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INCB054329 Racemate
Catalog No. A21609 -
CPI-0610 carboxylic acid
Catalog No. A21714 BET inhibitorCPI-0610 carboxylic acid is a potent bromodomain and extra-terminal (BET) protein inhibitor. CPI-0610 carboxylic acid has the potential in the therapy of multiple myeloma. 了解更多 -
AZD5153 6-Hydroxy-2-naphthoic acid
Catalog No. A21852 BET/BRD4 bromodomain inhibitorAZD5153 6-Hydroxy-2-naphthoic acid is the 6-Hydroxy-2-naphthoic acid of AZD5153. AZD5153 is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor; disrupts BRD4 with an IC50 of 1.7 nM. 了解更多 -
Molibresib besylate
Catalog No. A21855 BET bromodomain inhibitorMolibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM. 了解更多 -
C646
Catalog No. A12815 -
GSK2801
Catalog No. A14015 -
GSK1324726A (I-BET726)
Catalog No. A14133 BET 抑制剂GSK1324726A (I-BET726)是一种新型、高效、选择性的BET蛋白小分子抑制剂，对BRD2（IC50 = 41 nM）、BRD3（IC50 = 31 nM）和BRD4（IC50 = 22 nM）具有高度的亲和力。 了解更多 -
GSK 525768A
Catalog No. A14134 GSK 525768A是GSK 525762A的对映体化合物，GSK 525762A是一种有效的小分子抑制剂，可破坏溴多糖BET家族（Brd2、Brd3和Brd4）的功能；GSK 525768A对BET没有活性。 了解更多 -
Anacardic Acid
Catalog No. A14226 -
Apabetalone (RVX-208)
Catalog No. A13956 BET bromodomain 抑制剂RVX-208是一种有效的BET溴结构域抑制剂，对BD2的IC50为0.510 uM，是BD1选择性的170倍。 了解更多 -
UNC 926 hydrochloride
Catalog No. A15367 -
BAZ2-ICR
Catalog No. A15947 -
EML 425
Catalog No. A16180 -
CeMMEC13
Catalog No. A16355 -
CPI-637
Catalog No. A16470 -
ABBV-744
Catalog No. A16831 -
BAY1238097
Catalog No. A16881 BET 抑制剂BAY1238097是一种有效的选择性BET抑制剂。BAY1238097与BET蛋白BRD上的乙酰化赖氨酸识别基序结合，从而防止BET蛋白与组蛋白之间的相互作用。 了解更多 -
HJB-97
Catalog No. A16872 -
ARV-825
Catalog No. A16859 -
PLX51107
Catalog No. A18345 selective BET inhibitorPLX51107 is a potent and selective BET inhibitor, with Kds of 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1, and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively; PLX51107 also interacts with the bromodomains of CBP and EP300 (Kd, in the 100 nM range). 了解更多 -
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最新产品
Mivebresib (ABBV-075)
Catalog No. A17226 BET inhibitorMivebresib, also known as ABBV-075, is a potent BET inhibitor (bromodomain (BRD)-containing proteind) with potential antineoplastic activity. 了解更多 -
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P300/CBP-IN-3
Catalog No. A18544 p300/CBP histone acetyltransferase inhibitorP300/CBP-IN-3, a p300/CBP histone acetyltransferase inhibitor. 了解更多 -
T-3775440 hydrochloride
Catalog No. A18340 LSD1 inhibitorT-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM. 了解更多 -
QC6352
Catalog No. A19477 -
NCGC00244536
Catalog No. A13025 -
Toxoflavin
Catalog No. A12174 KDM4A inhibitorToxoflavin (Xanthothricin) is an antagonist of transcription factor 4 (TCF4)/β-catenin complex, also acts as an inhibitor of KDM4A, with antitumor activity. 了解更多 -
ORY-1001(trans)
Catalog No. A21622 KDM1A/LSD1 inhibitorORY-1001 trans is a selective irreversible lysine (K)-specific demethylase 1A (KDM1A/LSD1) inhibitor. 了解更多 -
GSK-LSD1 dihydrochloride
Catalog No. A21815 LSD1 inhibitorGSK-LSD1 dihydrochloride is a potent, selective and irreversible lysine specific demethylase 1 (LSD1) inhibitor with an IC50 of 16 nM. 了解更多
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