主页 /
JAK / Stat /
JAK /
Momelotinib Mesylate

Momelotinib Mesylate

Name: Momelotinib Mesylate
SKU: A21658

目录号: A21658

JAK1/JAK2 inhibitor

Product Citations (1)

Momelotinib Mesylate Chemical Structure

CAS NO. 1056636-07-7

Momelotinib Mesylate (CYT387 Mesylate) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, appr 10-fold selectivity versus JAK3.

库存：现货

规格	价格	数量
1 mg	￥ 2,240.00
5 mg	￥ 6,720.00
10 mg	￥ 11,200.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

Momelotinib Mesylate (CYT387 Mesylate) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, appr 10-fold selectivity versus JAK3.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.59 mL	97.93 mL	195.86 mL
0.5 mM	3.92 mL	19.59 mL	39.17 mL
1 mM	1.96 mL	9.79 mL	19.59 mL
5 mM	0.39 mL	1.96 mL	3.92 mL

*The above data is based on the productmolecular weight 510.57. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A21658
作用机制	Inhibitor (抑制剂)
M. Wt	510.57
Formula	C24H26N6O5S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1056636-07-7
Synonyms	CYT387 (Mesylate), CYT 387, CYT-387
SMILES	O=C(C1=CC=C(C2=NC(NC3=CC=C(N4CCOCC4)C=C3)=NC=C2)C=C1)NCC#N.O=S(O)(C)=O