Prostanoid Receptors

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  1. Grapiprant (CJ-023423)

    Catalog No. A15964
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    prostaglandin EP4 receptor 拮抗剂
    Grapiprant (CJ-023423)是一种具有抗痛觉过敏特性的新型,有效且选择性的前列腺素EP4受体拮抗剂。 了解更多
  2. TG6-10-1

    Catalog No. A15968
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    Prostaglandin E2 receptor 拮抗剂
    TG6-10-1是前列腺素E2受体亚型EP2的有效和选择性拮抗剂。 了解更多
  3. PF-04418948

    Catalog No. A12894
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    EP2 Receptor 拮抗剂
    PF-04418948是一种有效的选择性前列腺素EP2受体拮抗剂,IC50为16 nM。 了解更多
  4. MF498

    Catalog No. A15532
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    EP4 receptor 拮抗剂
    MF498是一种新型的选择性E前列腺素类受体4(EP4受体)拮抗剂,对EP4受体具有很强的结合亲和力,Ki为0.7 nM。 了解更多
  5. GW627368

    Catalog No. A15525
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    EP4 receptor 拮抗剂
    GW627368是一种新型,有效且选择性的前列腺素EP4受体竞争拮抗剂(Ki = 100 nM),具有额外的人TP受体亲和力(Ki = 150 nM)。 了解更多
  6. BAY-u 3405

    Catalog No. A13751
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    dual 拮抗剂 of TP/DP2
    BAY-u 3405是用于治疗变应性鼻炎的经过批准的人用药物,已证明其具有作为血栓烷受体(TP受体)的拮抗剂的活性。 了解更多
  7. MK-2894

    Catalog No. A11497
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    EP4 receptor 拮抗剂
    MK-2894是一种高度有效和选择性的第二代EP4拮抗剂。 了解更多
  8. CJ-42794

    Catalog No. A21948
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    EP4 antagonist
    CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多
  9. Terutroban

    Catalog No. A20884
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    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多
  10. MK-2894 sodium salt

    Catalog No. A11498
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    EP4 antagonist
    MK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. 了解更多
  11. ONO-AE3-208

    Catalog No. A11516
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    EP4 antagonist
    ONO-AE3-208 is an EP4 antagonist, and suppresses cell invasion, migration, and metastasis of prostate cancer. 了解更多
  12. CAY10471 Racemate

    Catalog No. A11760
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    Prostaglandin D2 receptor CRTH2 antagonist
    CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多
  13. Aligeron

    Catalog No. A13241
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    prostaglandin (PG) antagonist
    Aligeron is a non-selective prostaglandin (PG) antagonist, and has vasodilatory properties. 了解更多
  14. GSK-269984A

    Catalog No. A17096
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    EP1 receptor 拮抗剂
    GSK-269984A是新型的EP1受体拮抗剂。pIC50 值为 7.9。 了解更多

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