Endocrinology / Hormones

产品 201 到 236 共 236个

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  1. Beclometasone

    Catalog No. A18177
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    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. 了解更多
  2. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  3. OP-3633

    Catalog No. A18468
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    Glucocorticoid Receptor Antagonist
    OP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). 了解更多
  4. Ercalcidiol

    Catalog No. A11413
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    VD/VDR 抑制剂
    Ercalcidiol是D2的代谢物。 了解更多
  5. (R)-Elagolix

    Catalog No. A21184
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    GnRHR antagonist
    Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多
  6. Alarelin Acetate

    Catalog No. A20968
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    synthetic GnRH agonist
    Alarelin acetate is a synthetic GnRH agonist. 了解更多
  7. Ozarelix

    Catalog No. A12350
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    GnRH 拮抗剂
    Ozarelix是第四代GnRH拮抗剂,诱导激素难治性雄激素受体阴性前列腺癌细胞凋亡,调节死亡受体的表达和活性。 了解更多
  8. Abarelix Acetate

    Catalog No. A12613
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    GnRH 拮抗剂
    Abarelix acetate是一种合成的肽促性腺激素释放激素受体(GnRH)拮抗剂。 了解更多
  9. NBI-42902

    Catalog No. A12375
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    GnRH receptor 抑制剂
    NBI-42902是人促性腺激素释放激素受体的新型非肽拮抗剂。 了解更多
  10. SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂,对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM,对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  11. Ganirelix

    Catalog No. A12862
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    Ganirelix是一种可注射的竞争性促性腺激素释放激素拮抗剂(GnRH拮抗剂)。 了解更多
  12. Degarelix acetate

    Catalog No. A12840
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    GnRH 拮抗剂
    Degarelix acetate是促性腺激素释放激素(GnRH)受体拮抗剂。 了解更多
  13. GHRP-6 Acetate

    Catalog No. A13464
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    GHRP-6 Acetate是一种生长激素释放肽。 了解更多
  14. Elagolix sodium

    Catalog No. A13893
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    GnRH 拮抗剂
    Elagolix sodium是促性腺激素释放激素(GnRH)拮抗剂。Elagolix sodium抑制垂体腺中的促性腺激素释放激素(GnRH)受体,并最终降低循环性激素水平。 了解更多
  15. AEZS-108

    Catalog No. A13536
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    GnRH-1 激动剂
    AEZS-108是促性腺激素释放激素1受体(GnRH-1R)的肽激动剂,其与蒽环类抗生素阿霉素结合,具有潜在的抗肿瘤活性。 了解更多
  16. Leuprolide Acetate

    Catalog No. A15143
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    GnRH 激动剂
    Leuprolide Acetate是GnRH类似物;醋酸亮丙瑞林在垂体GnRH受体上起激动剂的作用。 了解更多
  17. Triptorelin Acetate

    Catalog No. A15997
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    GnRH 激动剂
    Triptorelin Acetate是一种促性腺激素释放激素激动剂(GnRH激动剂),用作乙酸盐或pamoate盐。 了解更多
  18. Goserelin Acetate

    Catalog No. A15959
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    GnRH 激动剂
    Goserelin Acetate是具有抗肿瘤活性的促黄体激素释放激素(LHRH)的合成十肽类似物。 了解更多
  19. Relugolix

    Catalog No. A17783
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    GnRH antagonist
    Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. 了解更多
  20. Leuprorelin Acetate

    Catalog No. A17986
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    GnRH/LHRH receptor agonist
    Leuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. 了解更多
  21. Nafarelin Acetate

    Catalog No. A17992
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    GnRH agonist
    Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. 了解更多
  22. Cetrorelix Acetate

    Catalog No. A18282
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    GnRH antagonist
    Cetrorelix acetate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity used in infertility treatment. The IC50 of 1.21 nM. 了解更多
  23. Goserelin

    Catalog No. A21197
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    GnRH agonist
    Goserelin(ICI 118630) is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). 了解更多
  24. SR1078

    Catalog No. A15245
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    ROR 激动剂
    SR1078是视黄酸受体相关的孤儿受体(ROR)RORα/γ的激动剂;增加RORα靶基因的转录;认为可以增加p53的稳定性。 了解更多
  25. SR3335

    Catalog No. A15246
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    RORα 激动剂
    SR3335是一种选择性RORα合成配体,直接与RORα结合,但不与其他ROR结合,并且在基于细胞的测定中用作RORα的选择性部分反向激动剂。 了解更多
  26. SR1001

    Catalog No. A13193
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    ROR 激动剂
    SR1001是选择性的ROR-α和ROR-γ反向激动剂;抑制TH17细胞分化并抑制自身免疫。 了解更多
  27. ROR gamma modulator 1

    Catalog No. A16291
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    RORγ modulator
    ROR gamma modulator 1 是类维生素A相关的孤儿受体γ(RORy)调节剂 了解更多
  28. SR-2211

    Catalog No. A13568
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    RORr 激动剂
    SR-2211选择性结合RORr(Ki = 105 nM),充当体外本构RORr活性的反向激动剂(IC50 = 320 nM)。 了解更多
  29. AGN-242428

    Catalog No. A16935
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    RORγt 抑制剂
    AGN-242428,也称为VTP-43742,是一种有效的,选择性的和口服活性的RORγ抑制剂,Ki值为<100 nM。用于治疗自身免疫性疾病,包括多发性硬化症和牛皮癣。 了解更多
  30. Cintirorgon (LYC-55716)

    Catalog No. A16863
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    RORγ 激动剂
    Cintirorgon (LYC-55716)是新型口服RAR相关孤儿受体γ(RORγ)激动剂。 了解更多
  31. AZD-0284

    Catalog No. A18766
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    RORγ 激动剂
    AZD-0284 is a potent, selective, inverse agonist of the nuclear receptor RORγ for the potential treatment of Plaque psoriasis. 了解更多
  32. XY101

    Catalog No. A18437
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    RORγ inverse 激动剂
    XY101 is a potent, selective, metabolically stable and orally available RORγ inverse agonist with an IC50 of 30 nM and a Kd of 380 nM. 了解更多
  33. S18-000003

    Catalog No. A19105
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    RORγt 抑制剂
    S18-000003 is a potent orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t (RORγt) inhibitor with an IC50 of 29 nM. S18-000003 inhibits IL-17 production. 了解更多
  34. A-9758

    Catalog No. A19078
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    RORγt inverse 激动剂
    A-9758 is a RORγ ligand and a potent, selective RORγt inverse agonist (IC50=5 nM), and exhibits robust potency against IL-17A release. 了解更多
  35. ROR agonist-1

    Catalog No. A18569
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    ROR 激动剂
    ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多
  36. (Glp1)-Apelin-13

    Catalog No. A13215
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    Apelin Receptor activator
    (Glp1)-Apelin-13是Apelin受体的激活剂。 了解更多

产品 201 到 236 共 236个

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