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￥ 0.00 Histamine Receptors
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Decloxizine
Catalog No. A20964 histamine 1 receptor antagonistDecloxizine(UCB-1402; NSC289116) is a histamine 1 receptor antagonist. 了解更多 -
GSK189254A
Catalog No. A22005 histamine H3 receptor antagonistGSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. 了解更多 -
Niperotidine
Catalog No. A21981 histamine H2-receptor antagonistNiperotidine is a histamine H2-receptor antagonist. 了解更多 -
JNJ-5207852
Catalog No. A21480 histamine H3 receptor antagonistJNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively. 了解更多 -
PF-03654746 Tosylate
Catalog No. A21434 histamine H3 receptor antagonistPF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
PF-03654746
Catalog No. A21429 histamine H3 receptor antagonistPF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
Toreforant
Catalog No. A21058 histamine H4 receptor (H4R) antagonistToreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多 -
Chlorcyclizine hydrochloride
Catalog No. A18025 histamine H1 antagonistChlorcyclizine hydrochloride is a histamine H1 antagonist. 了解更多 -
H4 Receptor antagonist 1
Catalog No. A18929 histamine H4 receptor inverse agonistH4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多 -
Cyproheptadine hydrochloride
Catalog No. A16169 -
Lidocaine hydrochloride
Catalog No. A16132 -
CarbinoxaMine Maleate
Catalog No. A16129 histamine-H1 receptor blocking agentCarbinoxamine maleate是一种具有抗组胺和抗胆碱能特性的组胺-H1受体阻断剂。 了解更多 -
Bavisant dihydrochloride hydrate
Catalog No. A15016 -
Bavisant dihydrochloride
Catalog No. A15015 -
Pitolisant oxalate
Catalog No. A15214 Nonimidazole inverse 激动剂Pitolisant oxalate是一种在重组人H3受体上的新型，有效且选择性的壬咪唑反向激动剂（Ki = 0.16 nM）。 了解更多 -
Pitolisant hydrochloride
Catalog No. A15213 Nonimidazole inverse 激动剂Pitolisant hydrochloride是一种在重组人H3受体（Ki = 0.16 nM）处新颖，有效且选择性的壬二唑反向激动剂。 了解更多 -
Ebrotidine
Catalog No. A15075 -
Clemizole hydrochloride
Catalog No. A15047 H1 histamine receptor 拮抗剂Clemizole hydrochloride是H1组胺受体的拮抗剂，对NS4B RNA结合的IC50值为8 mM。 了解更多 -
Alcaftadine
Catalog No. A16393 H1 histamine receptor 拮抗剂Alcaftadine是H1受体的高亲和力配体，其pKi（8.5）与其他H1抗组胺药相当。Alcaftadine还是H2和H4受体的拮抗剂，对H3受体没有亲和力。 了解更多 -
Antazoline HCl
Catalog No. A16411 -
Azatadine dimaleate
Catalog No. A16418 -
Cyclizine 2HCl
Catalog No. A16472 -
Terfenadine
Catalog No. A17373 H1 histamine receptor antagonistTerfenadine ((??)-Terfenadine) is a potent open-channel blocker of hERG with an IC50 of 204 nM. Terfenadine, an H1 histamine receptor antagonist, acts as a potent apoptosis inducer in melanoma cells through modulation of Ca2+ homeostasis. Terfenadine induces ROS-dependent apoptosis, simultaneously activates Caspase-4, -2, -9 and induces p73, Noxa. 了解更多 -
Levocetirizine Dihydrochloride
Catalog No. A17440 L-isomer of cetirizine and histamine H1 receptor antagonistLevocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多 -
Hydroxyzine pamoate
Catalog No. A17712 Histamine H1 receptor antagonistHydroxyzine pamoate is an histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does cause drowsiness. 了解更多 -
Diphenylpyraline hydrochloride
Catalog No. A17717 antihistamineDiphenylpyraline hydrochloride is a first-generation antihistamine with anticholinergic effects of the diphenylpiperidine class. 了解更多 -
Acrivastine
Catalog No. A17746 Histamine 1 receptor antagonistAcrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. 了解更多 -
Mebhydrolin napadisylate
Catalog No. A17997 -
Mequitazine
Catalog No. A18206 Histamine H1 antagonistMequitazine is a potent histamine H1 antagonist or antihistamine. It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. 了解更多 -
Ciproxifan maleate
Catalog No. A11117 -
Azelastine HCl (Allergodil)
Catalog No. A10117 Azelastine HCl (Allergodil)是有效的第二代选择性组胺拮抗剂（组胺-H1-受体拮抗剂）。 了解更多 -
Clemastine fumarate
Catalog No. A10226 Histamine Receptor antagonisClemastine fumarate是一种选择性的组胺H1拮抗剂。它与组胺H1受体结合，从而阻断了内源性组胺的作用，从而暂时缓解了由组胺引起的阴性症状。 了解更多 -
Cyproheptadine hydrochloride
Catalog No. A11709 Cyproheptadine hydrochloride 是 5-HT2 受体拮抗剂，IC50为0.6 nM。 了解更多 -
Orphenadrine citrate
Catalog No. A11712 -
Asenapine maleate
Catalog No. A10091 H1 拮抗剂Asenapine maleate平对多种受体具有高亲和力（pKi），包括5-羟色胺5-HT1A（8.6），5-HT1B（8.4），5-HT2A（10.2），5-HT2B（9.8），5-HT2C（10.5），5 -HT5A（8.8），5-HT6（9.5）和5-HT7（9.9）受体，肾上腺素α1（8.9），α2A（8.9），α2B（9.5）和α2C（8.9）受体，多巴胺D1（ 8.9），D2（8.9），D3（9.4）和D4（9.0）受体以及组胺H1（9.0）和H2（8.2）受体。 了解更多 -
Cetirizine Dihydrochloride
Catalog No. A10195 Cetirizine Dihydrochloride是第二代抗组胺药，是羟嗪的主要代谢产物，是用于治疗过敏，花粉症，血管性水肿和荨麻疹的消旋选择性H1受体反向激动剂。 了解更多 -
Chlorpheniramine maleate
Catalog No. A10205 Chlorpheniramine maleate是用于预防过敏性疾病如鼻炎和荨麻疹症状的第一代烷基胺抗组胺药。 了解更多 -
Bepotastine Besilate
Catalog No. A11340 -
Roxatidine acetate hydrochloride
Catalog No. A11921 Roxatidine acetate hydrochloride是一种用于溃疡治疗的组胺H2受体拮抗剂。 了解更多 -
Rupatadine Fumarate
Catalog No. A12356 PAFR 抑制剂/H1 receptor 抑制剂Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂，Ki分别为550和102 nM。 了解更多 -
Rupatadine
Catalog No. A11222 PAFR 抑制剂/H1 receptor 抑制剂Rupatadine是PAFR和组胺（H1）受体的抑制剂，Ki分别为550和102 nM。 了解更多 -
Loratadine
Catalog No. A10538 Loratadine是一种非镇静抗组胺药，抑制组胺诱导的内皮细胞分泌IL-6和IL-8的活性。氯雷他定是一种选择性外周组胺h1受体拮抗剂，IC50 > 32 μM。 了解更多 -
Fexofenadine HCl
Catalog No. A11859 COX 抑制剂/histamine H1 receptor 激动剂Fexofenadine Hydrochloride是一种抗组胺药，可抑制Cox-1，Cox-2，并且是组胺H1受体激动剂，IC50为246 nM。 了解更多
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