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Metabotropic glutamate receptors (mGluR)

15 个项目

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  1. DL-AP3
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    DL-AP3

    Catalog No. A15378
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    mGluR1 拮抗剂
    DL-AP3是D-AP3和L-AP3的外消旋制剂，是磷酸丝氨酸磷酸酶的抑制剂和代谢型谷氨酸受体（mGluR）的拮抗剂，阻断了由mGluR介导的磷酸肌醇转换。 了解更多
  2. MTEP hydrochloride
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    MTEP hydrochloride

    Catalog No. A15174
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    mGlu5 拮抗剂
    MTEP hydrochloride是一种有效的，选择性和非竞争性的mGlu5拮抗剂，IC50和Ki分别为5 nM和16 nM。 了解更多
  3. Dipraglurant
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    Dipraglurant

    Catalog No. A11382
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    mGluR5 antagonists
    Dipraglurant (ADX 48621) is a mGluR5 antagonists with IC50 of 0.021 μM. 了解更多
  4. Mavoglurant
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    Mavoglurant

    Catalog No. A21223
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    mGlu5 receptor antagonist
    Mavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist, has an IC50 of 30 nM in a functional assay with human mGluR5. 了解更多
  5. LY 541850
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    LY 541850

    Catalog No. A21651
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    mGlu2 agonist/mGlu3 antagonist
    LY541850 is a selective orthosteric mGlu2 agonist and mGlu3 antagonist with IC50 values of 0.161 μM and 0.038 μM, respectively. 了解更多
  6. Mavoglurant racemate
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    Mavoglurant racemate

    Catalog No. A21799
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    mGlu5 receptor antagonist
    Mavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. 了解更多
  7. Methoxy-PEPy
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    Methoxy-PEPy

    Catalog No. A21899
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    mGlu5 receptor antagonist
    Methoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM. 了解更多
  8. Auglurant
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    Auglurant

    Catalog No. A20958
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    mGlu5 antagonist
    Auglurant (VU0424238) is a novel and selective mGlu5 antagonist with an IC50 value of 11 nM (rat) and an IC50 value of 14 nM (human). Auglurant (VU0424238) has an acceptable CNS penetration. 了解更多
  9. MPEP
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    MPEP

    Catalog No. A12589
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    mGlu5 receptor 拮抗剂
    MPEP是mGlu5受体亚型（IC50 = 36 nM）的有效且高度选择性的非竞争性拮抗剂，并且是mGlu4受体的正构构调节剂。 了解更多
  10. PHCCC
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    PHCCC

    Catalog No. A12705
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    mGluR 拮抗剂
    PHCCC是I组代谢型谷氨酸受体拮抗剂（IC50?3μM）。 了解更多
  11. SIB 1893
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    SIB 1893

    Catalog No. A13759
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    mGluR 拮抗剂
    SIB 1893是代谢型谷氨酸mGlu5受体亚型的高度选择性非竞争性拮抗剂。 了解更多
  12. SIB 1757
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    SIB 1757

    Catalog No. A13758
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    mGluR 拮抗剂
    SIB 1757是mGlu5代谢型谷氨酸受体亚型的高度选择性拮抗剂。 了解更多
  13. MPEP HCl
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    MPEP HCl

    Catalog No. A13236
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    mGlu5 receptor 拮抗剂
    MPEP HCl是对mGlu5a受体亚型（IC50 = 36 nM）的有效，高度选择性的非竞争性拮抗剂，但在浓度高达30 uM的mGlu1b受体上无激动剂或拮抗剂活性。 了解更多
  14. LY341495
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    LY341495

    Catalog No. A11484
    mGluR-2 拮抗剂
    LY 341495已被证明是一种高效的选择性II类代谢型谷氨酸受体(mGluR-2)拮抗剂，对于人类mGluR-2，mGluR，Ki/IC50值分别为2.3、1.3、173、990、6800、8200和22000 nM。mGluR-3，mGluR-8，mGluR-7a，mGluR-1a，mGluR-5a和mGluR-4a。 了解更多
  15. A-841720
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    A-841720

    Catalog No. A13854
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    mGluR-1 拮抗剂
    841720是一种有效的非竞争性mGluR-1拮抗剂，相对于mGluR-5具有34倍的选择性（IC50值分别为10和342 nM）。 了解更多

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