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Neuronal Signaling

产品 1 到 50 共 86个

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  1. Ticagrelor (AZD6140)
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    Ticagrelor (AZD6140)

    Catalog No. A11238
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    P2Y12 拮抗剂
    Ticagrelor (AZD6140)是第一个可逆结合的口服P2Y（12）受体拮抗剂，可阻断ADP诱导的血小板聚集。 了解更多
  2. MRS 2578
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    MRS 2578

    Catalog No. A11486
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    P2Y6 Receptor 拮抗剂
    MRS 2578是P2Y6核苷酸受体的选择性拮抗剂。 了解更多
  3. AZD1283
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    AZD1283

    Catalog No. A15443
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    P2Y12 receptor 拮抗剂
    AZD1283是P2Y12受体的有效拮抗剂，EC50为3.0 ug/kg/min，TI> 10；结合IC50为11 nM。 了解更多
  4. Prasugrel Hydrochloride
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    Prasugrel Hydrochloride

    Catalog No. A16144
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    P2Y12 拮抗剂
    Prasugrel Hydrochloride是噻吩并吡啶ADP受体（P2Y12）拮抗剂，用于减少血栓性心血管事件。 了解更多
  5. BPTU
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    BPTU

    Catalog No. A16952
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    P2Y1 拮抗剂
    BPTU是P2Y1拮抗剂。已经显示出它具有抗血栓形成的功效并减少了出血的可能性。 了解更多
  6. Elinogrel
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    Elinogrel

    Catalog No. A21468
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    platelet P2Y12 antagonist
    Elinogrel (PRT060128) is a potent, direct acting, competitive, and reversible platelet P2Y12 antagonist (IC50=20 nM). It is orally and intravenously available and has potent antiplatelet effects. 了解更多
  7. A 740003
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    A 740003

    Catalog No. A11316
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    P2X7 receptor 拮抗剂
    A740003是P2X7受体的新型竞争性拮抗剂（人的IC50值= 40 nM，大鼠的IC50值= 18 nM）。 了解更多
  8. NF 279
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    NF 279

    Catalog No. A11972
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    P2X1 拮抗剂
    NF279是一种苏拉明类似物，可作为P2X受体的高选择性，竞争性和可逆性ATP拮抗剂（平滑肌中IC50/KB1μM）。 了解更多
  9. A-317491 sodium salt hydrate
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    A-317491 sodium salt hydrate

    Catalog No. A12412
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    P2X3 and P2X2/3 receptor 拮抗剂
    A-317491 sodium salt hydrate是一种非核苷酸的P2X3和P2X2/3受体拮抗剂，可抑制受体介导的钙通量。 了解更多
  10. A-804598
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    A-804598

    Catalog No. A16066
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    P2X7 receptor 拮抗剂
    A-804598是一种P2X7选择性竞争性拮抗剂，对人，大鼠和小鼠通道的IC50值分别为11、10和9 nM。 了解更多
  11. A-438079 HCl
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    A-438079 HCl

    Catalog No. A12597
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    P2X7 receptor 拮抗剂
    A-438079 HCl是一种竞争性P2X7受体拮抗剂（抑制人重组P2X7细胞系中Ca2+流入的pIC50 = 6.9）。在其他P2受体上没有活性（IC50 > 10 uM）。 了解更多
  12. A 438079 hydrochloride
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    A 438079 hydrochloride

    Catalog No. A14983
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    P2X7 receptor 拮抗剂
    A 438079 hydrochloride是一种竞争性P2X7受体拮抗剂（抑制人重组P2X7细胞系中Ca2+流入的pIC50 = 6.9）。 了解更多
  13. AF-353
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    AF-353

    Catalog No. A13131
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    P2X3/P2X2/3 receptor 拮抗剂
    AF-353是一种新型、有效的P2X3/P2X2/3受体拮抗剂，可抑制人和大鼠的P2X3（pIC50 = 8.0）。 了解更多
  14. JNJ-54175446
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    JNJ-54175446

    Catalog No. A18675
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    P2X7 receptor antagonist
    JNJ-54175446 is a potent and selective brain penetrant P2X7 receptor antagonist, with pIC50s of 8.46 and 8.81 for hP2X7 receptor and rP2X7 receptor, respectively. 了解更多
  15. A 839977
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    A 839977

    Catalog No. A21178
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    P2X7 selective antagonist
    A 839977 is a P2X7 selective antagonist. 了解更多
  16. CE-224535
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    CE-224535

