微信关注
Total item
Cart Subtotal
￥ 0.00 Endocrinology / Hormones
42 个项目
每页
-
AGN-242428
Catalog No. A16935 RORγt 抑制剂AGN-242428，也称为VTP-43742，是一种有效的，选择性的和口服活性的RORγ抑制剂，Ki值为<100 nM。用于治疗自身免疫性疾病，包括多发性硬化症和牛皮癣。 了解更多 -
S18-000003
Catalog No. A19105 RORγt 抑制剂S18-000003 is a potent orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t (RORγt) inhibitor with an IC50 of 29 nM. S18-000003 inhibits IL-17 production. 了解更多 -
Anastrozole
Catalog No. A10075 Aromatase 抑制剂Anastrozole是第三代非甾体选择性芳香化酶抑制剂。与其他芳香酶抑制剂相比，它可能具有更高的选择性，没有任何内在的内分泌作用，并且对肾上腺类固醇的合成也没有明显的作用。 了解更多 -
Exemestane
Catalog No. A10378 -
Alpha-Naphthoflavone
Catalog No. A18474 aromatase inhibitorAlpha-Naphthoflavone is a synthetic flavonoid, acts as a potent and competitive aromatase inhibitor with an IC50 and a Ki of 0.5 and 0.2 μM, respectively. 了解更多 -
Fadrozole hydrochloride
Catalog No. A21258 Aromatase inhibitorFadrozole hydrochloride is a potent, selective and nonsteroidal inhibitor of aromatase with an IC50 of 6.4 nM. 了解更多 -
Aliskiren hemifumarate
Catalog No. A11123 -
Benazepril HCl
Catalog No. A10123 -
Clinofibrate
Catalog No. A11184 HMG-CoA Reductase 抑制剂Clinofibrate是一种脂质清除剂，似乎可以改变脂质代谢，减少类固醇诱导的骨细胞内脂质堆积。它还可以有效降低血浆纤维蛋白原水平。抑制hydroxymethylglutaryl coenzyme A reductase (HMGCR)（羟甲基戊二酰辅酶A还原酶），IC50为0.47 mM。 了解更多 -
Rosuvastatin
Catalog No. A11122 -
Aliskiren (CGP 60536)
Catalog No. A11616 -
Cilazapril monohydrate
Catalog No. A11747 -
Enalapril maleate
Catalog No. A10350 -
Enalaprilat dihydrate
Catalog No. A10351 -
LCZ696 (Valsartan)
Catalog No. A14206 angiotensin receptor-neprilysin 抑制剂LCZ696 (Valsartan)是一种生物利用型双效血管紧张素受体-中性溶血素抑制剂（ARNi），用于治疗高血压和心力衰竭。 了解更多 -
Captopril disulfide
Catalog No. A13521 LTA4 hydrolase 抑制剂Captopril disulfide是LTA4水解酶的可逆竞争性抑制剂（IC50 = 11 M）。Captopril已被证明是血管紧张素转化酶-1（ACE1）的一种，而不是ACE2（IC50 = 22 nM）。 了解更多 -
VTP-27999 2,2,2-trifluoroacetate
Catalog No. A15281 -
Spinorphin
Catalog No. A15314 -
MLN-4760
Catalog No. A16884 -
Fosinopril sodium
Catalog No. A11748 -
Zofenopril calcium
Catalog No. A12769 -
H-Val-Pro-Pro-OH
Catalog No. A18868 ACE inhibitorH-Val-Pro-Pro-OH, a milk-derived proline peptides derivative, is an inhibitor of Angiotensin I converting enzyme (ACE), with an IC50 of 9 μM. 了解更多 -
Zofenopril
Catalog No. A13615 ACE inhibitorZofenopril is an angiotensin-converting enzyme (ACE) inhibitor with an IC50 of 81 μM. 了解更多 -
Imidaprilate
Catalog No. A20003 ACE inhibitorImidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM, and is used in the research of hypertensive disease. 了解更多 -
Lisinopril
Catalog No. A21064 angiotensin-converting enzyme inhibitorLisinopril (MK-521) is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks. 了解更多 -
β-Sitosterol
Catalog No. A11015 -
Dutasteride (Avodart)
Catalog No. A10338 dual 5alpha-reductase 抑制剂Dutasteride (Avodart)是双重的5-a还原酶抑制剂，可抑制睾丸激素转化为二氢睾丸激素（DHT）。 了解更多 -
Epristeride
Catalog No. A18231 5 alpha-reductase inhibitorEpristeride is a selective and specific uncompetitive inhibitor of human steroid 5 alpha-reductase isoform 2. 了解更多 -
Diphenyleneiodonium chloride
Catalog No. A13359 GPR3 激动剂/NOS/ NADPH oxidases 抑制剂Diphenyleneiodonium是一种有效的不可逆的巨噬细胞抑制剂NOS2（iNOS）和内皮细胞NOS3（eNOS）抑制剂。 了解更多 -
TOK-001 (Galeterone)
Catalog No. A11138 -
AZD3514
Catalog No. A12396 -
Fulvestrant (Faslodex)
Catalog No. A10410 Aromatase 抑制剂Fulvestrant是一种雌激素受体拮抗剂，没有激动剂作用，它通过下调和降解雌激素受体发挥作用。 了解更多 -
Kaempferol
Catalog No. A10495 ERRα and ERRγ inverse 激动剂Kaempferol被发现抑制Ki为0.3-0.5 μM的牛主动脉肌球蛋白轻链激酶，并且还被发现通过新的ERK-NFκB-cMyc-p21途径抑制VEGF表达和体外血管生成。 了解更多
42 个项目
每页
FILTER BY:
Filtering:
- 作用机制: Inhibitor (抑制剂) 删除该内容
购物选项
- 分类
-
- Estrogen Receptors (3)
- Androgen Receptors (2)
- GPR (1)
- 5-alpha-reductase (3)
- Pregnane X Receptors (1)
- renin-angiotensin-aldosterone system (RAAS) (21)
- Aromatase (8)
- Vitamin D Receptors (1)
- GnRH receptor (1)
- ROR (2)
- 靶点
-
- Aromatase (4)
ADOOQ 产品质量保证
We promise all products to perform as described.