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￥ 0.00 Histamine Receptors
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Immethridine hydrobromide
Catalog No. A13641 histamine H3 receptor 激动剂Immethridine hydrobromide是一种强而高选择性的组胺H3受体激动剂（pEC50 = 9.74），其选择性是H4受体的300倍（pKi值分别为9.07和6.61）。 了解更多 -
A 943931 2HCl
Catalog No. A13442 -
Cetirizine
Catalog No. A15041 -
Clemizole hydrochloride
Catalog No. A15047 H1 histamine receptor 拮抗剂Clemizole hydrochloride是H1组胺受体的拮抗剂，对NS4B RNA结合的IC50值为8 mM。 了解更多 -
Ebrotidine
Catalog No. A15075 -
Pitolisant hydrochloride
Catalog No. A15213 Nonimidazole inverse 激动剂Pitolisant hydrochloride是一种在重组人H3受体（Ki = 0.16 nM）处新颖，有效且选择性的壬二唑反向激动剂。 了解更多 -
Pitolisant oxalate
Catalog No. A15214 Nonimidazole inverse 激动剂Pitolisant oxalate是一种在重组人H3受体上的新型，有效且选择性的壬咪唑反向激动剂（Ki = 0.16 nM）。 了解更多 -
Bavisant dihydrochloride
Catalog No. A15015 -
Bavisant dihydrochloride hydrate
Catalog No. A15016 -
CarbinoxaMine Maleate
Catalog No. A16129 histamine-H1 receptor blocking agentCarbinoxamine maleate是一种具有抗组胺和抗胆碱能特性的组胺-H1受体阻断剂。 了解更多 -
Lidocaine hydrochloride
Catalog No. A16132 -
Cyproheptadine hydrochloride
Catalog No. A16169 -
Alcaftadine
Catalog No. A16393 H1 histamine receptor 拮抗剂Alcaftadine是H1受体的高亲和力配体，其pKi（8.5）与其他H1抗组胺药相当。Alcaftadine还是H2和H4受体的拮抗剂，对H3受体没有亲和力。 了解更多 -
Antazoline HCl
Catalog No. A16411 -
Azatadine dimaleate
Catalog No. A16418 -
Cyclizine 2HCl
Catalog No. A16472 -
Terfenadine
Catalog No. A17373 H1 histamine receptor antagonistTerfenadine ((??)-Terfenadine) is a potent open-channel blocker of hERG with an IC50 of 204 nM. Terfenadine, an H1 histamine receptor antagonist, acts as a potent apoptosis inducer in melanoma cells through modulation of Ca2+ homeostasis. Terfenadine induces ROS-dependent apoptosis, simultaneously activates Caspase-4, -2, -9 and induces p73, Noxa. 了解更多 -
Levocetirizine Dihydrochloride
Catalog No. A17440 L-isomer of cetirizine and histamine H1 receptor antagonistLevocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多 -
Hydroxyzine pamoate
Catalog No. A17712 Histamine H1 receptor antagonistHydroxyzine pamoate is an histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does cause drowsiness. 了解更多 -
Diphenylpyraline hydrochloride
Catalog No. A17717 antihistamineDiphenylpyraline hydrochloride is a first-generation antihistamine with anticholinergic effects of the diphenylpiperidine class. 了解更多 -
Acrivastine
Catalog No. A17746 Histamine 1 receptor antagonistAcrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. 了解更多 -
Mebhydrolin napadisylate
Catalog No. A17997 -
Mequitazine
Catalog No. A18206 Histamine H1 antagonistMequitazine is a potent histamine H1 antagonist or antihistamine. It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. 了解更多 -
Ciproxifan maleate
Catalog No. A11117 -
Azelastine HCl (Allergodil)
Catalog No. A10117 Azelastine HCl (Allergodil)是有效的第二代选择性组胺拮抗剂（组胺-H1-受体拮抗剂）。 了解更多 -
Clemastine fumarate
Catalog No. A10226 Histamine Receptor antagonisClemastine fumarate是一种选择性的组胺H1拮抗剂。它与组胺H1受体结合，从而阻断了内源性组胺的作用，从而暂时缓解了由组胺引起的阴性症状。 了解更多 -
Cyproheptadine hydrochloride
Catalog No. A11709 Cyproheptadine hydrochloride 是 5-HT2 受体拮抗剂，IC50为0.6 nM。 了解更多 -
Orphenadrine citrate
Catalog No. A11712 -
Asenapine maleate
Catalog No. A10091 H1 拮抗剂Asenapine maleate平对多种受体具有高亲和力（pKi），包括5-羟色胺5-HT1A（8.6），5-HT1B（8.4），5-HT2A（10.2），5-HT2B（9.8），5-HT2C（10.5），5 -HT5A（8.8），5-HT6（9.5）和5-HT7（9.9）受体，肾上腺素α1（8.9），α2A（8.9），α2B（9.5）和α2C（8.9）受体，多巴胺D1（ 8.9），D2（8.9），D3（9.4）和D4（9.0）受体以及组胺H1（9.0）和H2（8.2）受体。 了解更多 -
Cetirizine Dihydrochloride
Catalog No. A10195 Cetirizine Dihydrochloride是第二代抗组胺药，是羟嗪的主要代谢产物，是用于治疗过敏，花粉症，血管性水肿和荨麻疹的消旋选择性H1受体反向激动剂。 了解更多 -
Chlorpheniramine maleate
Catalog No. A10205 Chlorpheniramine maleate是用于预防过敏性疾病如鼻炎和荨麻疹症状的第一代烷基胺抗组胺药。 了解更多 -
Astemizole
Catalog No. A13899 H1-receptor 拮抗剂Astemizole是一种有效的抗组胺药物（H1-受体拮抗剂，IC50 = 4 nM），对多巴胺，5-HT和毒蕈碱乙酰胆碱受体具有选择性。该化合物显示出有效的hERG K+通道阻断活性（IC50 = 0.9 nM），在体外多药耐药菌株中具有抗疟疾活性（IC50 = 227-734 nM），并已被用作分子伴侣来纠正折叠缺陷并恢复蛋白质功能 hERG通道的某些突变形式。 了解更多 -
Promethazine HCl
Catalog No. A14248 -
Olopatadine hydrochloride
Catalog No. A10671 Olopatadine hydrochloride是一种双重作用的组胺H1受体拮抗剂和肥大细胞稳定剂。 了解更多 -
Fexofenadine HCl
Catalog No. A11859 COX 抑制剂/histamine H1 receptor 激动剂Fexofenadine Hydrochloride是一种抗组胺药，可抑制Cox-1，Cox-2，并且是组胺H1受体激动剂，IC50为246 nM。 了解更多 -
Loratadine
Catalog No. A10538 Loratadine是一种非镇静抗组胺药，抑制组胺诱导的内皮细胞分泌IL-6和IL-8的活性。氯雷他定是一种选择性外周组胺h1受体拮抗剂，IC50 > 32 μM。 了解更多 -
Rupatadine
Catalog No. A11222 PAFR 抑制剂/H1 receptor 抑制剂Rupatadine是PAFR和组胺（H1）受体的抑制剂，Ki分别为550和102 nM。 了解更多
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