sildenafil citrate
Catalog No. A10841 PDE5 inhibitorSildenafil citrate is a potent phosphodiesterase type 5 (PDE5) inhibitor with IC50 of 5.22 nM. 了解更多 -
Mirodenafil dihydrochloride
Catalog No. A18047 PDE-5 inhibitorMirodenafil dihydrochloride (SK3530 dihydrochloride) is a phosphodiesterase type 5 (PDE-5) inhibitor developed for the treatment of erectile dysfunction. 了解更多 -
D159687
Catalog No. A21228 -
PF-04957325
Catalog No. A21246 PDE8 inhibitorPF-04957325 is a highly potent and selective PDE8 inhibitor, with IC50s of 0.7 nM and 0.3 nM for PDE8A and PDE8B, respectively. 了解更多 -
Mirodenafil
Catalog No. A21260 PDE-5 inhibitorMirodenafil(SK3530) is a phosphodiesterase type 5 (PDE-5) inhibitor developed for the treatment of erectile dysfunction. 了解更多 -
Saterinone hydrochloride
Catalog No. A21402 PDE3 inhibitorSaterinone hydrochloride is a phosphodiesterase III (PDE III) inhibitor. 了解更多
FILTER BY:
Filtering:
- 作用机制: Inhibitor (抑制剂) 删除该内容
购物选项
- 分类
-
- Cytochrome P450 (29)
- PPAR (1)
- PDE (71)
- HSP (42)
- Hydroxylases (12)
- Factor Xa (16)
- MAO (30)
- DHFR (6)
- Dehydrogenases (19)
- Procollagen C-proteinase (1)
- Carbonic Anhydrase (12)
- FAAH (11)
- 15-PGDH (2)
- CETP (6)
- Ferroptosis (5)
- HMG-CoA Reductase (15)
- Isocitrate Dehydrogenase (IDH) (14)
- IDO (13)
- Lipase (9)
- Phospholipases (10)
- Lipoxygenase (11)
- NAMPT (5)
- GLUT (3)
- Antimetabolite (3)
- Lipid Metabolism (1)
- SREBP (2)
- LDL (1)
- Foxo1 (1)
- DGAT (6)
- Farnesyl Transferase (6)
- CRM1 (6)
- Thioredoxin (2)
- Decarboxylase (1)
- ACLY (2)
- Fatty acid synthase (FASN) (6)
- Lactate dehydrogenase A (LDHA) (1)
- PFKFB3 (3)
- Ribonucleotide Reductase (2)
- Acetyl-CoA Carboxylase (6)
- Glucosidase (3)
- Phosphatase (4)
- 靶点
-
- 5-lipoxygenase (1)
- Carbonic Anhydrase (6)
- Carbonic Anhydrase I (3)
- Carbonic Anhydrase II (3)
- Carbonic Anhydrase IV (2)
- Carbonic Anhydrase IX (2)
- CETP (4)
- COX (1)
- COX-1 (1)
- COX-2 (2)
- DNMT (1)
- FTase (4)
- HDAC1 (1)
- HMG-CoA Reductase (9)
- HSP90 (1)
- KDM1A (LSD1) (1)
- MAO-A (1)
- MAO-B (1)
- PDE4 (1)
- PDE5 (1)
- Src (1)
- TNF-α (1)
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
最近查看过的产品
ADOOQ 产品质量保证
We promise all products to perform as described.