    Catalog No. A21183
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    P2X7 receptor antagonist
    CE-224535 is a selective P2X7 receptor antagonist. 了解更多
  17. Minodronic acid
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    Minodronic acid

    Catalog No. A21975
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    purinergic P2X2/3 receptors antagonist
    Minodronic acid (YM-529) is an antagonist of purinergic P2X2/3 receptors involved in pain. 了解更多
  18. Tropisetron HCL
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    Tropisetron HCL

    Catalog No. A14375
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    5-HT3 receptor 拮抗剂
    Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂，对5-HT3受体的IC50为70.1±0.9 nM。 了解更多
  19. Mecamylamine Hydrochloride
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    Mecamylamine Hydrochloride

    Catalog No. A17884
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    nAChR antagonist
    Mecamylamine hydrochloride is a nAChR antagonist previously used to treat hypertension. It displays a wide variety of activities, including reducing depression-like behaviors in subjects with Tourette's syndrome and improving rates of smoking cessation. 了解更多
  20. Diphenidol HCl
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    Diphenidol HCl

    Catalog No. A14244
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    M2/M3 拮抗剂
    Diphenidol HCl是毒蕈碱M2和M3受体的有效拮抗剂，pKb为6.72和7.02。 了解更多
  21. AF-DX 384
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    AF-DX 384

    Catalog No. A13856
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    mAChR 拮抗剂
    AF-DX 384是充当毒蕈碱乙酰胆碱受体的选择性拮抗剂的药物。 了解更多
  22. PF-3635659
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    PF-3635659

    Catalog No. A13548
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    muscarinic M(3) receptor 拮抗剂
    PF-3635659是有效的毒蕈碱M3受体拮抗剂。 了解更多
  23. Umeclidinium bromide
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    Umeclidinium bromide

    Catalog No. A15268
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    Muscarinic receptor 拮抗剂
    Umeclidinium bromide (GSK573719A)是毒蕈碱受体拮抗剂，可用于治疗慢性阻塞性肺疾病（COPD）。 了解更多
  24. Revefenacin
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    Revefenacin

    Catalog No. A15986
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    muscarinic receptor 拮抗剂
    Revefenacin是正在研发中的有效，选择性毒蕈碱受体拮抗剂，可用于治疗COPD。 了解更多
  25. Glycopyrrolate
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    Glycopyrrolate

    Catalog No. A12641
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    muscarinic 拮抗剂
    Glycopyrrolate是一种毒蕈碱竞争性拮抗剂，可用作解痉挛药。 了解更多
  26. Flavoxate
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    Flavoxate

    Catalog No. A12900
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    muscarinic AChR antagonist
    Flavoxate结合并抑制毒蕈碱受体，从而通过改变脑干的排尿中心来抑制排尿反射并增加膀胱容量。 了解更多
  27. Atropine methyl bromide
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    Atropine methyl bromide

    Catalog No. A18026
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    mAChR antagonist
    Atropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and a mydriatic for dilation of the pupil during ophthalmic examination. It is introduced for relieving pyloric spasm in infants for its highly polar nature. It penetrates less readily into the central nervous system than atropine. 了解更多
  28. Cimetropium Bromide
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    Cimetropium Bromide

    Catalog No. A18290
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    mAChR antagonist
    Cimetropium Bromide (DA-3177) is a mAChR antagonist for long-term treatment of irritable bowel syndrome. 了解更多
  29. Tiotropium Bromide
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    Tiotropium Bromide

    Catalog No. A10934
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    muscarinic acetylcholine receptor (mAChR) antagonist
    Tiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多
  30. mAChR-IN-1 hydrochloride
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    mAChR-IN-1 hydrochloride

    Catalog No. A21398
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    mAChR antagonist
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多
  31. mAChR-IN-1
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    mAChR-IN-1

    Catalog No. A21518
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    mAChR antagonist
    mAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. 了解更多
  32. Fesoterodine fumarate (Toviaz)
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    Fesoterodine fumarate (Toviaz)

    Catalog No. A10386
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    AChR 拮抗剂
    Fesoterodine fumarate是一种用于尿急的药物，可减少尿液通过的频率并促使尿失禁。 了解更多
  33. 5-hydroxymethyl tolterodine (PNU 200577)
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    5-hydroxymethyl tolterodine (PNU 200577)

