Istradefylline (KW-6002)

Name: Istradefylline (KW-6002)
SKU: A11451

目录号: A11451

A2A 拮抗剂

Product Citations (1)

Istradefylline (KW-6002) Chemical Structure

CAS NO. 155270-99-8

Istradefylline (KW-6002)是A2A受体的选择性拮抗剂。

库存：现货

规格	价格	数量
5 mg	￥ 385.00
10 mg	￥ 490.00
25 mg	￥ 595.00
50 mg	￥ 770.00

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生物活性

Istradefylline (KW-6002)是A2A受体的选择性拮抗剂。

靶点信息

Adenosine A2A receptor
2.2 nM(Ki)

溶解度 *

In vitro (25°C)	DMSO	5 mg/mL (13 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	30% propylene glycol, 5% Tween 80, 65% D5W	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	26.01 mL	130.07 mL	260.15 mL
0.5 mM	5.2 mL	26.01 mL	52.03 mL
1 mM	2.6 mL	13.01 mL	26.01 mL
5 mM	0.52 mL	2.6 mL	5.2 mL

*The above data is based on the productmolecular weight 384.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11451
作用机制	Antagonist (拮抗剂)
M. Wt	384.4
Formula	C20H24N4O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	155270-99-8
Synonyms	KW-6002,KW6002
SMILES	CCN1C2=C(C(=O)N(C1=O)CC)N(C(=N2)/C=C/C3=CC(=C(C=C3)OC)OC)C