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￥ 0.00 GABA Receptors
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Vigabatrin
Catalog No. A15277 GABA-transaminase 抑制剂Vigabatrin是抑制性神经递质β-氨基丁酸（GABA）的结构类似物，它不可逆地抑制GABA转氨酶对GABA的分解代谢。 了解更多 -
MRK-016
Catalog No. A12046 GABAA α5 receptor agonistMRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多 -
Acamprosate calcium
Catalog No. A11308 GABA receptor agonistAcamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. 了解更多 -
(R)-Baclofen
Catalog No. A16680 GABAB receptor agonist(R)-Baclofen(STX209) is a selective GABAB receptor agonist. 了解更多 -
Basmisanil
Catalog No. A21321 GABAAα5 modulatorBasmisanil is a highly selective GABAAα5 negative allosteric modulator. 了解更多 -
CP-409092 hydrochloride
Catalog No. A21397 GABAA receptor partial agonistCP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. 了解更多 -
Gaboxadol hydrochloride
Catalog No. A21730 GABAA receptors agonistGaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. 了解更多 -
Piperazine
Catalog No. A16171 -
Lorediplon
Catalog No. A13449 -
(-)-Securinine
Catalog No. A17102 GABA receptor 拮抗剂(-)-Securinine是一种最初从S. suffructicosa分离的生物碱。Securinine是一种特定的GABA受体拮抗剂，已发现在体内具有显着的CNS活性。 了解更多 -
Afloqualone
Catalog No. A17276 GABA receptor agonistAfloqualone, also known as HQ-495, is a centrally acting muscle relaxant. Afloqualone inhibits vestibular nystagmus probably due to both inhibition of selective polysynaptic transmission and enhancement of the effects of GABA and glycine in the lateral vestibular nucleus (LVN), and its GABA-enhancing effect is thought to be attributable to the increased sensitivity of GABA receptors of the LVN neuron site. 了解更多 -
Homotaurine
Catalog No. A17944 GABA receptor agonistTramiprosate, also known as homotaurine, is a gamma-Aminobutyric acid (GABA) receptor agonist and a glycosaminoglycan mimetic used in the treatment of Alzheimer's disease. 了解更多 -
Baclofen
Catalog No. A18248 GABA agonistBaclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing It acts at spinal and supraspinal sites, reducing excitatory transmission. 了解更多 -
Dihydromyricetin (Ampeloptin)
Catalog No. A10252 -
Nefiracetam (Translon)
Catalog No. A10631 Nefiracetam (Translon)是认知增强剂。它激活L/N型钙通道，胆碱能，单胺能和GABA能系统。 了解更多 -
SKF 89976A HCl
Catalog No. A10849 GABA uptake 抑制剂SKF 89976A HCl是一种有效的GABA吸收抑制剂，hGAT-1，rGAT-2，hGAT-3和hBGT-1的IC50分别为0.13、550、944和7210μM。 了解更多 -
Flumazenil
Catalog No. A10397 Benzodiazepine 拮抗剂Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂，但在人类中很少或没有激动剂活性。 了解更多 -
(+)-Bicuculline
Catalog No. A12590 -
AWD 131-138
Catalog No. A13726 -
2-Hydroxysaclofen
Catalog No. A13696 -
Cloflubicyne
Catalog No. A13932 -
a5IA
Catalog No. A14343 -
Guvacine hydrochloride
Catalog No. A13613 GABA uptake 抑制剂Guvacine hydrochloride可抑制GABA的摄取（hGABA T-1，rGABA T-2，hGABA T-3和hBGT-1的IC50值分别为14、58、119和1870 uM）。 了解更多 -
Muscimol hydrobromide
Catalog No. A13459 GABA(A) receptor 激动剂Muscimol hydrobromide是抗抑郁药氟西汀的活性代谢产物，可抑制5-羟色胺的摄取，pKi值为7.35.1。诺氟西汀的S-对映体的5-羟色胺再摄取阻断效能比R-对映体高20倍（分别为pKis = 7.86与6.51）。 了解更多
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