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Cytoskeleton

产品 51 到 100 共 109个

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  1. GNE 2861
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    GNE 2861

    Catalog No. A21697
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    PAK inhibitor
    GNE 2861 is a PAK inhibitor that displays group II selectivity. GNE 2861 inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively. 了解更多
  2. PF-3758309
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    PF-3758309

    Catalog No. A11930
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    PAK4 抑制剂
    PF-3758309是抑制致癌信号和肿瘤生长的小分子p21活化激酶抑制剂。 了解更多
  3. LOR-253
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    LOR-253

    Catalog No. A13838
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    MTF-1 抑制剂
    LOR-253是人类金属调节转录因子1（MTF-1）的小分子抑制剂。 了解更多
  4. FRAX486
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    FRAX486

    Catalog No. A13691
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    PAK 抑制剂
    FRAX486是一种小分子PAK抑制剂。 了解更多
  5. KPT-9274
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    KPT-9274

    Catalog No. A15506
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    PAK4 抑制剂
    KPT-9274是有口服活性的PAK4/烟酰胺磷酸核糖基转移酶 (Nampt) 抑制剂，IC50值分别为小于 100 和 125 nM。 了解更多
  6. FRAX597
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    FRAX597

    Catalog No. A12553
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    PAK 抑制剂
    FRAX597是一种小分子吡啶并嘧啶酮，是I类PAK（PAK1 IC50 = 8 nM，PAK2 IC50 = 13 nM，PAK3 IC50 = 19 nM）的有效和ATP竞争性抑制剂。 了解更多
  7. FRAX1036
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    FRAX1036

    Catalog No. A16557
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    PAK inhibitor
    FRAX1036 is a PAK inhibitor with Kis of 23.3 nM, 72.4 nM, and 2.4 μM for PAK1, PAK2 and PAK4, respectively. 了解更多
  8. NVS-PAK1-1
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    NVS-PAK1-1

    Catalog No. A12708
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    allosteric PAK1 inhibitor
    NVS-PAK1-1 is a potent and selective allosteric PAK1 inhibitor with an IC50 of 5 nM. 了解更多
  9. Dynasore
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    Dynasore

    Catalog No. A12726
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    Dynamin 抑制剂
    dynasore是一种非竞争性的dynamin 1，dynamin 2和线粒体dynamin（Drp1）GTPase活性抑制剂。 了解更多
  10. Mdivi-1
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    Mdivi-1

    Catalog No. A14316
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    DRP1 抑制剂
    Mdivi-1是线粒体分裂DRP1（与动力蛋白相关的GTPase）和线粒体分裂动力蛋白I（Dnm1）的选择性细胞渗透性抑制剂，IC50为1-10 uM。 了解更多
  11. Dynamin inhibitory peptide
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    Dynamin inhibitory peptide

    Catalog No. A14867
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    Dynamin 抑制剂
    Dynamin inhibitory peptide是GTPase动力蛋白的肽抑制剂。 了解更多
  12. Dyngo-4a
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    Dyngo-4a

    Catalog No. A15915
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    Dynamin inhibitor
    Dyngo-4a is a potent dynamin inhibitor with IC50 of 0.38 uM, 1.1uM, and 2.3 uM for DynI (brain), DynI (rec), and DynII (rec), respectively. 了解更多
  13. GLPG0187
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    GLPG0187

    Catalog No. A13423
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    Integrin receptor antagonist
    GLPG0187 is a broad spectrum integrin receptor antagonist with antitumor activity; inhibits αvβ1-integrin with an IC50 of 1.3 nM. 了解更多
  14. Integrin Antagonists 27
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    Integrin Antagonists 27

    Catalog No. A20895
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    integrin αvβ3 antagonist
    Integrin Antagonists 27 is a small molecule integrin αvβ3 antagonist with binding affinity of 18 nM, as s novel anticancer agent. 了解更多
  15. MK-0429
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    MK-0429

