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￥ 0.00 Neuronal Signaling
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EVP-6124 hydrochloride
Catalog No. A15087 nAChR 抑制剂EVP-6124 hydrochloride是一种新型的α7神经元烟碱型乙酰胆碱受体（nAChRs）的部分激动剂。EVP-6124对α7nAChRs具有选择性，并且不激活或抑制异源α4β2nAChRs。 了解更多 -
GTS-21 (DMBX-A)
Catalog No. A15950 nAChR 激动剂GTS-21 dihydrochloride (DMBX-A)是一种选择性的α7烟碱乙酰胆碱受体激动剂，最近已被确定为一种有希望的炎症治疗方法。 了解更多 -
Benzethonium Chloride
Catalog No. A13653 nAChR 抑制剂Benzethonium Chloride是nAChRs的有效抑制剂，可抑制α4β2nAChRs和α7nAChRs，IC50分别为49 nM和122 nM。 了解更多 -
Mecamylamine Hydrochloride
Catalog No. A17884 nAChR antagonistMecamylamine hydrochloride is a nAChR antagonist previously used to treat hypertension. It displays a wide variety of activities, including reducing depression-like behaviors in subjects with Tourette's syndrome and improving rates of smoking cessation. 了解更多 -
(-)-(S)-B-973B
Catalog No. A18761 α7 nAChR modulator-)-(S)-B-973B is a potent allosteric agonist and positive allosteric modulator of α7 nAChR, with antinociceptive activity. 了解更多 -
Catharanthine sulfate
Catalog No. A12161 Catharanthine sulfate是长春碱型生物碱前体，具有抗肿瘤活性。它通过离子通道阻断和脱敏来抑制AChR。 了解更多 -
Diphenidol HCl
Catalog No. A14244 -
Xanomeline oxalate
Catalog No. A13685 mAChR 激动剂Xanomeline oxalate是毒蕈碱型乙酰胆碱受体的有效激动剂（M1，M2，M3，M4和M5的EC50值分别为0.3、92.5、5、52和42 nM）。 了解更多 -
PF-3635659
Catalog No. A13548 -
Cevimeline hydrochloride hemihydrate
Catalog No. A15042 -
Umeclidinium bromide
Catalog No. A15268 Muscarinic receptor 拮抗剂Umeclidinium bromide (GSK573719A)是毒蕈碱受体拮抗剂，可用于治疗慢性阻塞性肺疾病（COPD）。 了解更多 -
Imidafenacin
Catalog No. A15490 M3 receptors 抑制剂Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。 了解更多 -
TBPB
Catalog No. A14205 -
Revefenacin
Catalog No. A15986 -
Glycopyrrolate
Catalog No. A12641 -
Flavoxate
Catalog No. A12900 -
Acetylcholine iodide
Catalog No. A16390 Acetylcholine iodide是一种神经递质，存在于神经肌肉接头，植物神经节，副交感神经效应接头，交感神经效应接头的子集以及中枢神经系统的许多部位。 了解更多 -
Atropine methyl bromide
Catalog No. A18026 mAChR antagonistAtropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and a mydriatic for dilation of the pupil during ophthalmic examination. It is introduced for relieving pyloric spasm in infants for its highly polar nature. It penetrates less readily into the central nervous system than atropine. 了解更多 -
Cevimeline hydrochloride
Catalog No. A18092 mAChR agonistCevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多 -
Anisodamine
Catalog No. A18215 alpha-1 adrenergic receptors / mAChRs inhibitorAnisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多 -
Cimetropium Bromide
Catalog No. A18290 mAChR antagonistCimetropium Bromide (DA-3177) is a mAChR antagonist for long-term treatment of irritable bowel syndrome. 了解更多 -
Darenzepine
Catalog No. A12333 muscarinic receptor inhibitorDarenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多 -
Tiotropium Bromide
Catalog No. A10934 muscarinic acetylcholine receptor (mAChR) antagonistTiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多 -
Rapacuronium bromide
Catalog No. A21119 mAChR modulatorRapacuronium bromide is an allosteric modulator of muscarinic acetylcholine receptor (mAChR). 了解更多 -
mAChR-IN-1 hydrochloride
Catalog No. A21398 mAChR antagonistmAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多 -
mAChR-IN-1
Catalog No. A21518 mAChR antagonistmAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. 了解更多 -
(Rac)-VU 6008667
Catalog No. A21939 mAChR M5 negative allosteric modulator(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration. 了解更多 -
Oxotremorine M iodide
Catalog No. A21977 mAChR agonistOxotremorine M iodide is a potent and non-selective muscarinic acetylcholine receptor (mAChR) agonist. 了解更多 -
Fesoterodine fumarate (Toviaz)
Catalog No. A10386 -
5-hydroxymethyl tolterodine (PNU 200577)
Catalog No. A11166 muscarinic receptor 拮抗剂5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多 -
Rocuronium bromide
Catalog No. A10803 -
Biperiden HCl
Catalog No. A10147 -
Tolterodine tartrate (Detrol LA)
Catalog No. A10937 -
Solifenacin succinate
Catalog No. A11215 muscarinic M3 receptor antagoinstSolifenacin succinate是毒蕈碱M3受体拮抗剂，用于治疗尿失禁。 了解更多 -
SVT-40776 (Tarafenacin)
Catalog No. A10808 -
Bethanechol chloride
Catalog No. A10180 Muscarinic receptor 激动剂Bethanechol chloride是拟副交感神经的胆碱氨基甲酸酯，可选择性刺激毒蕈碱受体，而不会对烟碱样受体产生任何影响。 了解更多 -
Gallamine triethiodide
Catalog No. A10417 -
Methscopolamine bromide
Catalog No. A10579 Methscopolamine bromide是一种竞争性抗毒蕈碱剂，可阻断乙酰胆碱与毒蕈碱型乙酰胆碱受体（mAChR M）的结合。 了解更多
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