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G Protein

26 个项目

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  1. AMG 837
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    AMG 837

    Catalog No. A21160
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    GPR40 agonist
    AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多
  2. MK-0354
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    MK-0354

    Catalog No. A22008
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    GPR109a receptor agonist
    MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. 了解更多
  3. AMG 837 sodium salt
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    AMG 837 sodium salt

    Catalog No. A21793
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    GPR40 agonist
    AMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多
  4. AM-4668
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    AM-4668

    Catalog No. A21778
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    GPR40 agonist
    AM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively. 了解更多
  5. (1R,2R)-2-PCCA(hydrochloride)
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    (1R,2R)-2-PCCA(hydrochloride)

    Catalog No. A21655
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    GPR88 receptor agonist
    (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多
  6. GPR40 Activator 2
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    GPR40 Activator 2

    Catalog No. A21642
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    GPR40 activator
    GPR40 Activator 2 is a potent GPR40 activator from patents WO 2012147516 A1, WO 2012046869A1 and WO 2011078371 A1. 了解更多
  7. AF64394
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    AF64394

    Catalog No. A21574
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    GPR3 inverse agonist
    AF64394 is a GPR3 inverse agonist, with a pIC50 of 7.3. 了解更多
  8. AM-1638
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    AM-1638

    Catalog No. A21505
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    GPR40/FFA1 full agonist
    AM-1638 is a potent and orally bioavailable GPR40/FFA1 full agonist with an EC50 of 0.16 μM. 了解更多
  9. GLPG0974
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    GLPG0974

    Catalog No. A21466
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    FFA2/GPR43 antagonist
    GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM. 了解更多
  10. GPR40 Activator 1
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    GPR40 Activator 1

    Catalog No. A21154
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    GPR40 activator
    GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. 了解更多
  11. PSN632408
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    PSN632408

    Catalog No. A20902
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    GPR119 receptors agonist
    PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多
  12. Kynurenic acid sodium
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    Kynurenic acid sodium

    Catalog No. A20000
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    GPR35/CXCR8 agonist
    Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多
  13. GPR35 agonist 1
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    GPR35 agonist 1

    Catalog No. A12462
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    GPR35/CXCR8 agonist
    GPR35 agonist 1 (compound 50) is a potent and specific G protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM, displays good druggability. 了解更多
  14. LY2922470
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    LY2922470

    Catalog No. A12181
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    GPR40 agonist
    LY2922470 is a potent, selective and orally available agonist of the G protein-coupled receptor 40 (GPR40), with EC50s of 7 nM, 1 nM and 3 nM for human GPR40, mouse GPR40 and rat GPR40, respectively. 了解更多
  15. G15
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    G15

    Catalog No. A13675
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    GPER/GPR30 antagonist
    G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM. 了解更多
  16. GPR4 antagonist 1
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    GPR4 antagonist 1

    Catalog No. A12340
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    GPR4 antagonist
    GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM. 了解更多
  17. DJ-V-159
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    DJ-V-159

    Catalog No. A18853
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    GPRC6A agonist
    DJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A). 了解更多
  18. GW-1100
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    GW-1100

    Catalog No. A11445
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    GPR40 antagonist
    GW-1100 is a selective GPR40 antagonist with a pIC50 of 6.9. 了解更多
  19. Kynurenic acid
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    Kynurenic acid

    Catalog No. A16581
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    GPR35/CXCR8 拮抗剂
    Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多
  20. TM N1324
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    TM N1324

    Catalog No. A17038
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    GPR39 激动剂
    TM N1324是G蛋白偶联受体39（GPR39）的激动剂，在Zn2+存在下的EC50为9 nM/5 nM，而对于人/鼠GPR39，则在Zn2+不存在时的EC50为280 nM/180 nM。 了解更多
  21. CID16020046
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    CID16020046

    Catalog No. A16818
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    GPR55 拮抗剂
    CID16020046是一种选择性的GPR55拮抗剂，在酵母中抑制GPR55的组成活性，IC50为150 nM。它对其他广谱GPCRs、离子通道、激酶和核受体表现出弱活性。 了解更多
  22. MK-6892
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    MK-6892

    Catalog No. A12982
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    GPR109A 激动剂
    MK-6892是高亲和力烟酸（NA）受体GPR109A的有效，选择性和完全激动剂。人GPR109A的MK-6892的Ki和GTPγSEC 50分别为4 nM和16 nM。 了解更多
  23. CCG 50014
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    CCG 50014

    Catalog No. A16432
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    RGS4 抑制剂
    CCG 50014是RGS4的有效和选择性抑制剂，IC50为30 nM。 了解更多
  24. CASIN
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    CASIN

    Catalog No. A12912
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    Cdc42 GTPase 抑制剂
    CASIN是一种新型有效的Cdc42抑制剂。 了解更多
  25. CCG-63802
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    CCG-63802

    Catalog No. A11373
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    CCG-63802是G蛋白信号(RGS)蛋白调节因子的可逆抑制剂。在RGS蛋白中具有选择性，在RGS4中具有最大效力。 了解更多
  26. QS 11
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    QS 11

    Catalog No. A11228
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    ATPase and GTPase 抑制剂
    QS-11是ADP-核糖基化因子1（ARFGAP1）抑制剂的GTPase活化蛋白。 了解更多

26 个项目

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  1. Inhibitor (抑制剂) (3)
  2. Agonist (激动剂) (15)
  3. Antagonist (拮抗剂) (5)
  4. Activator (激活剂) (2)
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