MLN1117 (Serabelisib)

Name: MLN1117 (Serabelisib)
SKU: A15529

目录号: A15529

p110α 抑制剂

MLN1117 (Serabelisib) Chemical Structure

CAS NO. 1268454-23-4

MLN1117，也称为INK1117和TAK-117，是具有潜在抗肿瘤活性的I类磷酸肌醇3激酶（PI3K）α同工型的生物利用抑制剂。

库存：现货

规格	价格	数量
10 mg	￥ 840.00
25 mg	￥ 1,680.00
50 mg	￥ 2,450.00

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生物活性

MLN1117，也称为INK1117和TAK-117，是具有潜在抗肿瘤活性的I类磷酸肌醇3激酶（PI3K）α同工型的生物利用抑制剂。

溶解度 *

In vitro	DMSO	15 mg/mL (41.28 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	27.54 mL	137.69 mL	275.38 mL
0.5 mM	5.51 mL	27.54 mL	55.08 mL
1 mM	2.75 mL	13.77 mL	27.54 mL
5 mM	0.55 mL	2.75 mL	5.51 mL

*The above data is based on the productmolecular weight 363.13. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15529
作用机制	Inhibitor (抑制剂)
M. Wt	363.13
Formula	C19H17N5O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1268454-23-4
Synonyms	INK1117, INK-1117, INK 1117, MLN 1117, MLN-1117, TAK-117, TAK 117, TAK117
SMILES	O=C(C1=CN=C2C=CC(C3=CC=C(OC(N)=N4)C4=C3)=CN21)N5CCOCC5