主页 /
GLP-1R Antagonist 1

GLP-1R Antagonist 1

Name: GLP-1R Antagonist 1
SKU: A20679

目录号: A20679

glucagon-like peptide 1 receptor antagonist

GLP-1R Antagonist 1 Chemical Structure

CAS NO. 488097-06-9

GLP-1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non-competitive antagonist of glucagon-like peptide 1 receptor (GLP-1R), with an IC50 of 650 nM.

库存：现货

规格	价格	数量
1 mg	￥ 2,240.00
5 mg	￥ 6,720.00
10 mg	￥ 11,200.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

GLP-1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non-competitive antagonist of glucagon-like peptide 1 receptor (GLP-1R), with an IC50 of 650 nM.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	22.69 mL	113.45 mL	226.9 mL
0.5 mM	4.54 mL	22.69 mL	45.38 mL
1 mM	2.27 mL	11.34 mL	22.69 mL
5 mM	0.45 mL	2.27 mL	4.54 mL

*The above data is based on the productmolecular weight 440.73. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A20679
M. Wt	440.73
Formula	C16H11ClF6N4O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	488097-06-9
SMILES	O=C1C2=C(NC(C3=CC=C(Cl)C=C3)=NC2(C(F)(F)F)C(F)(F)F)N(C)C(N1C)=O