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Edoxaban (tosylate Monohydrate)

Edoxaban (tosylate Monohydrate)

Name: Edoxaban (tosylate Monohydrate)
SKU: A14317

目录号: A14317

Factor Xa 抑制剂

Product Citations (1)

Edoxaban (tosylate Monohydrate) Chemical Structure

CAS NO. 1229194-11-9

Edoxaban (tosylate Monohydrate)是选择性Factor Xa抑制剂，Ki为0.561 nM。

库存：现货

规格	价格	数量
10 mg	￥ 560.00
25 mg	￥ 1,050.00
50 mg	￥ 1,400.00
10mM * 1mL in DMSO	￥ 630.00

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生物活性

Edoxaban (tosylate Monohydrate)是选择性Factor Xa抑制剂，Ki为0.561 nM。

靶点信息

Factor Xa	Thrombin	FIXa
0.561 nM(Ki)	6 μM(Ki)	41.7 μM(Ki)

溶解度 *

In vitro	DMSO	89 mg/mL (120.55 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	13.55 mL	67.73 mL	135.45 mL
0.5 mM	2.71 mL	13.55 mL	27.09 mL
1 mM	1.35 mL	6.77 mL	13.55 mL
5 mM	0.27 mL	1.35 mL	2.71 mL

*The above data is based on the productmolecular weight 738.27. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A14317
作用机制	Inhibitor (抑制剂)
M. Wt	738.27
Formula	C24H30ClN7O4S.C7H8O3S.H2O
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1229194-11-9
Synonyms	DU-176b
SMILES	CC1=CC=C(C=C1)S(=O)(=O)O.CN1CCC2=C(C1)SC(=N2)C(=O)N[C@@H]3C[C@H](CC[C@@H]3NC(=O)C(=O)NC4=NC=C(C=C4)Cl)C(=O)N(C)C.O