Guanabenz acetate

Name: Guanabenz acetate
SKU: A13635

目录号: A13635

2A-AR adrenergic 激动剂

Guanabenz acetate Chemical Structure

CAS NO. 23256-50-0

Guanabenz acetate是a2A-AR肾上腺素能激动剂和IGRS（咪唑啉I2结合位点）选择性配体。

库存：现货

规格	价格	数量
100 mg	￥ 665.00
500 mg	￥ 2,800.00
10mM * 1mL in DMSO	￥ 434.00

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生物活性

Guanabenz acetate是a2A-AR肾上腺素能激动剂和IGRS（咪唑啉I2结合位点）选择性配体。

靶点信息

α2a-adrenergic receptor	α2b-adrenergic receptor	α2c-adrenergic receptor
8.25(pEC50)	7.01(pEC50)	<5(pEC50)

溶解度 *

In vitro (25°C)	DMSO	56 mg/mL (192.35 mM)
	Water	Insoluble
	Ethanol	5 mg/mL (17.17 mM)
In vivo	4% DMSO+30% PEG 300+ddH2O	4 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	34.35 mL	171.74 mL	343.49 mL
0.5 mM	6.87 mL	34.35 mL	68.7 mL
1 mM	3.43 mL	17.17 mL	34.35 mL
5 mM	0.69 mL	3.43 mL	6.87 mL

*The above data is based on the productmolecular weight 291.13. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13635
作用机制	Agonist (激动剂)
M. Wt	291.13
Formula	C10H12Cl2N4O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	23256-50-0
SMILES	CC(=O)O.C1=CC(=C(C(=C1)Cl)/C=N/N=C(N)N)Cl