产品详情
DDR1-IN-1是一种有效的选择性DDR1受体酪氨酸激酶抑制剂,IC50/EC50为105 nM/87 nM,对DDR2的效力低4倍(IC50 = 413 nM)。
靶点信息
DDR1 | DDR2 | |||
105 nM | 413 nM |
In vitro | DMSO | Warmed: 87 mg/mL (157.44 mM) | |
Water | Insoluble | ||
Ethanol | Warmed: 3 mg/mL (5.42 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 18.1 mL | 90.48 mL | 180.97 mL |
0.5 mM | 3.62 mL | 18.1 mL | 36.19 mL |
1 mM | 1.81 mL | 9.05 mL | 18.1 mL |
5 mM | 0.36 mL | 1.81 mL | 3.62 mL |
*The above data is based on the productmolecular weight 552.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
目录号 | A13985 |
---|---|
作用机制 | Inhibitor (抑制剂) |
M. Wt | 552.59 |
Formula | C30H31F3N4O3 |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. |
CAS No. | 1449685-96-4 |
SMILES | CCN1CCN(CC1)CC2=C(C=C(C=C2)C(=O)NC3=CC(=C(C=C3)C)OC4=CC5=C(C=C4)NC(=O)C5)C(F)(F)F |
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