Opioid Receptors

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BTRX-335140

Catalog No. A18583
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κ opioid receptor antagonist

BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. 了解更多

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Naloxegol Oxalate

Catalog No. A15972
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Opioid 拮抗剂

Naloxegol Oxalate是用于治疗阿片类药物引起的便秘的外周选择性阿片类药物拮抗剂。了解更多

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JTC-801

Catalog No. A11076
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Opioid Receptor 拮抗剂

JTC-801是nociceptin receptor（也称为ORL-1受体）的选择性拮抗剂。了解更多

Product Citations (2)

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- Lihao Gu, .et al. 10-Hydroxy-2-Decenoic Acid in Royal Jelly Extract Induced Both Filaggrin and Amino Acid in a Cultured Human Three-Dimensional Epidermis Model, Cosmetics, 2017, 4(4), 48
- Toshio Yawata, .et al. Brain opioid and nociceptin receptors are involved in regulation of bombesin-induced activation of central sympatho-adrenomedullary outflow in the rat, Mol Cell Biochem, 2016, Jan;411(1-2):201-11 PMID: 26427671
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Alvimopan (ADL 8-2698)

Catalog No. A11292
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Opioid 拮抗剂

Alvimopan (ADL 8-2698)表现为外周作用的opioid拮抗剂，Alvimopan竞争性结合胃肠道中的mu-opioid receptor。了解更多

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BAN ORL 24

Catalog No. A11322
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NOP 拮抗剂

BAN ORL 24是一种强效选择性NOP受体拮抗剂。了解更多

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Methylnaltrexone Bromide

Catalog No. A15159
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μ-opioid 拮抗剂

Methylnaltrexone Bromide是一种作用于胃肠道以减少阿片类药物引起的便秘的具有信息素作用的?-opioid拮抗剂。了解更多

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LY2795050

Catalog No. A15149
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k-opioid receptor 拮抗剂

LY2795050是新型选择性κ阿片受体（KOR）拮抗剂（IC50 = 0.72 nM），具有作为PET示踪剂在体内对KOR成像的潜力。了解更多

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GSK1521498 free base

Catalog No. A18994
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μ-opioid receptor antagonist

GSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多

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JDTic

Catalog No. A11468
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κ-opioid receptor antagonist

JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. 了解更多

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GSK1521498 free base (hydrochloride)

Catalog No. A21792
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μ-opioid receptor (MOR) antagonist

GSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多

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