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Diazepinomicin
Catalog No. A12891 -
L-779450
Catalog No. A13525 -
Regorafenib monohydrate
Catalog No. A15218 Tyrosine kinase 抑制剂Regorafenib monohydrate是VEGFR1/VEGFR2/VEGFR3/PDGFRβ/Kit/RET和Raf-1的多靶点抑制剂，IC50分别为13 nM/4.2 nM/46 nM/22 nM/7 nM/1.5 nM和2.5 nM。 了解更多 -
Locostatin
Catalog No. A16079 -
LXH254
Catalog No. A16841 -
Lifirafenib (BGB-283)
Catalog No. A16844 BRAF 抑制剂Lifirafenib (BGB-283)，也称为Beigene-283，在生化分析中有效抑制RAF家族激酶和EGFR活性，重组BRAFV600E激酶结构域，EGFR和EGFR T790M/L858R突变体的IC50值为23、29和495 nM。 了解更多 -
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最新产品
AZ304
Catalog No. A17225 dual BRAF 抑制剂AZ304 is a potent dual BRAF inhibitor targeting the kinase domains of wild type BRAF, V600E mutant BRAF. AZ304 exerted potent inhibitory effects on both wild type and V600E mutant forms of the serine/threonine-protein kinase BRAF, with IC50 values of 79?nM and 38?nM, respectively. 了解更多 -
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OTS514
Catalog No. A16023 -
HI TOPK 032
Catalog No. A16042 TOPK 抑制剂HI-TOPK-032是一种有效的选择性TOPK抑制剂。在体外，HI-TOPK-032强烈抑制TOPK激酶活性，但对细胞外信号调节激酶1（ERK1），c-jun-NH2-激酶1或p38激酶活性影响很小。 了解更多 -
CGP 57380
Catalog No. A13883 -
Cercosporamide
Catalog No. A15362 Mnk2/JAK3 抑制剂Cercosporamide是一种USnic酰胺，最初在Cercosporidium henningsii中被鉴定为宿主选择性植物毒素和广谱抗真菌剂，并且是MAP激酶相互作用激酶2（Mnk2；IC50 = 11 nM），JAK3（IC50 = 31）和Mnk1（IC50 = 116 nM）。 了解更多
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