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￥ 0.00 Endocrinology / Hormones
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Ozarelix
Catalog No. A12350 -
Abarelix Acetate
Catalog No. A12613 -
Degarelix acetate
Catalog No. A12840 -
Elagolix sodium
Catalog No. A13893 GnRH 拮抗剂Elagolix sodium是促性腺激素释放激素（GnRH）拮抗剂。Elagolix sodium抑制垂体腺中的促性腺激素释放激素（GnRH）受体，并最终降低循环性激素水平。 了解更多 -
Relugolix
Catalog No. A17783 GnRH antagonistRelugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. 了解更多 -
Cetrorelix Acetate
Catalog No. A18282 GnRH antagonistCetrorelix acetate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity used in infertility treatment. The IC50 of 1.21 nM. 了解更多 -
(R)-Elagolix
Catalog No. A21184 GnRHR antagonistElagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多 -
RU43044
Catalog No. A14340 -
Candesartan (Atacand)
Catalog No. A10175 RAAS 拮抗剂Candesartan (Atacand)是一种血管紧张素受体阻滞剂（也称为血管紧张素II受体拮抗剂或AIIRA）。 了解更多 -
Irbesartan (Avapro)
Catalog No. A10477 -
PD 123319 ditrifluoroacetate
Catalog No. A13201 angiotensin AT2 receptor 拮抗剂PD 123319 ditrifluoroacetate是一种有效的，选择性的非肽血管紧张素AT2受体拮抗剂。大鼠肾上腺组织和大脑的IC50值分别为34和210 nM。 了解更多 -
EXP-3174
Catalog No. A15451 -
Eprosartan
Catalog No. A11121 -
Telmisartan
Catalog No. A10905 -
Tasosartan
Catalog No. A10891 -
Azilsartan Medoxomil
Catalog No. A16420 angiotensin II receptor type 1 拮抗剂Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂，IC50为0.62 nM。 了解更多 -
Fimasartan
Catalog No. A17477 non-peptide angiotensin II receptor antagonistFimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多 -
Azilsartan medoxomil monopotassium
Catalog No. A20860 angiotensin II receptor type 1 antagonistAzilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多 -
Sparsentan
Catalog No. A20879 angiotensin II and endothelin A receptor antagonistSparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多 -
Losartan (D4 Carboxylic Acid)
Catalog No. A21578 angiotensin II receptor antagonistLosartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. 了解更多 -
Azilsartan D5
Catalog No. A21600 angiotensin II type 1 receptor antagonistAzilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多 -
NCRW0005-F05
Catalog No. A16184 GPR139 拮抗剂NCRW0005-F05是第一个对GPR139有选择性的拮抗剂（IC50值为0.21 uM）；是研究GPR139药理学的有用工具，尤其是与GPR139激动剂JNJ 63533054结合使用时。 了解更多 -
(R)-Bicalutamide
Catalog No. A10008 Androgen Receptor 拮抗剂(R)-Bicalutamide是一种活性的竞争性非甾体雄激素受体拮抗剂，对MDA 453细胞的IC50为0.17μM。 了解更多 -
Bicalutamide (Casodex)
Catalog No. A10142 Androgen Receptor 拮抗剂Bicalutamide (Casodex)是一种口服非甾体抗雄激素，用于治疗前列腺癌和多毛症。 了解更多 -
Cyproterone acetate
Catalog No. A11409 Androgen Receptor 拮抗剂Cyproterone acetate是17-羟孕酮的合成衍生物，可作为雄激素受体拮抗剂以及具有弱孕激素和糖皮质激素活性的弱孕激素受体激动剂。 了解更多 -
17 alpha-propionate
Catalog No. A10009 -
N-desMethyl EnzalutaMide
Catalog No. A13964 -
ODM-201
Catalog No. A15797 -
Lonaprisan
Catalog No. A14130 progesterone receptor 拮抗剂Lonaprisan是米非司酮相关类固醇的口服生物可利用的五氟乙基衍生物，具有抗孕激素活性。 了解更多 -
ACT-129968 (Setipiprant)
Catalog No. A15780 -
AZD9496
Catalog No. A15822 -
(E/Z)-4-hydroxy Tamoxifen
Catalog No. A12532 Estrogen receptor 拮抗剂(E/Z)-4-hydroxy Tamoxifen是他莫昔芬的活性代谢产物，是一种选择性雌激素受体（ER）调节剂，广泛用于乳腺癌的治疗和化学预防治疗。 了解更多 -
Tamoxifen Citrate
Catalog No. A10885 Estrogen receptor 拮抗剂Tamoxifen Citrate是哺乳动物甾醇异构酶的选择性和有效抑制剂。 了解更多 -
Fulvestrant R enantiomer
Catalog No. A21545 estrogen receptor antagonistFulvestrant R enantiomer (ICI 182780 R enantiomer; ZD 9238 R enantiomer; ZM 182780 R enantiomer) is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. 了解更多
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- Estrogen Receptors (11)
- Progesterone Receptors (3)
- Androgen Receptors (10)
- GPR (4)
- renin-angiotensin-aldosterone system (RAAS) (17)
- Glucocorticoid receptors (2)
- GnRH receptor (7)
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