CGRP Receptor
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CGRP 8-37 (human)
Catalog No. A16949 CGRP receptor 拮抗剂CGRP 8-37 (human)是人降钙素基因相关肽(hCGRP)片段,也是CGRP受体的拮抗剂。序列:Val-Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-Ser-Gly-Gly-Val-Val-Lys-Asn-Asn-Phe-Val-Pro-Thr-Asn- Val-Gly-Ser-Lys-Ala-Phe;VTHRLAGLLSRSGGVVKNNFVPTNVGSKAF。 了解更多 -
Olcegepant
Catalog No. A11512 CGRP1 receptorOlcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. 了解更多 -
Ubrogepant
Catalog No. A21670 CGRP antagonistUbrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine. 了解更多 -
Olcegepant hydrochloride
Catalog No. A21900 CGRP1 receptor antagonistOlcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. 了解更多 -
MK 3207 HCl
Catalog No. A10598 CGRP Receptor 拮抗剂MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂,IC50为0.12 nM。 了解更多 -
MK-0974 (Telcagepant)
Catalog No. A11255 -
BMS-927711
Catalog No. A13102 CGRP receptor 拮抗剂BMS-927711是一种有效的,选择性的,竞争性的人降钙素基因相关肽(CGRP)受体拮抗剂,已显示出体内功效,而没有血管收缩作用。 了解更多