Neuronal Signaling
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CIQ
Catalog No. A15523 -
RO 25-6981 maleate
Catalog No. A16083 NMDA receptors blockerRO 25-6981 maleate是含有NR2B亚基的NMDA受体的强效和选择性活性依赖性阻断剂。克隆的受体亚基组合NR1C/NR2B和NR1C/NR2A的IC50值分别为0.009和52 uM。 了解更多 -
Ro 25-6981 maleate
Catalog No. A13144 -
D-AP5
Catalog No. A17044 -
Mephenesin
Catalog No. A17493 NMDA receptor antagonistMephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. 了解更多 -
Flupirtine maleate
Catalog No. A10251 NMDA 拮抗剂Flupirtine maleate是Flupirine的盐形式,是一种非阿片类中枢性镇痛药,是一种选择性的神经元钾离子通道开放剂,也具有NMDA受体拮抗剂特性。 了解更多 -
TCN 201
Catalog No. A11947 -
SDZ 220-581
Catalog No. A12426 -
(-)-MK 801 maleate
Catalog No. A13435 NMDA receptor 拮抗剂.(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。 了解更多 -
SDZ 220-581 Ammonium salt
Catalog No. A15235 -
L-701324
Catalog No. A15522 -
(+)-MK 801 Maleate
Catalog No. A12761 -
GV-196771A
Catalog No. A13438 NMDA receptor antagonistGV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多 -
Ifenprodil tartrate
Catalog No. A16583 NMDA receptor antagonistIfenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多 -
Transcrocetinate disodium
Catalog No. A21051 NMDA receptor antagonistTranscrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多 -
MDL 105519
Catalog No. A21192 NMDA receptor antagonistMDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多 -
Radiprodil
Catalog No. A21193 NMDA NR2B antagonistRadiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. 了解更多 -
7-Chlorokynurenic acid sodium salt
Catalog No. A21879 NMDA receptor antagonist7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多 -
SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
Catalog No. A21897 NMDA receptor antagonistSDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多 -
Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多 -
Dihydromyricetin (Ampeloptin)
Catalog No. A10252 -
Nefiracetam (Translon)
Catalog No. A10631 Nefiracetam (Translon)是认知增强剂。它激活L/N型钙通道,胆碱能,单胺能和GABA能系统。 了解更多 -
SKF 89976A HCl
Catalog No. A10849 GABA uptake 抑制剂SKF 89976A HCl是一种有效的GABA吸收抑制剂,hGAT-1,rGAT-2,hGAT-3和hBGT-1的IC50分别为0.13、550、944和7210μM。 了解更多 -
Flumazenil
Catalog No. A10397 Benzodiazepine 拮抗剂Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂,但在人类中很少或没有激动剂活性。 了解更多 -
Furosemide
Catalog No. A10412 Furosemide是GABAA受体的非竞争性拮抗剂,对含α6受体的选择性比含α1受体高约100倍。 了解更多 -
(+)-Bicuculline
Catalog No. A12590 -
AWD 131-138
Catalog No. A13726 -
2-Hydroxysaclofen
Catalog No. A13696 -
Cloflubicyne
Catalog No. A13932 -
a5IA
Catalog No. A14343