EPI-001

Name: EPI-001
SKU: A15814

目录号: A15814

Androgen Receptor 拮抗剂

EPI-001 Chemical Structure

CAS NO. 227947-06-0

EPI-001是雄激素受体（AR）的拮抗剂，它通过与AR的N末端结构域（NTD）共价结合并阻断AR及其剪接变体（转录因子IC50）的转录活性所需的蛋白质相互作用抑制AR NTD反式激活6μM）

库存：现货

规格	价格	数量
10 mg	￥ 490.00
25 mg	￥ 1,050.00
50 mg	￥ 1,470.00

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生物活性

靶点信息

PPARγ	Androgen Receptor
N/A	6 μM

溶解度 *

In vitro	DMSO	72 mg/mL (182.32 mM)
	Water	Insoluble
	Ethanol	72 mg/mL (182.32 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.32 mL	126.62 mL	253.24 mL
0.5 mM	5.06 mL	25.32 mL	50.65 mL
1 mM	2.53 mL	12.66 mL	25.32 mL
5 mM	0.51 mL	2.53 mL	5.06 mL

*The above data is based on the productmolecular weight 394.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15814
作用机制	Antagonist (拮抗剂)
M. Wt	394.89
Formula	C21H27ClO5
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	227947-06-0
Synonyms	EPI001, EPI 001
SMILES	CC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O