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ORY-1001 (RG-6016)

ORY-1001 (RG-6016)

Name: ORY-1001 (RG-6016)
SKU: A15893

目录号: A15893

LSD1 抑制剂

ORY-1001 (RG-6016) Chemical Structure

CAS NO. 1431326-61-2

ORY-1001 (RG-6016)是一种活性的选择性赖氨酸脱甲基酶LSD1/KDM1A抑制剂，IC50 <20 nM，对相关FAD依赖性氨氧化酶具有高选择性。

库存：现货

规格	价格	数量
5 mg	￥ 882.00
10 mg	￥ 1,498.00
25 mg	￥ 2,646.00

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生物活性

ORY-1001 (RG-6016)是一种活性的选择性赖氨酸脱甲基酶LSD1/KDM1A抑制剂，IC50 <20 nM，对相关FAD依赖性氨氧化酶具有高选择性。

靶点信息

LSD1/KDM1A
20 nM

溶解度 *

In vitro	DMSO	4 mg/mL (13.18 mM)
	Water	53 mg/mL (174.76 mM)
	Ethanol	Warmed: 3 mg/mL (9.89 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	32.97 mL	164.87 mL	329.74 mL
0.5 mM	6.59 mL	32.97 mL	65.95 mL
1 mM	3.3 mL	16.49 mL	32.97 mL
5 mM	0.66 mL	3.3 mL	6.59 mL

*The above data is based on the productmolecular weight 303.27. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15893
作用机制	Inhibitor (抑制剂)
M. Wt	303.27
Formula	C15H22N2.2HCl
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1431326-61-2
Synonyms	RG6016, RG-6016
SMILES	NC1CCC(N[C@@H]2C[C@H]2C3=CC=CC=C3)CC1.Cl.Cl