    Catalog No. A11166
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    muscarinic receptor 拮抗剂
    5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多
  34. Rocuronium bromide
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    Rocuronium bromide

    Catalog No. A10803
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    AchR 拮抗剂
    Rocuronium Bromide是一种竞争性AchR拮抗剂，用于现代麻醉中。 了解更多
  35. Biperiden HCl
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    Biperiden HCl

    Catalog No. A10147
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    Muscarinic receptor antagonist
    Biperiden HCl是毒蕈碱受体拮抗剂，对M1亚型表现出一定的选择性。 了解更多
  36. Tolterodine tartrate (Detrol LA)
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    Tolterodine tartrate (Detrol LA)

    Catalog No. A10937
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    muscarinic receptor 拮抗剂
    Tolterodine tartrate (Detrol LA)是毒蕈碱受体拮抗剂。 了解更多
  37. Solifenacin succinate
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    Solifenacin succinate

    Catalog No. A11215
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    muscarinic M3 receptor antagoinst
    Solifenacin succinate是毒蕈碱M3受体拮抗剂，用于治疗尿失禁。 了解更多
  38. Atropine
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    Atropine

    Catalog No. A10098
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    mAChR 拮抗剂
    Atropine是M1，M2，M3，M4和M5型毒蕈碱乙酰胆碱受体的竞争性拮抗剂。 了解更多
  39. SVT-40776 (Tarafenacin)
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    SVT-40776 (Tarafenacin)

    Catalog No. A10808
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    muscarinic receptor 拮抗剂
    SVT-40776 (Tarafenacin)是新型M3毒蕈碱受体拮抗剂，用于治疗膀胱过度活动症。 了解更多
  40. Gallamine triethiodide
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    Gallamine triethiodide

    Catalog No. A10417
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    mAChR M2 拮抗剂
    Gallamine Triethiodide是一种具有显著心脏选择性的mAChR M2拮抗剂。 了解更多
  41. Ipratropium bromide
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    Ipratropium bromide

    Catalog No. A10476
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    Ipratropium bromide是毒蕈碱拮抗剂、支气管扩张剂、阿托品的N-异丙基盐。 了解更多
  42. Phenoxybenzamine hydrochloride
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    Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多
  43. Memantine hydrochloride
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    Memantine hydrochloride

    Catalog No. A11708
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    NMDA receptor 拮抗剂
    Memantine hydrochloride是nmda受体的拮抗剂，与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂，作用于重组CYP2B6和CYP2D6，Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。 了解更多
  44. Orphenadrine citrate
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    Orphenadrine citrate

    Catalog No. A11712
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    NMDA receptor 拮抗剂
    Orphenadrine柠檬酸盐是NMDA受体拮抗剂，Ki为6.0μM，还是HERG钾离子通道阻断剂。 了解更多
  45. Felbamate
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    Felbamate

    Catalog No. A11862
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    Felbamate是NMDA相关甘氨酸结合位点的拮抗剂。 了解更多
  46. MDL 29951
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    MDL 29951

    Catalog No. A13729
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    NMDA receptor 拮抗剂
    MDL-29951是在体外和体内均能激活NMDA受体的新型甘氨酸拮抗剂（Ki = 0.14 mM，[3H]甘氨酸结合）。 了解更多
  47. NVP-AAM077 Tetrasodium Hydrate (PEAQX)
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    NVP-AAM077 Tetrasodium Hydrate (PEAQX)

    Catalog No. A14071
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    NMDA receptors 拮抗剂
    NVP-AAM077抑制成年小鼠在脑室下区域和齿状回中的祖细胞增殖，并降低了齿状回中的新生细胞的存活。 了解更多
  48. ARL-15896
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    ARL-15896

    Catalog No. A13858
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    NMDA receptor ion channel 拮抗剂
    ARL-15896是新型的N-甲基-D-天冬氨酸受体离子通道拮抗剂。 了解更多
  49. CNQX
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    CNQX

    Catalog No. A16109
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    AMPA/kainate 拮抗剂
    CNQX是一种竞争性的非NMDA谷氨酸受体拮抗剂（AMPA和海藻酸酯受体的IC50分别为0.3和1.5 uM，而NMDA受体的IC50 = 25 uM）。 了解更多
  50. 7CKA
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    7CKA

    Catalog No. A17070
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    NMDA receptor 拮抗剂
    7CKA是在甘氨酸位点起作用的NMDA受体拮抗剂。 了解更多

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