PD318088 | MEK 抑制剂 | 美国进口 | PD318088 供应商 AdooQ®

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PD318088

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产品详情

生物活性

PD318088是MEK1和MEK2的抑制剂。

靶点信息

MEK1/2

溶解度 *

In vitro	DMSO	105 mg/mL (187.13 mM)
	Water	Insoluble
	Ethanol	13 mg/mL (23.17 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.82 mL	89.11 mL	178.22 mL
0.5 mM	3.56 mL	17.82 mL	35.64 mL
1 mM	1.78 mL	8.91 mL	17.82 mL
5 mM	0.36 mL	1.78 mL	3.56 mL

*The above data is based on the productmolecular weight 561.1 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10704
作用机制	Inhibitor (抑制剂)
M. Wt	561.1
Formula	C16H13BrF3IN2O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	391210-00-7
Synonyms	PD-318088
SMILES	C1=CC(=C(C=C1I)F)NC2=C(C(=C(C=C2C(=O)NOCC(CO)O)Br)F)F

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产品资料

Download PD318088 SD file

Products Specification Data Sheet

Safety Data Sheet (SDS)

产品标签

产品标签

其他人对该产品使用了下列标签：

MEK2 (7)
MEK1 (14)

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