Metabotropic glutamate receptors (mGluR)

15 个项目

每页

设置降序顺序
  1. VU0652835

    Catalog No. A18885
    Quick View
    mGlu5 modulator
    VU0652835 is a metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 of 81 nM. 了解更多
  2. VU 0364770

    Catalog No. A12139
    Quick View
    mGlu4 receptors modulator
    VU 0364770是mGlu4受体的正变构调节剂,在表达mGlu4的HEK 293细胞中EC50值为290 nM。 了解更多
  3. VU0364289

    Catalog No. A15832
    Quick View
    mGluR5 Modulator
    VU0364289是新型N-芳基哌嗪mGlu5阳性变构调节剂。 了解更多
  4. JNJ 42153605

    Catalog No. A14330
    Quick View
    mGluR-2 modulator
    JNJ-42153605是亲代谢型谷氨酸2受体的正变构调节剂。 了解更多
  5. ADX-47273

    Catalog No. A11181
    Quick View
    mGluR5 modulator
    ADX-47273是一种有效的,特异性的mGlu5正变构调节剂(PAM)EC50为0.17 μM,对其他亚型没有作用活性。 了解更多
  6. BINA

    Catalog No. A11126
    Quick View
    mGluR2 modulator
    BINA是mGlu2的选择性正构构调节剂(在表达人mGlu2的CHO细胞中EC50 = 33.2 nM)。 了解更多
  7. VU 0364439

    Catalog No. A12664
    Quick View
    GluR modulator
    VU 0364439是mGlu4受体的正变构调节剂(PAM)(对于人mGlu4,体外EC50 = 19.8 nM)。 了解更多
  8. VU 0361737

    Catalog No. A12467
    Quick View
    mGlu4 receptors modulator
    VU 0361737是mGluR-4的选择性正变构调节剂(人和大鼠受体的EC50值分别为240和110 nM)。 了解更多
  9. Basimglurant

    Catalog No. A21225
    Quick View
    mGlu5 negative allosteric modulator
    Basimglurant (RG7090) is a potent, selective and orally available mGlu5 negative allosteric modulator with a Kd of 1.1 nM. 了解更多
  10. (R)-ADX-47273

    Catalog No. A21887
    Quick View
    mGluR5 positive allosteric modulator
    (R)-ADX-47273 is a potent mGluR5 positive allosteric modulator, with an EC50 of 168 nM for potentiation . 了解更多
  11. TCN238

    Catalog No. A21191
    Quick View
    mGlu4 receptor modulator
    TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM. 了解更多
  12. Lu AF21934

    Catalog No. A12140
    Quick View
    mGlu4 receptor modulator
    Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多
  13. BMT-145027

    Catalog No. A12457
    Quick View
    mGluR5 positive allosteric modulator
    BMT-145027 is an mGluR5 positive allosteric modulator without inherent agonist activity, exhibits an EC50 of 47 nM. 了解更多
  14. CBiPES HCl

    Catalog No. A15811
    Quick View
    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂,IC50值为98.2 nM。 了解更多
  15. CPPHA

    Catalog No. A15053
    Quick View
    mGluR1 modulator
    CPPHA是mGluR5受体的选择性正变构调节剂。 了解更多

15 个项目

每页

设置降序顺序
Rewards