产品详情
PDGFRα kinase inhibitor 1 is a highly selective type II PDGFRα kinase inhibitor with IC50s of 132 nM and 6115 nM for PDGFRα and PDGFRβ, respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 17.04 mL | 85.22 mL | 170.45 mL |
0.5 mM | 3.41 mL | 17.04 mL | 34.09 mL |
1 mM | 1.7 mL | 8.52 mL | 17.04 mL |
5 mM | 0.34 mL | 1.7 mL | 3.41 mL |
*The above data is based on the productmolecular weight 586.69. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
目录号 | A19632 |
---|---|
M. Wt | 586.69 |
Formula | C34H34N8O2 |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. |
CAS No. | 2209053-93-8 |
SMILES | CC(C=CC(NC(C1=CC=C(CN(CCN(C)C)C(C2=CC=CN=C2)=O)C=C1)=O)=C3)=C3NC4=NC=CC(C5=CC=CN=C5)=N4 |
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