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47 个项目
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Chiglitazar
Catalog No. A12701 PPARα/γ dual agonistChiglitazar is a PPARα/γ dual agonist, with EC50s of 1.2, 0.08, 1.7 μM for PPARα, PPARγ and PPARδ, respectively. 了解更多 -
Leriglitazone
Catalog No. A18636 PPAR gamma agonistLeriglitazone is a peroxisome proliferator activated receptor (PPAR) gamma agonist. 了解更多 -
MA-0204
Catalog No. A19031 PPARδ modulatorMA-0204 is a potent, highly selective and orally available peroxisome proliferator activated receptor δ (PPARδ) modulator with EC50s of 0.4 nM, 7.9 nM and 10 nM for human, mouse and rat PPARδ, respectively. Potential treatment for Duchene Muscular Dystrophy (DMD). 了解更多 -
NXT629
Catalog No. A18771 PPAR-α antagonistNXT629 is a potent, selective, and competitive PPAR-α antagonist, with an IC50 of 77 nM for human PPARα, shows high selectivity over other nuclear hormone receptor, such as PPARδ, PPARγ, ERβ, GR and TRβ, IC50s are 6.0, 15, 15.2, 32.5 and >100 μM, respectively. 了解更多 -
Etofylline
Catalog No. A17491 PPAR agonistEtofylline, also known as BRN-0251760, is a peroxisome proliferator-activated receptor (PPAR) agonist used to treat respiratory and cardiovascular disorders. Etofylline is often used as a bronchodilator. 了解更多 -
Inolitazone dihydrochloride
Catalog No. A15129 PPARγ 激动剂Inolitazone dihydrochloride是一种新型的高亲和力PPARγ激动剂，可激活PPARγ，其EC50约为罗格列酮的EC50，对RIE细胞无影响。 了解更多 -
Choline Fenofibrate
Catalog No. A15044 -
Rosiglitazone maleate
Catalog No. A10809 -
Pioglitazone (Actos)
Catalog No. A11680 PPARγ 激动剂Pioglitazone (Actos)是选择性刺激核受体过氧化物酶体增殖物激活的受体γ（PPAR-γ），并在较小程度上刺激PPAR-α。 了解更多 -
Rosiglitazone (BRL-49653)
Catalog No. A10807 PPAR 激动剂Rosiglitazone (BRL-49653)是有效的降糖药，也是有效的噻唑烷二酮类胰岛素增敏剂，在大鼠，3T3-L1和人体脂肪细胞中IC50分别为12，4和9 nM。Rosiglitazone是PPAR-gamma的配体，对PPAR-alpha没有结合力。 了解更多 -
Troglitazone
Catalog No. A11981 PPARγ 激动剂Troglitazone是一种选择性PPARγ受体激动剂（鼠和人PPARγ受体的EC50值分别为780和555 nM）。 了解更多 -
pirinixic acid (WY 14643)
Catalog No. A12360 -
GSK-3787
Catalog No. A12391 -
GW6471
Catalog No. A12413 -
Tesaglitazar
Catalog No. A20891 PPAR alpha/gamma agonistTesaglitazar is a dual peroxisome proliferator-activated receptor (PPAR) alpha/gamma agonist that is more potent on PPARγ than on PPARα, with EC50s of 13.4 μM and 3.6 μM for rat PPARα and human PPARα, respectively. 了解更多 -
Fonadelpar
Catalog No. A20848 PPARδ agonistFonadelpar is a PPARδ agonist, used in the research of neuroparalytic keratopathy. 了解更多 -
Arhalofenate
Catalog No. A21135 PPARγ agonistArhalofenate (MBX 102) is a selective partial agonist of peroxisome proliferator-activated receptor (PPAR)-γ, used for the treatment of type 2 diabetes. 了解更多 -
Pioglitazone hydrochloride
Catalog No. A16670 PPARγ agonistPioglitazone hydrochloride is a potent and selective PPARγ agonist with EC50s of 0.93 and 0.99 μM for human and mouse PPARγ, respectively. 了解更多 -
5-Aminosalicylic Acid
Catalog No. A10570 PPARγ agonist5-Aminosalicylic acid (Mesalamine) acts as a specific PPARγ agonist and also inhibits p21-activated kinase 1 (PAK1) and NF-κB. 了解更多 -
Indeglitazar
Catalog No. A21148 PPAR agonistIndeglitazar is an orally available peroxisome proliferator-activated receptor (PPAR) pan-agonist for all three PPAR subtypes alpha (α), delta (δ) and gamma (γ). 了解更多 -
Inolitazone
Catalog No. A21180 PPARγ agonistInolitazone a novel high-affinity PPARγ agonist that is dependent upon PPARγ for its biological activity with IC50 of 0.8 nM for growth inhibition. 了解更多 -
Peliglitazar racemate
Catalog No. A21411 dual α/γ PPAR activatorPeliglitazar racemate is the racemate of Peliglitazar. Peliglitazar is a novel dual α/γ PPAR activator. 了解更多 -
DG172 dihydrochloride
Catalog No. A16309 PPARβ/δ inverse 激动剂DG-172是一种口服活性强效PPARβ/δ反向激动剂 (IC50 = 26.9 nM)。DG-172在体外抑制小鼠成肌细胞中Angptl4基因的表达 (IC50 = 9.5 nM)。 了解更多 -
CDDO-Im
Catalog No. A16308 -
Elafibranor
Catalog No. A15454 PPAR 激动剂Elafibranor是过氧化物酶体增殖物激活的受体-α和-δ的激动剂，可诱导非酒精性脂肪性肝炎消退，而不会使纤维化恶化。 了解更多 -
Aleglitazar
Catalog No. A12492 -
T0070907
Catalog No. A11588 -
BMS-687453
Catalog No. A15836 PPAR 激动剂BMS-687453是一种有效的选择性过氧化物酶体增殖物激活受体（PPAR）α激动剂，对人PPARα的EC（50）为10 nM，在PPAR-GAL4反式激活试验中，选择性是对人PPARgamma的410倍。 了解更多 -
Balaglitazone
Catalog No. A15013 -
GW1929
Catalog No. A15099
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