    Catalog No. A21173
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    αvβ3 integrin antagonist
    MK-0429 (L-000845704) is an orally active, potent, selective and nonpeptide αvβ3 integrin antagonist with an IC50 of 80 nM. 了解更多
  16. ATN-161
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    ATN-161

    Catalog No. A21307
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    integrin α5β1 antagonist
    ATN-161 is a novel integrin α5β1 antagonist, which inhibits angiogenesis and growth of liver metastases in a murine model. 了解更多
  17. ATN-161 trifluoroacetate salt
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    ATN-161 trifluoroacetate salt

    Catalog No. A21412
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    integrin α5β1 antagonist
    ATN-161 trifluoroacetate salt is a novel integrin α5β1 antagonist, which inhibits angiogenesis and growth of liver metastases in a murine model. 了解更多
  18. Carotegrast
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    Carotegrast

    Catalog No. A21997
    α4 integrin receptor inhibitor
    Carotegrast is an orally available α4 integrin receptor inhibitor with anti-inflammatories activities. 了解更多
  19. Cyclo(RGDyK)
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    Cyclo(RGDyK)

    Catalog No. A21819
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    αVβ3 integrin inhibitor
    Cyclo(RGDyK) is a potent and selective αVβ3 integrin inhibitor with an IC50 of 20 nM. 了解更多
  20. Zaurategrast (CDP323)
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    Zaurategrast (CDP323)

    Catalog No. A11614
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    VCAM-1 拮抗剂
    Zaurategrast (CDP323)是与α4-整合素结合的血管细胞粘附分子1的小分子前药拮抗剂。 了解更多
  21. Cilengitide
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    Cilengitide

    Catalog No. A12372
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    Integrin 抑制剂
    Cilengitide是一种具有潜在抗肿瘤活性的环状精氨酸-甘氨酸-天冬氨酸肽。西仑吉肽结合并抑制α(v)β(3)和α(v)β(5)整联蛋白的活性，从而抑制内皮细胞-细胞相互作用、内皮细胞-基质相互作用和血管生成。 了解更多
  22. Cilengitide trifluoroacetate
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    Cilengitide trifluoroacetate

    Catalog No. A12371
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    Integrin 抑制剂
    Cilengitide trifluoroacetate是一种具有潜在抗肿瘤活性的环状精氨酸-甘氨酸-天冬氨酸肽。西仑吉肽结合并抑制α(v)β(3)和α(v)β(5)整联蛋白的活性，从而抑制内皮细胞-细胞相互作用、内皮细胞-基质相互作用和血管生成。 了解更多
  23. Firategrast (SB 683699)
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    Firategrast (SB 683699)

    Catalog No. A12787
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    α4β1/α4β7 integrin 拮抗剂
    Firategrast (SB 683699)是一种口服可生物利用的alpha4 beta1/alpha4 beta7整联蛋白拮抗剂，旨在减少淋巴细胞向中枢神经系统（CNS）的运输。 了解更多
  24. Pyrintegrin
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    Pyrintegrin

    Catalog No. A12876
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    pyintegrin是一种细胞可渗透的小分子，可将人类胚胎干细胞（hESC）的存活率提高30倍以上。 了解更多
  25. Leukadherin 1
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    Leukadherin 1

    Catalog No. A13968
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    Integrin 激动剂
    Leukadherin 1是CD11b/CD18的变构激活剂。增加CD11b/CD18依赖性细胞对血纤蛋白原的粘附（EC50 = 4μM）。 了解更多
  26. Cyclo (-RGDfK)
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    Cyclo (-RGDfK)

    Catalog No. A14923
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    αvβ3 integrin 抑制剂
    Cyclo (-RGDfK)是一种有效的、选择性的整合素抑制剂。 了解更多
  27. RGD (Arg-Gly-Asp) Peptides
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    RGD (Arg-Gly-Asp) Peptides

