Histone Demethylases
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GSK-LSD1 dihydrochloride
Catalog No. A21815 LSD1 inhibitorGSK-LSD1 dihydrochloride is a potent, selective and irreversible lysine specific demethylase 1 (LSD1) inhibitor with an IC50 of 16 nM. 了解更多 -
ORY-1001(trans)
Catalog No. A21622 KDM1A/LSD1 inhibitorORY-1001 trans is a selective irreversible lysine (K)-specific demethylase 1A (KDM1A/LSD1) inhibitor. 了解更多 -
Toxoflavin
Catalog No. A12174 KDM4A inhibitorToxoflavin (Xanthothricin) is an antagonist of transcription factor 4 (TCF4)/β-catenin complex, also acts as an inhibitor of KDM4A, with antitumor activity. 了解更多 -
NCGC00244536
Catalog No. A13025 -
QC6352
Catalog No. A19477 -
T-3775440 hydrochloride
Catalog No. A18340 LSD1 inhibitorT-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM. 了解更多 -
GSK467
Catalog No. A18807 KDM5B (JARID1B or PLU1) inhibitorGSK467 is a potent and selective inhibitor of KDM5 (also known as JARID1) with a Ki of 10 nM, shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members. GSK467 exploits unique binding modes. 了解更多 -
CBB1007
Catalog No. A16374 -
2,4-Pyridinedicarboxylic Acid
Catalog No. A16372 KDM 抑制剂2,4-Pyridinedicarboxylic Acid是针对JMJD2A(KDM4A),KDM4C,KDM4E(IC50、1.4μM),KDM5B(IC50、3μM),KDM6A和 其他的2-氧合酶。 了解更多 -
CPI 455
Catalog No. A16178 -
ORY-1001 (RG-6016)
Catalog No. A15893 LSD1 抑制剂ORY-1001 (RG-6016)是一种活性的选择性赖氨酸脱甲基酶LSD1/KDM1A抑制剂,IC50 <20 nM,对相关FAD依赖性氨氧化酶具有高选择性。 了解更多 -
SP2509 (HCI-2509)
Catalog No. A14443 LSD1 抑制剂SP2509 (HCI-2509)是一种新型组蛋白脱甲基酶LSD1(KDM1A)拮抗剂,IC50为13 nM。对MAO-A和MAO-B没有抑制作用。 了解更多 -
GSK2879552
Catalog No. A15547 -
Tranylcypromine hydrochloride
Catalog No. A13358 LSD1/BHC110 & MAO 抑制剂Tranylcypromine hydrochloride是一种非选择性的MAO-A/B抑制剂。 了解更多 -
OG-L002
Catalog No. A13246