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￥ 0.00 Epigenetics
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A-366
Catalog No. A15969 -
UNC 2400
Catalog No. A13282 -
EI1
Catalog No. A12711 -
AZ505 ditrifluoroacetate
Catalog No. A13169 SMYD2 抑制剂AZ505 ditrifluoroacetate是一种有效且高度选择性的致癌蛋白SMYD2抑制剂（IC50 = 0.12 uM），具有潜在的抗癌活性，是SMYD3的> 600倍（IC50> 83.3 uM）。DOT1L（IC50> 83.3 uM）；EZH2（IC50> 83.3 uM）。 了解更多 -
CPI-1205
Catalog No. A16357 -
EPZ031686
Catalog No. A16375 -
JQEZ5
Catalog No. A16961 -
PF-06726304
Catalog No. A16937 -
JNJ-64619178
Catalog No. A16861 Histone Methyltransferase 抑制剂JNJ-64619178是PRMT5抑制剂，在不同的体外和细胞条件下均具有高选择性和强效性（亚纳摩尔范围，PRMT5-MEP-50 IC50 = 0.14 nM），并具有良好的药代动力学和安全性。 了解更多 -
BIX-01338 hydrate
Catalog No. A21812 histone lysine methyltransferase inhibitorBIX-01338 hydrate is a histone lysine methyltransferase inhibitor. 了解更多 -
CPI-360
Catalog No. A15908 -
Flopropione
Catalog No. A16550 5-HT1A receptor antagonist/COMT inhibitorFlopropione是5-HT1A受体拮抗剂，也是儿茶酚-邻甲基转移酶（COMT）抑制剂。 了解更多 -
SMYD3-IN-1
Catalog No. A18572 SMYD3 inhibitorSMYD3-IN-1 (compound 29) is an irreversible and selective inhibitor of SMYD3 (SET and MYND domain containing 3), with an IC50 of 11.7 nM. 了解更多 -
Entacapone
Catalog No. A10355 COMT inhibitorEntacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment. 了解更多 -
CPUY074020
Catalog No. A12190 G9a inhibitorCPUY074020 is a potent G9a inhibitor with an IC50 of 2.18 μM, and possesses anti-proliferative activity . 了解更多 -
PF-06821497
Catalog No. A21388 EZH2 inhibitorPF-06821497 (compound 23a) is a potent, selective and orally active Enhancer of Zeste Homolog 2 (EZH2) inhibitor, with a Ki value <0.1 nM against mutant Y641N EZH2. Exhibits robust tumor growth inhibition. 了解更多 -
GSK2807 Trifluoroacetate
Catalog No. A21731 SMYD3 inhibitorGSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM. 了解更多 -
Tazemetostat hydrobromide
Catalog No. A21759 EZH2 inhibitorTazemetostat hydrobromide (EPZ-6438 hydrobromide) is a potent, selective and orally available EZH2 inhibitor. 了解更多 -
Entacapone sodium salt
Catalog No. A21888 COMT inhibitorEntacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment. 了解更多 -
MM-589 TFA
Catalog No. A21892 WDR5 and MLL protein-protein interaction inhibitorMM-589 TFA is a potent inhibitor of WD repeat domain 5 (WDR5) and mixed lineage leukemia (MLL) protein-protein interaction. 了解更多 -
MM-102 TFA
Catalog No. A21941 WDR5/MLL interaction inhibitorMM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide. 了解更多 -
Remodelin Hydrobromide
Catalog No. A14215 -
MG149
Catalog No. A14267 -
Histone Acetyltransferase Inhibitor II
Catalog No. A12331 cell permeable p300 inhibitorHistone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 ?M; Histone Acetyltransferase Inhibitor II can be used in cancer research. 了解更多 -
Decitabine
Catalog No. A10292 DNA Methyltransferase 抑制剂Decitabine是一种次甲基化剂，它通过抑制DNA甲基转移酶来使DNA次甲基化。 了解更多 -
Azacitidine(Vidaza)
Catalog No. A10105 DNMT 抑制剂Azacitidine (Vidaza)是DNA和RNA中使用的胞嘧啶核苷的化学类似物，主要用于治疗骨髓增生异常综合症（MDS）。 了解更多 -
SGI-110 (Guadecitabine)
Catalog No. A12744 -
SGI 1027
Catalog No. A14120 -
Procainamide HCl
Catalog No. A14240 -
RG108
Catalog No. A13054 -
O6-Benzylguanine
Catalog No. A13706 -
Nanaomycin A
Catalog No. A13477 -
Lomeguatrib
Catalog No. A12785
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