    Catalog No. A15538
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    Inhibits integrin binding to RGD motifs
    RGD (Arg-Gly-Asp) Peptides是一种细胞粘附基序，可以模拟细胞粘附蛋白并与整联蛋白结合。 了解更多
  28. E7820
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    E7820

    Catalog No. A15456
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    lpha-2-integrin 抑制剂
    E7820是一种小分子芳香族磺酰胺衍生物，具有潜在的抗血管生成和抗肿瘤活性。E7820通过抑制整合素α2（一种在内皮细胞上表达的细胞粘附分子）来抑制血管生成。 了解更多
  29. Cyclo (RGDyK) trifluoroacetate
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    Cyclo (RGDyK) trifluoroacetate

    Catalog No. A15918
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    Integrin 抑制剂
    Cyclo (RGDyK) trifluoroacetate是一种有效的选择性αVbeta3整联蛋白抑制剂，IC50为20 nM。 了解更多
  30. CWHM12
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    CWHM12

    Catalog No. A15967
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    αV integrins 抑制剂
    CWHM 12可以抑制所有5个alpha V整联蛋白。CWHM12不仅以与遗传删除方法相同的方式预防纤维化，还可以防止肝和肺中现有纤维化的进展，并逆转了由纤维化对这些器官造成的某些损害。 了解更多
  31. A-205804
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    A-205804

    Catalog No. A13047
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    Integrin 抑制剂
    A-205804是E-选择素和ICAM-1的有效和选择性抑制剂，IC50值分别为20 nM和25 nM。 了解更多
  32. BIO-1211
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    BIO-1211

    Catalog No. A17210
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    Integrin alpha4beta1 抑制剂
    BIO-1211是整联蛋白alpha4beta1抑制剂。 了解更多
  33. BOP sodium salt
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    BOP sodium salt

    Catalog No. A17201
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    α9β1/α4β1 integrin 抑制剂
    BOP sodium salt是新型的双重alpha9beta1/alpha4beta1整联蛋白抑制剂。 了解更多
  34. BTT-3033
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    BTT-3033

    Catalog No. A17200
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    α2β1 integrin 抑制剂
    BTT-3033是α2β1整联蛋白抑制剂。 了解更多
  35. TCS2314
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    TCS2314

    Catalog No. A17193
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    Integrin 抑制剂
    TCS2314是整联蛋白极晚期抗原4（VLA-4，α4β1）拮抗剂，IC50值为4.4 nM。 了解更多
  36. Obtustatin
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    Obtustatin

    Catalog No. A17185
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    α1β1 抑制剂
    Obtustatin是高度有效的整联蛋白α1β1抑制剂（α1β1与IV型胶原的结合的IC 50 = 0.8 nM）。与α2β1，βIIbβ3，αvβ3，α4β1，β5β6，α9β1和α4β7相比，α1β1具有选择性。在鸡绒膜尿囊炎模型中抑制FGF2刺激的血管生成。在Lewis肺癌的协同小鼠模型中显示抗肿瘤功效；阻止人黑素瘤在裸鼠中的生长。 了解更多
  37. R-BC154
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    R-BC154

    Catalog No. A17184
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    α4β1/α9β1 抑制剂
    R-BC154是高亲和力的荧光α4β1/α9 9β1抑制剂。 了解更多
  38. Litronesib Racemate
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    Litronesib Racemate

    Catalog No. A21498
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    kinesin Eg5 inhibitor
    Litronesib (Racemate) is the racemate of litronesib. Litronesib is a selective, allosteric inhibitor of kinesin Eg5. 了解更多
  39. Arry-520 (Filanesib)
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    Arry-520 (Filanesib)

    Catalog No. A11050
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    KSP 抑制剂
    Arry-520 (Filanesib)是一种特异性KSP抑制剂,具有潜在抗肿瘤活性的KSP（驱动蛋白5或Eg5）。 了解更多
  40. Ispinesib (SB-715992)
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    Ispinesib (SB-715992)

