微信关注
Total item
Cart Subtotal
￥ 0.00 Opioid Receptors
15 个项目
每页
-
Trimebutine maleate
Catalog No. A18115 ?- opioid receptor agonistTrimebutine Maleate is a drug with antimuscarinic and weak mu opioid agonist effects. Trimebutine Maleate modulates the calcium and potassium channels, relieves abdominal pain in patients with irritable bowel syndrome. 了解更多 -
Cebranopadol (GRT-6005)
Catalog No. A12670 Opioid Receptor 激动剂Cebranopadol是一种有效的伤害感受器/孤儿蛋白FQ肽（NOP）和阿片受体激动剂。作用于人NOP，MOP，KOP 和δ-阿片肽(DOP)受体，Ki/EC50 分别为 0.9 nM/13 nM，0.7 nM/1.2 nM，2.6 nM/17 nM，18 nM/110 nM。 了解更多 -
Alvimopan monohydrate
Catalog No. A14992 ?-opioid receptor 激动剂Alvimopan monohydrate是一种外围作用的类阿片受体（PAM-OR，IC50 = 1.7 nM）拮抗剂，可促进术后肠胃的恢复。 了解更多 -
Alvimopan dihydrate
Catalog No. A14991 ?-opioid receptor 激动剂Alvimopan dihydrate (LY 246736,ADL 8-2698)是一种外周作用的类阿片受体（PAM-OR，IC50 = 1.7 nM）拮抗剂，可促进术后胃肠道恢复。 了解更多 -
ADL5859 HCl
Catalog No. A11072 Opioid Receptor 激动剂ADL5859 HCl是高效的选择性δ阿片受体激动剂，Ki值为0.84 nM，ED50值为20 nM。 了解更多 -
MCOPPB 3HCl
Catalog No. A10561 -
BRL 52537 HCl
Catalog No. A11210 Opioid Receptors 激动剂BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂（Ki = 0.24 nM）。比吗啡强25倍。 了解更多 -
Nalfurafine hydrochloride
Catalog No. A12579 opioid κ-selective 激动剂Nalfurafine hydrochloride是一种κ-opioid激动剂。 了解更多 -
Nalmefene hydrochloride
Catalog No. A13843 dopamine receptor 激动剂Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多 -
U-69593
Catalog No. A14187 -
TRV130 HCl (Oliceridine)
Catalog No. A15444 u-opioid receptor 激动剂TRV130 HCl (Oliceridine)是一种新型的μ-opioid 受体（MOR）G蛋白偏向配体。诱导强大的G蛋白信号传导（pEC50 = 8.1），效力和功效与吗啡相似，但β-arrestin募集和受体内在化作用要低得多。 了解更多 -
CYT-1010 hydrochloride
Catalog No. A21348 mu-opioid receptor agonistCYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多 -
AR-M 1000390 hydrochloride
Catalog No. A21911 δ opioid receptor agonistAR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多
15 个项目
每页