Endocrinology / Hormones
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Beclometasone
Catalog No. A18177 glucocorticoid receptor agonistBeclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. 了解更多 -
(R)-Elagolix
Catalog No. A21184 GnRHR antagonistElagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多 -
Alarelin Acetate
Catalog No. A20968 -
Ozarelix
Catalog No. A12350 -
Abarelix Acetate
Catalog No. A12613 -
Degarelix acetate
Catalog No. A12840 -
Elagolix sodium
Catalog No. A13893 GnRH 拮抗剂Elagolix sodium是促性腺激素释放激素(GnRH)拮抗剂。Elagolix sodium抑制垂体腺中的促性腺激素释放激素(GnRH)受体,并最终降低循环性激素水平。 了解更多 -
AEZS-108
Catalog No. A13536 -
Leuprolide Acetate
Catalog No. A15143 -
Triptorelin Acetate
Catalog No. A15997 -
Goserelin Acetate
Catalog No. A15959 -
Relugolix
Catalog No. A17783 GnRH antagonistRelugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. 了解更多 -
Leuprorelin Acetate
Catalog No. A17986 GnRH/LHRH receptor agonistLeuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. 了解更多 -
Nafarelin Acetate
Catalog No. A17992 GnRH agonistNafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. 了解更多 -
Cetrorelix Acetate
Catalog No. A18282 GnRH antagonistCetrorelix acetate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity used in infertility treatment. The IC50 of 1.21 nM. 了解更多 -
SR1078
Catalog No. A15245 -
SR3335
Catalog No. A15246 -
ROR gamma modulator 1
Catalog No. A16291 -
SR-2211
Catalog No. A13568 -
AGN-242428
Catalog No. A16935 RORγt 抑制剂AGN-242428,也称为VTP-43742,是一种有效的,选择性的和口服活性的RORγ抑制剂,Ki值为<100 nM。用于治疗自身免疫性疾病,包括多发性硬化症和牛皮癣。 了解更多 -
Cintirorgon (LYC-55716)
Catalog No. A16863 -
S18-000003
Catalog No. A19105 RORγt 抑制剂S18-000003 is a potent orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t (RORγt) inhibitor with an IC50 of 29 nM. S18-000003 inhibits IL-17 production. 了解更多 -
ROR agonist-1
Catalog No. A18569 ROR 激动剂ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多 -
(Glp1)-Apelin-13
Catalog No. A13215