    Catalog No. A10486
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    KSP 抑制剂
    Ispinesib (SB-715992)是驱动蛋白纺锤体蛋白的有效抑制剂，驱动蛋白纺锤体蛋白是双极有丝分裂纺锤体形成和有丝分裂细胞周期进程所必需的驱动蛋白。 了解更多
  41. AZ 3146
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    AZ 3146

    Catalog No. A11170
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    Mps1 抑制剂
    AZ 3146是一种有效的选择性单极纺锤体1 (Mps1) 激酶抑制剂 (IC50 = 35 nM) 。它会干扰染色体对齐并覆盖纺锤体装配检查点，还抑制将Mad1，Mad2和着丝粒蛋白E（CENP-E）募集到动植物。 了解更多
  42. SB 743921
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    SB 743921

    Catalog No. A10828
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    KSP 抑制剂
    SB 743921是第二代KSP抑制剂，在癌症的临床前模型中是一种高效有效的治疗剂。 了解更多
  43. Monastrol
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    Monastrol

    Catalog No. A11976
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    Kinesin-5(KIF11) 抑制剂
    Monastrol是一种有效的，细胞可渗透的非微管蛋白相互作用的有丝分裂抑制剂。Monastrol通过与有丝分裂驱动蛋白Eg5结合来阻断有丝分裂（IC50 = 14μM），Eg5是纺锤体双极性所必需的运动蛋白。 了解更多
  44. GSK-923295
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    GSK-923295

    Catalog No. A11435
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    CENP-E 抑制剂
    GSK-923295是有丝分裂驱动蛋白着丝粒相关蛋白E（CENP-E）的小分子抑制剂。 了解更多
  45. ARQ 621
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    ARQ 621

    Catalog No. A14234
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    Eg5 mitotic motor protein 抑制剂
    ARQ 621是一种变构选择性Eg5有丝分裂运动蛋白抑制剂。 了解更多
  46. MPI-0479605
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    MPI-0479605

    Catalog No. A14290
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    Mps1 抑制剂
    MPI-0479605是有丝分裂激酶Mps1的ATP竞争性和选择性抑制剂。 了解更多
  47. ARRY-520 R enantiomer
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    ARRY-520 R enantiomer

    Catalog No. A15001
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    KSP 抑制剂
    ARRY-520 R enantiomer是ARRY-520的R形式，它是一种合成的小分子驱动蛋白纺锤体蛋白（KSP）抑制剂，IC50为6 nM。 了解更多
  48. Dimethylenastron
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    Dimethylenastron

    Catalog No. A15841
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    Kinesin Eg5 抑制剂
    Dimethylenastron是有丝分裂运动驱动蛋白Eg5的抑制剂，IC50值为200 nM。 了解更多
  49. K 858
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    K 858

    Catalog No. A15844
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    Kinesin Eg5 抑制剂
    K 858是一种选择性ATP不竞争的有丝分裂驱动蛋白Eg5抑制剂，IC50值为1.3 uM。 了解更多
  50. EMD534085
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    EMD534085

    Catalog No. A15956
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    Kinesin 抑制剂
    EMD534085是有效选择性的有丝分裂驱动蛋白-5 (kinesin-5)的抑制剂，IC50值为8 nM。 了解更多

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  1. Microtubules (48)
  2. PAK (9)
  3. Dynamin (4)
  4. Integrin (26)
  5. Kinesin (14)
  6. Mps1 (3)
  7. Gap Junction Protein (8)
作用机制
  1. Inhibitor (抑制剂) (73)
  2. Agonist (激动剂) (1)
  3. Antagonist (拮抗剂) (8)
  4. Modulator (调节剂) (1)
  5. Blocker (阻断剂) (2)
  6. Stabilizer (稳定剂) (1)
  7. Stimulator (刺激物) (1)
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